JP2018506503A5 - - Google Patents
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- JP2018506503A5 JP2018506503A5 JP2017502582A JP2017502582A JP2018506503A5 JP 2018506503 A5 JP2018506503 A5 JP 2018506503A5 JP 2017502582 A JP2017502582 A JP 2017502582A JP 2017502582 A JP2017502582 A JP 2017502582A JP 2018506503 A5 JP2018506503 A5 JP 2018506503A5
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- JP
- Japan
- Prior art keywords
- group
- compound
- acid
- salt
- stereoisomer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR1020150024334A KR20160101554A (ko) | 2015-02-17 | 2015-02-17 | N-[4-(1-아미노에틸)-페닐]-메탄술폰아미드 유도체의 카이랄 분할 방법 |
| KR10-2015-0024334 | 2015-02-17 | ||
| EP15174617.9 | 2015-06-30 | ||
| EP15174617 | 2015-06-30 | ||
| PCT/KR2016/001474 WO2016133317A1 (ko) | 2015-02-17 | 2016-02-15 | Ｎ-[4-(1-아미노에틸)-페닐]-술폰아미드 유도체의 카이랄 분할 방법 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2018506503A JP2018506503A (ja) | 2018-03-08 |
| JP2018506503A5 true JP2018506503A5 (https=) | 2019-01-31 |
| JP6687596B2 JP6687596B2 (ja) | 2020-04-22 |
Family
ID=56692658
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017502582A Active JP6687596B2 (ja) | 2015-02-17 | 2016-02-15 | Ｎ−［４−（１−アミノエチル）−フェニル］−スルホンアミド誘導体のキラル分割方法 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US10479763B2 (https=) |
| EP (1) | EP3162793B1 (https=) |
| JP (1) | JP6687596B2 (https=) |
| KR (1) | KR101791119B1 (https=) |
| CN (1) | CN106660949B (https=) |
| BR (1) | BR112017001516B1 (https=) |
| TW (1) | TWI687396B (https=) |
| WO (1) | WO2016133317A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102565407B1 (ko) * | 2016-01-04 | 2023-08-10 | (주)아모레퍼시픽 | 극성 비양자성 용매를 이용한 n-[4-(1-아미노에틸)-페닐]-술폰아미드 유도체의 카이랄 분할 방법 |
| KR102599958B1 (ko) | 2016-09-28 | 2023-11-09 | (주)아모레퍼시픽 | (r)-n-[4-(1-아미노-에틸)-2,6-다이플루오로-페닐]-메테인설폰아마이드의 제조방법 |
| KR102587339B1 (ko) * | 2016-12-22 | 2023-10-12 | (주)아모레퍼시픽 | N-[4-(1-아미노-에틸)-2,6-다이플루오로-페닐]-메테인설폰아마이드의 거울상 이성질체들의 라세미화 방법 |
| CN109608368B (zh) * | 2018-10-24 | 2021-03-09 | 常州市阳光药业有限公司 | N-[4-(1-氨基乙基)-2,6-二氟苯基]甲磺酰胺的合成及拆分方法 |
| KR20200053746A (ko) | 2018-11-09 | 2020-05-19 | (주)아모레퍼시픽 | 졸-겔 조성물 |
| CN115103836A (zh) * | 2020-02-16 | 2022-09-23 | 艾雅拉制药公司 | 制备手性苯并二氮杂卓酮衍生物的方法 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS60152425A (ja) * | 1984-01-20 | 1985-08-10 | Oyo Seikagaku Kenkyusho:Kk | ラセミ体の新規な光学分割法 |
| US4968837A (en) | 1989-07-28 | 1990-11-06 | Ethyl Corporation | Resolution of racemic mixtures |
| EP0418770B1 (en) * | 1989-09-19 | 1995-07-19 | Hoechst-Roussel Pharmaceuticals Incorporated | Process for the chemical resolution of 5-alkoxy-substituted (+/-)-1,3-dimethyloxindolylethylamines |
| US6265615B1 (en) | 1998-07-01 | 2001-07-24 | The Regents Of The University Of California | Chiral recognition polymer and its use to separate enantiomers |
| DE19956786A1 (de) * | 1999-11-25 | 2001-05-31 | Basf Ag | Verfahren zur Herstellung optisch aktiver Amine |
| US7301023B2 (en) * | 2001-05-31 | 2007-11-27 | Pfizer Inc. | Chiral salt resolution |
| EA200701745A1 (ru) | 2005-03-17 | 2008-06-30 | Пфайзер, Инк. | Циклопропанкарбоксамидные производные |
| US20120041225A1 (en) * | 2006-02-03 | 2012-02-16 | Vaidya Niteen A | Kit for automated resolving agent selection and method thereof |
| WO2007129188A1 (en) * | 2006-05-10 | 2007-11-15 | Pfizer Japan Inc. | Cyclopropanecarboxamide compound |
| JP2009536657A (ja) | 2006-05-10 | 2009-10-15 | レノビス， インコーポレイテッド | イオンチャンネルリガンドとしてのアミド誘導体およびそれを用いる医薬組成物および方法 |
| EP1862454A1 (en) * | 2006-06-02 | 2007-12-05 | Amorepacific Corporation | Novel compounds, isomer thereof or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and a pharmaceutical composition containing the same |
| AU2007277519B2 (en) | 2006-07-27 | 2011-12-22 | Amorepacific Corporation | Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same |
| EP1882687A1 (en) * | 2006-07-27 | 2008-01-30 | Amorepacific Corporation | Heterocyclic compounds useful as vanilloid receptor antagonists and pharmaceutical compositions containing the same |
| JP2011201778A (ja) * | 2008-07-23 | 2011-10-13 | Mochida Pharmaceut Co Ltd | ｐ−置換アリールアセトアミドを有するヘテロシクリデン誘導体 |
| KR20110086723A (ko) * | 2008-11-07 | 2011-07-29 | 시플라 리미티드 | 조피클론을 광학분할하는 방법 |
| KR20160101554A (ko) | 2015-02-17 | 2016-08-25 | (주)아모레퍼시픽 | N-[4-(1-아미노에틸)-페닐]-메탄술폰아미드 유도체의 카이랄 분할 방법 |
-
2016
- 2016-02-15 JP JP2017502582A patent/JP6687596B2/ja active Active
- 2016-02-15 WO PCT/KR2016/001474 patent/WO2016133317A1/ko not_active Ceased
- 2016-02-15 CN CN201680002149.0A patent/CN106660949B/zh active Active
- 2016-02-15 US US15/325,349 patent/US10479763B2/en active Active
- 2016-02-15 EP EP16752647.4A patent/EP3162793B1/en active Active
- 2016-02-15 BR BR112017001516-1A patent/BR112017001516B1/pt not_active IP Right Cessation
- 2016-02-15 KR KR1020177000413A patent/KR101791119B1/ko not_active Expired - Fee Related
- 2016-02-16 TW TW105104399A patent/TWI687396B/zh not_active IP Right Cessation
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