JP2017504591A5 - - Google Patents
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- JP2017504591A5 JP2017504591A5 JP2016538757A JP2016538757A JP2017504591A5 JP 2017504591 A5 JP2017504591 A5 JP 2017504591A5 JP 2016538757 A JP2016538757 A JP 2016538757A JP 2016538757 A JP2016538757 A JP 2016538757A JP 2017504591 A5 JP2017504591 A5 JP 2017504591A5
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- JP
- Japan
- Prior art keywords
- methyl
- benzamido
- dihydrogen phosphate
- pain
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 **c(cc1)cc(*)c1Oc(cc(*)c(*)c1)c1C(NC(C=CN1CO*)=CC1=O)=O Chemical compound **c(cc1)cc(*)c1Oc(cc(*)c(*)c1)c1C(NC(C=CN1CO*)=CC1=O)=O 0.000 description 1
- SQDQNNKQTHOQHO-UHFFFAOYSA-N Cc1cc(F)ccc1Oc1cc(C(F)(F)F)ccc1C(NC(C=CN1COP(O)(O)=O)=CC1=O)=O Chemical compound Cc1cc(F)ccc1Oc1cc(C(F)(F)F)ccc1C(NC(C=CN1COP(O)(O)=O)=CC1=O)=O SQDQNNKQTHOQHO-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361915937P | 2013-12-13 | 2013-12-13 | |
| US61/915,937 | 2013-12-13 | ||
| PCT/US2014/069916 WO2015089361A1 (en) | 2013-12-13 | 2014-12-12 | Prodrugs of pyridone amides useful as modulators of sodium channels |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018221093A Division JP2019055974A (ja) | 2013-12-13 | 2018-11-27 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017504591A JP2017504591A (ja) | 2017-02-09 |
| JP2017504591A5 true JP2017504591A5 (enExample) | 2018-01-25 |
| JP6463580B2 JP6463580B2 (ja) | 2019-02-06 |
Family
ID=52293220
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016538757A Active JP6463580B2 (ja) | 2013-12-13 | 2014-12-12 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
| JP2018221093A Withdrawn JP2019055974A (ja) | 2013-12-13 | 2018-11-27 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
| JP2020134430A Active JP7465174B2 (ja) | 2013-12-13 | 2020-08-07 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2018221093A Withdrawn JP2019055974A (ja) | 2013-12-13 | 2018-11-27 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
| JP2020134430A Active JP7465174B2 (ja) | 2013-12-13 | 2020-08-07 | ナトリウムチャネルの調節剤として有用なピリドンアミドのプロドラッグ |
Country Status (33)
Families Citing this family (73)
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| KR20240031299A (ko) | 2021-06-04 | 2024-03-07 | 버텍스 파마슈티칼스 인코포레이티드 | (2r,3s,4s,5r)-4-[[3-(3,4-디플루오로-2-메톡시-페닐)-4,5-디메틸-5-(트리플루오로메틸)테트라하이드로푸란-2-카르보닐]아미노]피리딘-2-카르복사미드를 포함하는 고체 투여 형태 및 투여 요법 |
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