JP2016518399A5 - - Google Patents
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- JP2016518399A5 JP2016518399A5 JP2016512427A JP2016512427A JP2016518399A5 JP 2016518399 A5 JP2016518399 A5 JP 2016518399A5 JP 2016512427 A JP2016512427 A JP 2016512427A JP 2016512427 A JP2016512427 A JP 2016512427A JP 2016518399 A5 JP2016518399 A5 JP 2016518399A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- amino
- hydroxy
- benzamide
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1308409.0 | 2013-05-10 | ||
| GB201308409A GB201308409D0 (en) | 2013-05-10 | 2013-05-10 | Compounds |
| GB201315253A GB201315253D0 (en) | 2013-08-28 | 2013-08-28 | Compounds |
| GB1315253.3 | 2013-08-28 | ||
| PCT/GB2014/051454 WO2014181137A1 (en) | 2013-05-10 | 2014-05-12 | Novel histone deacetylase inhibitors |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019015446A Division JP2019077721A (ja) | 2013-05-10 | 2019-01-31 | 新規ヒストンデアセチラーゼインヒビター |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016518399A JP2016518399A (ja) | 2016-06-23 |
| JP2016518399A5 true JP2016518399A5 (enExample) | 2017-03-16 |
| JP6513078B2 JP6513078B2 (ja) | 2019-05-15 |
Family
ID=50736120
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016512427A Expired - Fee Related JP6513078B2 (ja) | 2013-05-10 | 2014-05-12 | 新規ヒストンデアセチラーゼインヒビター |
| JP2019015446A Withdrawn JP2019077721A (ja) | 2013-05-10 | 2019-01-31 | 新規ヒストンデアセチラーゼインヒビター |
| JP2020103565A Pending JP2020158523A (ja) | 2013-05-10 | 2020-06-16 | 新規ヒストンデアセチラーゼインヒビター |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019015446A Withdrawn JP2019077721A (ja) | 2013-05-10 | 2019-01-31 | 新規ヒストンデアセチラーゼインヒビター |
| JP2020103565A Pending JP2020158523A (ja) | 2013-05-10 | 2020-06-16 | 新規ヒストンデアセチラーゼインヒビター |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US9862685B2 (enExample) |
| EP (1) | EP2994465B1 (enExample) |
| JP (3) | JP6513078B2 (enExample) |
| KR (1) | KR20160007577A (enExample) |
| CN (1) | CN105358550B (enExample) |
| AU (1) | AU2014264370B2 (enExample) |
| BR (1) | BR112015028215A2 (enExample) |
| CA (1) | CA2911856A1 (enExample) |
| CY (1) | CY1120705T1 (enExample) |
| DK (1) | DK2994465T3 (enExample) |
| ES (1) | ES2688815T3 (enExample) |
| HR (1) | HRP20181381T1 (enExample) |
| HU (1) | HUE039690T2 (enExample) |
| IL (1) | IL242388B (enExample) |
| LT (1) | LT2994465T (enExample) |
| MX (1) | MX373196B (enExample) |
| NZ (1) | NZ714283A (enExample) |
| PL (1) | PL2994465T3 (enExample) |
| PT (1) | PT2994465T (enExample) |
| RS (1) | RS57816B1 (enExample) |
| SG (1) | SG11201509174UA (enExample) |
| SI (1) | SI2994465T1 (enExample) |
| SM (1) | SMT201800501T1 (enExample) |
| WO (1) | WO2014181137A1 (enExample) |
Families Citing this family (45)
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| SI2994465T1 (sl) | 2013-05-10 | 2018-10-30 | Karus Therapeutics Limited | Novi inhibitorji histon deacetilaze |
| GB201402431D0 (en) | 2014-02-12 | 2014-03-26 | Karus Therapeutics Ltd | Compounds |
| GB201419228D0 (en) | 2014-10-29 | 2014-12-10 | Karus Therapeutics Ltd | Compounds |
| GB201419264D0 (en) * | 2014-10-29 | 2014-12-10 | Karus Therapeutics Ltd | Compounds |
| GB201514756D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Compound and method of use |
| GB201514754D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Compounds |
| GB201514760D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Compounds and method of use |
| GB201514758D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Formulation |
| GB201514751D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Compounds |
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| CA2903481A1 (en) * | 2013-03-13 | 2014-10-09 | The University Of North Carolina At Chapel Hill | Nanofluidic devices for the rapid mapping of whole genomes and related systems and methods of analysis |
| US20160052926A1 (en) | 2013-03-15 | 2016-02-25 | Hutchison Medipharma Limited | Novel pyrimidine and pyridine compounds and usage thereof |
| WO2014153280A1 (en) | 2013-03-22 | 2014-09-25 | Merck Sharp & Dohme Corp. | 2-pyridyl carboxamide-containing spleen tyrosine kinase (syk) inhibitors |
| SI2994465T1 (sl) | 2013-05-10 | 2018-10-30 | Karus Therapeutics Limited | Novi inhibitorji histon deacetilaze |
| ES2818933T3 (es) | 2013-10-10 | 2021-04-14 | Acetylon Pharmaceuticals Inc | Inhibidores de la HDAC en combinación con los inhibidores de la pi3k, para el tratamiento del linfoma no Hodgkin |
| GB201402431D0 (en) | 2014-02-12 | 2014-03-26 | Karus Therapeutics Ltd | Compounds |
| EP3187497A4 (en) | 2014-08-26 | 2018-02-07 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
| GB201419228D0 (en) | 2014-10-29 | 2014-12-10 | Karus Therapeutics Ltd | Compounds |
| GB201419264D0 (en) | 2014-10-29 | 2014-12-10 | Karus Therapeutics Ltd | Compounds |
| GB201514756D0 (en) | 2015-08-19 | 2015-09-30 | Karus Therapeutics Ltd | Compound and method of use |
| GB201609786D0 (en) | 2016-06-03 | 2016-07-20 | Karus Therapeutics Ltd | Compounds and method of use |
| WO2017222952A1 (en) | 2016-06-23 | 2017-12-28 | Merck Sharp & Dohme Corp. | 3- heteroaryl substituted 5-trifluoromethyl oxadiazoles as histone deacetylase 6 (hdac6) inhibitors |
| WO2017222950A1 (en) | 2016-06-23 | 2017-12-28 | Merck Sharp & Dohme Corp. | 3-heterocyclyl substituted 5-trifluoromethyl oxadiazoles as histone deacetylase 6 (hdac6) inhibitors |
| EP3475275B1 (en) | 2016-06-23 | 2024-04-10 | Merck Sharp & Dohme LLC | 3-aryl and heteroaryl substituted 5-trifluoromethyl oxadiazoles as histone deacetylase 6 (hdac6) inhibitors |
| GB201803361D0 (en) | 2018-03-01 | 2018-04-18 | Karus Therapeutics Ltd | Histone deacetylase inhibitors |
-
2014
- 2014-05-12 SI SI201430874T patent/SI2994465T1/sl unknown
- 2014-05-12 PL PL14725240T patent/PL2994465T3/pl unknown
- 2014-05-12 HR HRP20181381TT patent/HRP20181381T1/hr unknown
- 2014-05-12 SM SM20180501T patent/SMT201800501T1/it unknown
- 2014-05-12 KR KR1020157034809A patent/KR20160007577A/ko not_active Abandoned
- 2014-05-12 AU AU2014264370A patent/AU2014264370B2/en not_active Ceased
- 2014-05-12 US US14/890,331 patent/US9862685B2/en not_active Expired - Fee Related
- 2014-05-12 CA CA2911856A patent/CA2911856A1/en not_active Abandoned
- 2014-05-12 CN CN201480035628.3A patent/CN105358550B/zh not_active Expired - Fee Related
- 2014-05-12 SG SG11201509174UA patent/SG11201509174UA/en unknown
- 2014-05-12 PT PT14725240T patent/PT2994465T/pt unknown
- 2014-05-12 LT LTEP14725240.7T patent/LT2994465T/lt unknown
- 2014-05-12 WO PCT/GB2014/051454 patent/WO2014181137A1/en not_active Ceased
- 2014-05-12 MX MX2015015450A patent/MX373196B/es active IP Right Grant
- 2014-05-12 NZ NZ714283A patent/NZ714283A/en not_active IP Right Cessation
- 2014-05-12 JP JP2016512427A patent/JP6513078B2/ja not_active Expired - Fee Related
- 2014-05-12 RS RS20181097A patent/RS57816B1/sr unknown
- 2014-05-12 BR BR112015028215A patent/BR112015028215A2/pt not_active IP Right Cessation
- 2014-05-12 EP EP14725240.7A patent/EP2994465B1/en active Active
- 2014-05-12 ES ES14725240.7T patent/ES2688815T3/es active Active
- 2014-05-12 DK DK14725240.7T patent/DK2994465T3/en active
- 2014-05-12 HU HUE14725240A patent/HUE039690T2/hu unknown
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2015
- 2015-11-01 IL IL242388A patent/IL242388B/en active IP Right Grant
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2017
- 2017-08-02 US US15/667,069 patent/US10870624B2/en not_active Expired - Fee Related
-
2018
- 2018-09-18 CY CY181100964T patent/CY1120705T1/el unknown
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2019
- 2019-01-31 JP JP2019015446A patent/JP2019077721A/ja not_active Withdrawn
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2020
- 2020-06-16 JP JP2020103565A patent/JP2020158523A/ja active Pending
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