JP2016509589A5 - - Google Patents
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- Publication number
- JP2016509589A5 JP2016509589A5 JP2015550733A JP2015550733A JP2016509589A5 JP 2016509589 A5 JP2016509589 A5 JP 2016509589A5 JP 2015550733 A JP2015550733 A JP 2015550733A JP 2015550733 A JP2015550733 A JP 2015550733A JP 2016509589 A5 JP2016509589 A5 JP 2016509589A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- phenyl
- benzyl
- alkyl
- plant
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims 18
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 7
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 claims 6
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 4
- 208000031888 Mycoses Diseases 0.000 claims 3
- 229910052736 halogen Inorganic materials 0.000 claims 3
- 150000002367 halogens Chemical class 0.000 claims 3
- 125000005842 heteroatom Chemical group 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 229920006395 saturated elastomer Polymers 0.000 claims 3
- 238000006467 substitution reaction Methods 0.000 claims 3
- -1 -S (O) 2 R 5 Chemical group 0.000 claims 2
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 2
- 125000005129 aryl carbonyl group Chemical group 0.000 claims 2
- 230000002538 fungal effect Effects 0.000 claims 2
- 238000000034 method Methods 0.000 claims 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 2
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 2
- 239000002689 soil Substances 0.000 claims 2
- 125000004890 (C1-C6) alkylamino group Chemical group 0.000 claims 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 claims 1
- 125000006771 (C1-C6) haloalkylthio group Chemical group 0.000 claims 1
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical group Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 claims 1
- CPELXLSAUQHCOX-UHFFFAOYSA-N Hydrogen bromide Chemical compound Br CPELXLSAUQHCOX-UHFFFAOYSA-N 0.000 claims 1
- 241001360088 Zymoseptoria tritici Species 0.000 claims 1
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 claims 1
- 239000012876 carrier material Substances 0.000 claims 1
- 229910052801 chlorine Inorganic materials 0.000 claims 1
- 125000001309 chloro group Chemical group Cl* 0.000 claims 1
- 125000004093 cyano group Chemical group *C#N 0.000 claims 1
- XMBWDFGMSWQBCA-UHFFFAOYSA-N hydrogen iodide Chemical compound I XMBWDFGMSWQBCA-UHFFFAOYSA-N 0.000 claims 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 1
- 230000003287 optical effect Effects 0.000 claims 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 1
- 241000894007 species Species 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261747128P | 2012-12-28 | 2012-12-28 | |
| US61/747,128 | 2012-12-28 | ||
| PCT/US2013/077478 WO2014105821A1 (en) | 2012-12-28 | 2013-12-23 | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016509589A JP2016509589A (ja) | 2016-03-31 |
| JP2016509589A5 true JP2016509589A5 (enExample) | 2017-02-09 |
| JP6336480B2 JP6336480B2 (ja) | 2018-06-06 |
Family
ID=51022027
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015550733A Active JP6336480B2 (ja) | 2012-12-28 | 2013-12-23 | １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US9271497B2 (enExample) |
| EP (2) | EP2945635A4 (enExample) |
| JP (1) | JP6336480B2 (enExample) |
| KR (1) | KR20150103095A (enExample) |
| CN (1) | CN104994859B (enExample) |
| AU (1) | AU2013370470B2 (enExample) |
| BR (1) | BR102013033840B1 (enExample) |
| CA (1) | CA2893776A1 (enExample) |
| CL (1) | CL2015001861A1 (enExample) |
| EC (1) | ECSP15032926A (enExample) |
| GT (1) | GT201500196A (enExample) |
| HK (1) | HK1214518A1 (enExample) |
| IL (1) | IL239562B (enExample) |
| MX (1) | MX2015008443A (enExample) |
| RU (2) | RU2656101C2 (enExample) |
| UA (1) | UA117123C2 (enExample) |
| WO (1) | WO2014105821A1 (enExample) |
| ZA (1) | ZA201504195B (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUE047711T2 (hu) | 2012-12-28 | 2020-05-28 | Adama Makhteshim Ltd | N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok |
| RU2015131149A (ru) | 2012-12-28 | 2017-02-03 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные |
| LT2938191T (lt) | 2012-12-28 | 2018-05-10 | Dow Agrosciences Llc | Sinergistiniai fungicidiniai mišiniai, skirti grybelių kontrolei javuose |
| CA2894553C (en) | 2012-12-31 | 2021-03-02 | Dow Agrosciences Llc | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides |
| EA030030B1 (ru) | 2013-12-31 | 2018-06-29 | Адама Мактешим Лтд. | Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами |
| EP3097096A4 (en) | 2013-12-31 | 2017-10-11 | Adama Makhteshim Ltd. | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
| EP3808181A1 (en) | 2014-12-30 | 2021-04-21 | Dow AgroSciences LLC | Use of picolinamide compounds as fungicides |
| MX2017008418A (es) | 2014-12-30 | 2017-09-28 | Dow Agrosciences Llc | Picolinamidas con actividad fungicida. |
| CN107205398B (zh) | 2014-12-30 | 2020-08-21 | 美国陶氏益农公司 | 具有杀真菌活性的吡啶酰胺化合物 |
| AU2015374379B2 (en) | 2014-12-30 | 2018-10-04 | Dow Agrosciences Llc | Picolinamides as fungicides |
| RU2704867C2 (ru) | 2014-12-30 | 2019-10-31 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Применение соединений пиколинамида с фунгицидным действием |
| TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
| CN110996665B (zh) | 2017-05-02 | 2021-10-26 | 陶氏益农公司 | 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途 |
| TW201842851A (zh) | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
| CN107192785B (zh) * | 2017-06-09 | 2019-10-15 | 西南大学 | 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用 |
| EP3655396A1 (en) | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
| EP3866597A4 (en) | 2018-10-15 | 2022-06-29 | Corteva Agriscience LLC | Methods for sythesis of oxypicolinamides |
| CR20210270A (es) | 2018-11-05 | 2021-07-20 | Adama Makhteshim Ltd | Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos |
| TWI808347B (zh) | 2019-09-23 | 2023-07-11 | 以色列商亞當馬赫特希姆有限公司 | 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法 |
| US12281076B2 (en) | 2019-10-18 | 2025-04-22 | Corteva Agriscience Llc | Process for synthesis of picolinamides |
| MX2022011088A (es) | 2020-03-09 | 2022-09-29 | Adama Makhteshim Ltd | Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona. |
Family Cites Families (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH421973A (de) | 1962-05-01 | 1966-10-15 | Hoffmann La Roche | Verfahren zur Herstellung eines Cytosin-Derivates |
| US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (enExample) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| GR80171B (en) | 1983-08-29 | 1985-01-02 | Ciba Geigy Ag | N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| ES2057172T3 (es) | 1988-03-09 | 1994-10-16 | Ciba Geigy Ag | Agente para la proteccion de plantas contra enfermedades. |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤 |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| MX9800136A (es) | 1995-07-05 | 1998-03-29 | Du Pont | Pirimidinonas fungicidas. |
| IL125589A0 (en) | 1996-03-11 | 1999-03-12 | Novartis Ag | Pyrimidin-4-one derivatives as pesticides |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| US7914799B2 (en) | 2001-08-27 | 2011-03-29 | Immunitor USA, Inc. | Anti-fungal composition |
| JPWO2005095419A1 (ja) | 2004-04-01 | 2008-02-21 | 武田薬品工業株式会社 | チアゾロピリミジン誘導体 |
| US20080004253A1 (en) | 2006-06-30 | 2008-01-03 | Bryan James Branstetter | Thiazolopyrimidine modulators of TRPV1 |
| CA2676173A1 (en) | 2007-02-16 | 2008-08-28 | Amgen Inc. | Nitrogen-containing heterocyclyl ketones and their use as c-met inhibitors |
| AR070228A1 (es) | 2008-01-22 | 2010-03-25 | Dow Agrosciences Llc | Derivados de 5-fluoro pirimidina |
| US20100284959A1 (en) * | 2008-01-23 | 2010-11-11 | Gene Arrest Ltd. | Sequence specific double-stranded dna/rna binding compounds and uses thereof |
| WO2010047866A2 (en) | 2008-08-01 | 2010-04-29 | Dow Agrosciences Llc | Use of 5-fluorocytosine as a fungicide |
| ME02254B (me) | 2009-01-23 | 2015-12-31 | Euro Celtique Sa | Derivati hidroksamske kiseline |
| UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| US8318758B2 (en) | 2009-08-07 | 2012-11-27 | Dow Agrosciences, Llc | 5-fluoro-2-oxopyrimidine-1(2H)-carboxylate derivatives |
| AU2010279411B2 (en) | 2009-08-07 | 2014-10-23 | Adama Makhteshim Ltd. | N1-sulfonyl-5-fluoropyrimidinone derivatives |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| UA112284C2 (uk) * | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| CN102946730B (zh) * | 2010-04-26 | 2015-02-04 | 陶氏益农公司 | N3-取代的-n1-磺酰基-5-氟嘧啶酮衍生物 |
| CN103501613B (zh) | 2011-02-11 | 2017-06-13 | 陶氏益农公司 | 稳定的农用化学品油分散体 |
| HUE047711T2 (hu) * | 2012-12-28 | 2020-05-28 | Adama Makhteshim Ltd | N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok |
| RU2015131149A (ru) * | 2012-12-28 | 2017-02-03 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные |
-
2013
- 2013-12-23 UA UAA201507549A patent/UA117123C2/uk unknown
- 2013-12-23 JP JP2015550733A patent/JP6336480B2/ja active Active
- 2013-12-23 CN CN201380068093.5A patent/CN104994859B/zh active Active
- 2013-12-23 RU RU2015131110A patent/RU2656101C2/ru not_active IP Right Cessation
- 2013-12-23 EP EP13869394.0A patent/EP2945635A4/en not_active Withdrawn
- 2013-12-23 AU AU2013370470A patent/AU2013370470B2/en not_active Ceased
- 2013-12-23 EP EP19217878.8A patent/EP3689142A1/en active Pending
- 2013-12-23 MX MX2015008443A patent/MX2015008443A/es unknown
- 2013-12-23 US US14/655,568 patent/US9271497B2/en active Active
- 2013-12-23 CA CA2893776A patent/CA2893776A1/en not_active Abandoned
- 2013-12-23 RU RU2018118951A patent/RU2018118951A/ru not_active Application Discontinuation
- 2013-12-23 WO PCT/US2013/077478 patent/WO2014105821A1/en not_active Ceased
- 2013-12-23 KR KR1020157020064A patent/KR20150103095A/ko not_active Withdrawn
- 2013-12-23 HK HK16102498.5A patent/HK1214518A1/zh unknown
- 2013-12-27 BR BR102013033840A patent/BR102013033840B1/pt active IP Right Grant
-
2015
- 2015-06-10 ZA ZA2015/04195A patent/ZA201504195B/en unknown
- 2015-06-21 IL IL239562A patent/IL239562B/en active IP Right Grant
- 2015-06-26 CL CL2015001861A patent/CL2015001861A1/es unknown
- 2015-06-26 GT GT201500196A patent/GT201500196A/es unknown
- 2015-07-28 EC ECIEPI201532926A patent/ECSP15032926A/es unknown
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