ECSP15032926A - Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona - Google Patents

Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Info

Publication number
ECSP15032926A
ECSP15032926A ECIEPI201532926A ECPI201532926A ECSP15032926A EC SP15032926 A ECSP15032926 A EC SP15032926A EC IEPI201532926 A ECIEPI201532926 A EC IEPI201532926A EC PI201532926 A ECPI201532926 A EC PI201532926A EC SP15032926 A ECSP15032926 A EC SP15032926A
Authority
EC
Ecuador
Prior art keywords
compounds
fungicides
dihydropyrimidin
imino
fluoro
Prior art date
Application number
ECIEPI201532926A
Other languages
English (en)
Spanish (es)
Inventor
W Owen
Beth Lorsbach
Chenglin Yao
Lindsay Stelzer
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP15032926A publication Critical patent/ECSP15032926A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ECIEPI201532926A 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona ECSP15032926A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
ECSP15032926A true ECSP15032926A (es) 2015-11-30

Family

ID=51022027

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201532926A ECSP15032926A (es) 2012-12-28 2015-07-28 Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona

Country Status (18)

Country Link
US (1) US9271497B2 (enExample)
EP (2) EP2945635A4 (enExample)
JP (1) JP6336480B2 (enExample)
KR (1) KR20150103095A (enExample)
CN (1) CN104994859B (enExample)
AU (1) AU2013370470B2 (enExample)
BR (1) BR102013033840B1 (enExample)
CA (1) CA2893776A1 (enExample)
CL (1) CL2015001861A1 (enExample)
EC (1) ECSP15032926A (enExample)
GT (1) GT201500196A (enExample)
HK (1) HK1214518A1 (enExample)
IL (1) IL239562B (enExample)
MX (1) MX2015008443A (enExample)
RU (2) RU2018118951A (enExample)
UA (1) UA117123C2 (enExample)
WO (1) WO2014105821A1 (enExample)
ZA (1) ZA201504195B (enExample)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6352302B2 (ja) 2012-12-28 2018-07-04 ダウ アグロサイエンシィズ エルエルシー 穀類における真菌防除のための相乗性殺真菌性混合物
KR20150103096A (ko) 2012-12-28 2015-09-09 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체
MX2015008444A (es) 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EA030056B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
SG11201605377VA (en) 2013-12-31 2016-08-30 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
UA121561C2 (uk) 2014-12-30 2020-06-25 Дау Аґросаєнсиз Елелсі Застосування сполук аміду як фунгіцидів
AU2015374380B2 (en) 2014-12-30 2018-01-18 Dow Agrosciences Llc Use of picolinamides as fungicides
MX2017008418A (es) 2014-12-30 2017-09-28 Dow Agrosciences Llc Picolinamidas con actividad fungicida.
EP3240413B1 (en) 2014-12-30 2020-05-13 Dow Agrosciences LLC Picolinamide compounds with fungicidal activity
WO2016109302A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
IL309708B1 (en) 2017-07-17 2025-10-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-4,3-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
US11639334B2 (en) 2018-10-15 2023-05-02 Corteva Agriscience Llc Methods for synthesis of oxypicolinamides
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
EP4034529A1 (en) 2019-09-23 2022-08-03 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
EP0332579B1 (de) 1988-03-09 1994-08-10 Ciba-Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
JP4010563B2 (ja) 1995-07-05 2007-11-21 イー・アイ・デユポン・ドウ・ヌムール・アンド・カンパニー 殺菌・殺カビ性のピリミジノン類
CN1213373A (zh) 1996-03-11 1999-04-07 诺瓦提斯公司 农药用嘧啶－4－酮衍生物
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2114898A2 (en) * 2007-02-16 2009-11-11 Amgen Inc. Nitrogen-containing heterocyclyl ketones and their use as c-met inhibitors
EP2562175A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
US20100284959A1 (en) * 2008-01-23 2010-11-11 Gene Arrest Ltd. Sequence specific double-stranded dna/rna binding compounds and uses thereof
EP2647287A1 (en) 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides
RS54192B1 (sr) * 2009-01-23 2015-12-31 Euro-Celtique S.A. Derivati hidroksamske kiseline
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
BR112012002807B1 (pt) 2009-08-07 2018-07-10 Adama Makhteshim Ltd. Derivados de 5-flúor-2-oxopirimidina-1(2h)- caboxilato, composição e processo para controle e prevenção de ataque fúngico em uma planta de ataque fúngico em uma planta
JP5784603B2 (ja) 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
UA106889C2 (uk) * 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-ацил-5-фторпіримідинону
UA112284C2 (uk) * 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
MX2012012530A (es) * 2010-04-26 2012-12-17 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluorpirimidinona.
EP2672825A4 (en) 2011-02-11 2014-09-10 Dow Agrosciences Llc STABLE AGROCHEMICAL OIL DISPERSIONS
KR20150103096A (ko) * 2012-12-28 2015-09-09 다우 아그로사이언시즈 엘엘씨 N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체
MX2015008444A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de n-(sustituido)-5-flouro-4-imino-3-metil-2-oxo-3,4-dih idropirimidin-1 (2h)-carboximida.

Also Published As

Publication number Publication date
EP3689142A1 (en) 2020-08-05
RU2015131110A (ru) 2017-02-03
CA2893776A1 (en) 2014-07-03
AU2013370470B2 (en) 2018-05-10
HK1214518A1 (zh) 2016-07-29
US9271497B2 (en) 2016-03-01
RU2018118951A3 (enExample) 2019-02-26
CL2015001861A1 (es) 2015-10-02
WO2014105821A1 (en) 2014-07-03
EP2945635A1 (en) 2015-11-25
RU2656101C2 (ru) 2018-05-31
GT201500196A (es) 2016-03-02
CN104994859A (zh) 2015-10-21
UA117123C2 (uk) 2018-06-25
IL239562A0 (en) 2015-08-31
AU2013370470A1 (en) 2015-07-02
KR20150103095A (ko) 2015-09-09
JP6336480B2 (ja) 2018-06-06
RU2018118951A (ru) 2018-11-02
BR102013033840A2 (pt) 2015-10-06
ZA201504195B (en) 2017-08-30
EP2945635A4 (en) 2016-05-25
HK1216147A1 (zh) 2016-10-21
IL239562B (en) 2018-02-28
JP2016509589A (ja) 2016-03-31
MX2015008443A (es) 2015-09-23
US20150342188A1 (en) 2015-12-03
BR102013033840B1 (pt) 2019-09-10
CN104994859B (zh) 2018-10-26

Similar Documents

Publication Publication Date Title
ECSP15032926A (es) Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona
MX2022012275A (es) Uso de compuestos de picolinamida como fungicidas.
ECSP15032846A (es) Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboximida
MX2015008565A (es) Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirim idin-2(1h)-ona como fungicidas.
MX357150B (es) Composicion de acaros que comprende un acaro depredador y una presa inmovilizada que se pone pone en contacto con un agente reductor de hongos y metodos y usos relacionados con el uso de dicha composicion.
ECSP15032859A (es) Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato
CO7170133A2 (es) Composición sinérgica para la protección de cultivos agrícolas y su uso
ECSP14016162A (es) Combinaciones de compuestos activos
CR20160503A (es) Compuestos de [1,2,4] triazol e imidazol sustituidos, como fungicidas
CO6341525A2 (es) Compuestos heterociclicos como pesticidas.
BR112012027439A8 (pt) Derivados de n1-sulfonil-5-flúor-pirimidinona n3-substituídos
UY35764A (es) El uso de picolinamidas macrociclicas como fungicidas.
CO6470837A2 (es) Quinazolinas sustituidas como fungicidas
CL2012002574A1 (es) Compuesto derivados de triazol; metodo para combatir y controlar insectos, ácaros, nemátodos o moluscos que comprende la aplicación del compuesto antes mencionado; composición insecticida que comprende el compùesto antes mencionado.
CO6491117A2 (es) Derivados de n1-acil-5-fluoropirimidinona
UY37442A (es) Derivados de fenilamina 4-sustituidos y su uso para proteger cultivos al combatir microorganismos fitopatogénicos indeseados
MX2012007541A (es) Derivados de hidroximoil-heterociclos fungicidas.
UY37116A (es) Imidazolil–carboxamidas sustituidas como plaguicidas
MX2014012449A (es) Derivados de n-cicloalquil-n-[(heterociclilfenil)metilen]-(tio) carboxamida.
CL2015003663A1 (es) Compuestos de pirimidinio sustituidos y derivados para combatir plagas animales.
MX382785B (es) Mezclas fungicidas binarias.
AR099596A1 (es) Combinaciones de compuestos activos que tienen propiedades insecticidas
CL2013000175A1 (es) Compuestos derivados de benzocicloalquenos como agentes antifungicos; composicion fungicida que comprende el compuesto; metodo para controlar hongos fitopatógenos de los cultivos.
UY34793A (es) ?derivados de isotiazolina útiles como compuestos insecticidas?.
CO6721051A2 (es) Mezclas de activos pesticidas que comprenden compuestos de pirazol