HK1214518A1 - 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3，4-二氢嘧啶-2(1h)-酮衍生物 - Google Patents

1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3，4-二氢嘧啶-2(1h)-酮衍生物 Download PDF

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Publication number
HK1214518A1
HK1214518A1 HK16102498.5A HK16102498A HK1214518A1 HK 1214518 A1 HK1214518 A1 HK 1214518A1 HK 16102498 A HK16102498 A HK 16102498A HK 1214518 A1 HK1214518 A1 HK 1214518A1
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HK
Hong Kong
Prior art keywords
dihydropyrimidin
imino
benzoyl
fluoro
derivatives
Prior art date
Application number
HK16102498.5A
Other languages
English (en)
Chinese (zh)
Inventor
Beth Lorsbach
W. John OWEN
Chenglin Yao
Lindsay Stelzer
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of HK1214518A1 publication Critical patent/HK1214518A1/zh

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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK16102498.5A 2012-12-28 2013-12-23 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3，4-二氢嘧啶-2(1h)-酮衍生物 HK1214518A1 (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
HK42021024260.8A Division HK40034526A (en) 2012-12-28 2016-03-04 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Related Child Applications (1)

Application Number Title Priority Date Filing Date
HK42021024260.8A Addition HK40034526A (en) 2012-12-28 2016-03-04 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (1)

Publication Number Publication Date
HK1214518A1 true HK1214518A1 (zh) 2016-07-29

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Family Applications (1)

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HK16102498.5A HK1214518A1 (zh) 2012-12-28 2013-12-23 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3，4-二氢嘧啶-2(1h)-酮衍生物

Country Status (18)

Country Link
US (1) US9271497B2 (enExample)
EP (2) EP3689142A1 (enExample)
JP (1) JP6336480B2 (enExample)
KR (1) KR20150103095A (enExample)
CN (1) CN104994859B (enExample)
AU (1) AU2013370470B2 (enExample)
BR (1) BR102013033840B1 (enExample)
CA (1) CA2893776A1 (enExample)
CL (1) CL2015001861A1 (enExample)
EC (1) ECSP15032926A (enExample)
GT (1) GT201500196A (enExample)
HK (1) HK1214518A1 (enExample)
IL (1) IL239562B (enExample)
MX (1) MX2015008443A (enExample)
RU (2) RU2656101C2 (enExample)
UA (1) UA117123C2 (enExample)
WO (1) WO2014105821A1 (enExample)
ZA (1) ZA201504195B (enExample)

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KR102309245B1 (ko) 2012-12-31 2021-10-06 아다마 마켓심 리미티드 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체
FI3096619T3 (fi) 2013-12-31 2025-09-03 Adama Makhteshim Ltd Synergistisiä sienituhoaineseoksia sienten torjuntaan viljakasveissa
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
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EP3240412A4 (en) 2014-12-30 2018-04-25 Dow Agrosciences LLC Use of picolinamide compounds with fungicidal activity
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CA2972408A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
US11639334B2 (en) 2018-10-15 2023-05-02 Corteva Agriscience Llc Methods for synthesis of oxypicolinamides
US12414559B2 (en) 2018-11-05 2025-09-16 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
WO2021059160A1 (en) 2019-09-23 2021-04-01 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

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Also Published As

Publication number Publication date
JP6336480B2 (ja) 2018-06-06
RU2656101C2 (ru) 2018-05-31
IL239562A0 (en) 2015-08-31
CN104994859B (zh) 2018-10-26
AU2013370470B2 (en) 2018-05-10
RU2018118951A (ru) 2018-11-02
CN104994859A (zh) 2015-10-21
US9271497B2 (en) 2016-03-01
GT201500196A (es) 2016-03-02
AU2013370470A1 (en) 2015-07-02
EP3689142A1 (en) 2020-08-05
WO2014105821A1 (en) 2014-07-03
JP2016509589A (ja) 2016-03-31
CL2015001861A1 (es) 2015-10-02
IL239562B (en) 2018-02-28
BR102013033840B1 (pt) 2019-09-10
ZA201504195B (en) 2017-08-30
BR102013033840A2 (pt) 2015-10-06
RU2018118951A3 (enExample) 2019-02-26
ECSP15032926A (es) 2015-11-30
RU2015131110A (ru) 2017-02-03
MX2015008443A (es) 2015-09-23
EP2945635A4 (en) 2016-05-25
HK1216147A1 (zh) 2016-10-21
EP2945635A1 (en) 2015-11-25
CA2893776A1 (en) 2014-07-03
US20150342188A1 (en) 2015-12-03
UA117123C2 (uk) 2018-06-25
KR20150103095A (ko) 2015-09-09

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