JP6336480B2 - １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体 - Google Patents

１−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体 Download PDF

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JP6336480B2
JP6336480B2 JP2015550733A JP2015550733A JP6336480B2 JP 6336480 B2 JP6336480 B2 JP 6336480B2 JP 2015550733 A JP2015550733 A JP 2015550733A JP 2015550733 A JP2015550733 A JP 2015550733A JP 6336480 B2 JP6336480 B2 JP 6336480B2
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compound according
compound
plant
phenyl
methyl
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JP2016509589A5 (enExample
JP2016509589A (ja
Inventor
ロールスバッハ，ベス
オーウェン，ダブリュー．，ジョン
ヤオ，チュンリン
ステルツァー，リンゼイ
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アダマ・マクテシム・リミテッド
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2015550733A 2012-12-28 2013-12-23 １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体 Active JP6336480B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (3)

Publication Number Publication Date
JP2016509589A JP2016509589A (ja) 2016-03-31
JP2016509589A5 JP2016509589A5 (enExample) 2017-02-09
JP6336480B2 true JP6336480B2 (ja) 2018-06-06

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US (1) US9271497B2 (enExample)
EP (2) EP2945635A4 (enExample)
JP (1) JP6336480B2 (enExample)
KR (1) KR20150103095A (enExample)
CN (1) CN104994859B (enExample)
AU (1) AU2013370470B2 (enExample)
BR (1) BR102013033840B1 (enExample)
CA (1) CA2893776A1 (enExample)
CL (1) CL2015001861A1 (enExample)
EC (1) ECSP15032926A (enExample)
GT (1) GT201500196A (enExample)
HK (1) HK1214518A1 (enExample)
IL (1) IL239562B (enExample)
MX (1) MX2015008443A (enExample)
RU (2) RU2656101C2 (enExample)
UA (1) UA117123C2 (enExample)
WO (1) WO2014105821A1 (enExample)
ZA (1) ZA201504195B (enExample)

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EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
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TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
EP3866597A4 (en) 2018-10-15 2022-06-29 Corteva Agriscience LLC Methods for sythesis of oxypicolinamides
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法
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RU2015131149A (ru) * 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные

Also Published As

Publication number Publication date
HK1214518A1 (zh) 2016-07-29
US20150342188A1 (en) 2015-12-03
EP2945635A1 (en) 2015-11-25
CN104994859A (zh) 2015-10-21
WO2014105821A1 (en) 2014-07-03
CL2015001861A1 (es) 2015-10-02
IL239562B (en) 2018-02-28
MX2015008443A (es) 2015-09-23
CA2893776A1 (en) 2014-07-03
HK1216147A1 (zh) 2016-10-21
RU2015131110A (ru) 2017-02-03
US9271497B2 (en) 2016-03-01
BR102013033840B1 (pt) 2019-09-10
CN104994859B (zh) 2018-10-26
BR102013033840A2 (pt) 2015-10-06
UA117123C2 (uk) 2018-06-25
AU2013370470A1 (en) 2015-07-02
IL239562A0 (en) 2015-08-31
RU2018118951A3 (enExample) 2019-02-26
GT201500196A (es) 2016-03-02
EP2945635A4 (en) 2016-05-25
ZA201504195B (en) 2017-08-30
RU2018118951A (ru) 2018-11-02
KR20150103095A (ko) 2015-09-09
AU2013370470B2 (en) 2018-05-10
JP2016509589A (ja) 2016-03-31
ECSP15032926A (es) 2015-11-30
EP3689142A1 (en) 2020-08-05
RU2656101C2 (ru) 2018-05-31

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