GT201500196A - Derivados de 1 - (benzoilo- sustituido) - 5 - fluoro - 4 - imino - 3 - metil - 3, 4 - dihidropirimidin- 2 (1h) - ona - Google Patents
Derivados de 1 - (benzoilo- sustituido) - 5 - fluoro - 4 - imino - 3 - metil - 3, 4 - dihidropirimidin- 2 (1h) - onaInfo
- Publication number
- GT201500196A GT201500196A GT201500196A GT201500196A GT201500196A GT 201500196 A GT201500196 A GT 201500196A GT 201500196 A GT201500196 A GT 201500196A GT 201500196 A GT201500196 A GT 201500196A GT 201500196 A GT201500196 A GT 201500196A
- Authority
- GT
- Guatemala
- Prior art keywords
- dihydropirimidin
- benzoil
- imino
- fluoro
- derivatives
- Prior art date
Links
- 101000740162 Homo sapiens Sodium- and chloride-dependent transporter XTRP3 Proteins 0.000 title 1
- 102100037189 Sodium- and chloride-dependent transporter XTRP3 Human genes 0.000 title 1
- 239000000417 fungicide Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261747128P | 2012-12-28 | 2012-12-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GT201500196A true GT201500196A (es) | 2016-03-02 |
Family
ID=51022027
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GT201500196A GT201500196A (es) | 2012-12-28 | 2015-06-26 | Derivados de 1 - (benzoilo- sustituido) - 5 - fluoro - 4 - imino - 3 - metil - 3, 4 - dihidropirimidin- 2 (1h) - ona |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US9271497B2 (enExample) |
| EP (2) | EP2945635A4 (enExample) |
| JP (1) | JP6336480B2 (enExample) |
| KR (1) | KR20150103095A (enExample) |
| CN (1) | CN104994859B (enExample) |
| AU (1) | AU2013370470B2 (enExample) |
| BR (1) | BR102013033840B1 (enExample) |
| CA (1) | CA2893776A1 (enExample) |
| CL (1) | CL2015001861A1 (enExample) |
| EC (1) | ECSP15032926A (enExample) |
| GT (1) | GT201500196A (enExample) |
| HK (1) | HK1214518A1 (enExample) |
| IL (1) | IL239562B (enExample) |
| MX (1) | MX2015008443A (enExample) |
| RU (2) | RU2656101C2 (enExample) |
| UA (1) | UA117123C2 (enExample) |
| WO (1) | WO2014105821A1 (enExample) |
| ZA (1) | ZA201504195B (enExample) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| KR102148190B1 (ko) | 2012-12-28 | 2020-08-26 | 다우 아그로사이언시즈 엘엘씨 | 곡류에서의 진균 방제를 위한 상승작용적 살진균 혼합물 |
| KR20150103096A (ko) | 2012-12-28 | 2015-09-09 | 다우 아그로사이언시즈 엘엘씨 | N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체 |
| US9642368B2 (en) | 2012-12-31 | 2017-05-09 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
| AU2014373853A1 (en) | 2013-12-31 | 2016-08-11 | Adama Makhteshim Ltd. | Synergistic fungicidal mixtures and compositions for fungal control |
| MX392211B (es) * | 2013-12-31 | 2025-03-21 | Adama Makhteshim Ltd | 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación. |
| RU2702697C2 (ru) | 2014-12-30 | 2019-10-09 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | Использование пиколинамидных соединений с фунгицидной активностью |
| KR20170100550A (ko) | 2014-12-30 | 2017-09-04 | 다우 아그로사이언시즈 엘엘씨 | 살진균 활성을 갖는 피콜린아미드 화합물 |
| BR112017013608B8 (pt) | 2014-12-30 | 2022-08-23 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
| WO2016109301A1 (en) | 2014-12-30 | 2016-07-07 | Dow Agrosciences Llc | Picolinamides with fungicidal activity |
| CA2972401C (en) | 2014-12-30 | 2023-09-05 | Dow Agrosciences Llc | Picolinamide compounds with fungicidal activity |
| CN110996665B (zh) | 2017-05-02 | 2021-10-26 | 陶氏益农公司 | 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途 |
| TW201842851A (zh) | 2017-05-02 | 2018-12-16 | 美商陶氏農業科學公司 | 用於穀類中的真菌防治之協同性混合物 |
| TWI774761B (zh) | 2017-05-02 | 2022-08-21 | 美商科迪華農業科技有限責任公司 | 用於穀物中的真菌防治之協同性混合物 |
| CN107192785B (zh) * | 2017-06-09 | 2019-10-15 | 西南大学 | 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用 |
| CN118515619A (zh) | 2017-07-17 | 2024-08-20 | 阿达玛克西姆股份有限公司 | 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物 |
| BR102019004480B1 (pt) | 2018-03-08 | 2023-03-28 | Dow Agrosciences Llc | Picolinamidas como fungicidas |
| US11639334B2 (en) | 2018-10-15 | 2023-05-02 | Corteva Agriscience Llc | Methods for synthesis of oxypicolinamides |
| EA202191250A1 (ru) | 2018-11-05 | 2021-08-20 | Адама Мактешим Лтд. | Смеси и композиции, включающие 5-фтор-4-имино-3-метил-1-тозил-3,4-дигидропиримидин-2-он, и способы их применения |
| AR120035A1 (es) | 2019-09-23 | 2022-01-26 | Adama Makhteshim Ltd | Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto |
| BR112022007354A2 (pt) | 2019-10-18 | 2022-08-23 | Corteva Agriscience Llc | Processo para síntese de picolinamidas |
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| CH421973A (de) | 1962-05-01 | 1966-10-15 | Hoffmann La Roche | Verfahren zur Herstellung eines Cytosin-Derivates |
| US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (enExample) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| EP0139613A1 (de) | 1983-08-29 | 1985-05-02 | Ciba-Geigy Ag | N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| ATE109776T1 (de) | 1988-03-09 | 1994-08-15 | Ciba Geigy Ag | Mittel zum schutz von pflanzen gegen krankheiten. |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤 |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| EP0836602B1 (en) | 1995-07-05 | 2002-01-30 | E.I. Du Pont De Nemours And Company | Fungicidal pyrimidinones |
| AU716248B2 (en) | 1996-03-11 | 2000-02-24 | Novartis Ag | Pyrimidin-4-one derivatives as pesticide |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| WO2003018051A1 (en) | 2001-08-27 | 2003-03-06 | Vic Jira | Anti-fungal composition |
| WO2005095419A1 (ja) | 2004-04-01 | 2005-10-13 | Takeda Pharmaceutial Company Limited | チアゾロピリミジン誘導体 |
| EP2044086A2 (en) | 2006-06-30 | 2009-04-08 | Janssen Pharmaceutica N.V. | Thiazolopyrimidine modulators of trpv1 |
| WO2008103277A2 (en) * | 2007-02-16 | 2008-08-28 | Amgen Inc. | Nitrogen-containing heterocyclyl ketones and their use as c-met inhibitors |
| DK2562162T3 (en) | 2008-01-22 | 2015-11-23 | Dow Agrosciences Llc | N-cyano-4-amino-5-fluoro-pyrimidine derivatives as fungicides |
| US20100284959A1 (en) * | 2008-01-23 | 2010-11-11 | Gene Arrest Ltd. | Sequence specific double-stranded dna/rna binding compounds and uses thereof |
| CA2731332A1 (en) | 2008-08-01 | 2010-04-29 | Zoltan L. Benko | Use of 5-fluorocytosine as a fungicide |
| USRE46144E1 (en) | 2009-01-23 | 2016-09-13 | Purdue Pharmaceutical Products L.P. | Hydroxamic acid derivatives |
| CN102548979B (zh) * | 2009-08-07 | 2015-05-13 | 陶氏益农公司 | 5-氟代-2-氧代嘧啶-1(2h)-甲酸酯衍生物 |
| UA112284C2 (uk) * | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| UA106889C2 (uk) * | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| RS53395B (sr) | 2009-08-07 | 2014-10-31 | Dow Agrosciences Llc | Derivati n1-sulfonil-5-fluorpirimidinona |
| UA108101C2 (xx) * | 2010-04-26 | 2015-03-25 | Похідні n3-заміщених n1-сульфоніл-5-фторпіримідинонів | |
| AU2011358608B2 (en) | 2011-02-11 | 2016-04-14 | Dow Agrosciences Llc | Stable agrochemical oil dispersions |
| US9321734B2 (en) * | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| KR20150103096A (ko) * | 2012-12-28 | 2015-09-09 | 다우 아그로사이언시즈 엘엘씨 | N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체 |
-
2013
- 2013-12-23 RU RU2015131110A patent/RU2656101C2/ru not_active IP Right Cessation
- 2013-12-23 EP EP13869394.0A patent/EP2945635A4/en not_active Withdrawn
- 2013-12-23 MX MX2015008443A patent/MX2015008443A/es unknown
- 2013-12-23 CA CA2893776A patent/CA2893776A1/en not_active Abandoned
- 2013-12-23 HK HK16102498.5A patent/HK1214518A1/zh unknown
- 2013-12-23 CN CN201380068093.5A patent/CN104994859B/zh active Active
- 2013-12-23 WO PCT/US2013/077478 patent/WO2014105821A1/en not_active Ceased
- 2013-12-23 AU AU2013370470A patent/AU2013370470B2/en not_active Ceased
- 2013-12-23 KR KR1020157020064A patent/KR20150103095A/ko not_active Withdrawn
- 2013-12-23 RU RU2018118951A patent/RU2018118951A/ru not_active Application Discontinuation
- 2013-12-23 JP JP2015550733A patent/JP6336480B2/ja active Active
- 2013-12-23 EP EP19217878.8A patent/EP3689142A1/en active Pending
- 2013-12-23 US US14/655,568 patent/US9271497B2/en active Active
- 2013-12-23 UA UAA201507549A patent/UA117123C2/uk unknown
- 2013-12-27 BR BR102013033840A patent/BR102013033840B1/pt active IP Right Grant
-
2015
- 2015-06-10 ZA ZA2015/04195A patent/ZA201504195B/en unknown
- 2015-06-21 IL IL239562A patent/IL239562B/en active IP Right Grant
- 2015-06-26 CL CL2015001861A patent/CL2015001861A1/es unknown
- 2015-06-26 GT GT201500196A patent/GT201500196A/es unknown
- 2015-07-28 EC ECIEPI201532926A patent/ECSP15032926A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CL2015001861A1 (es) | 2015-10-02 |
| CA2893776A1 (en) | 2014-07-03 |
| HK1214518A1 (zh) | 2016-07-29 |
| AU2013370470A1 (en) | 2015-07-02 |
| ZA201504195B (en) | 2017-08-30 |
| RU2015131110A (ru) | 2017-02-03 |
| US9271497B2 (en) | 2016-03-01 |
| RU2018118951A3 (enExample) | 2019-02-26 |
| EP3689142A1 (en) | 2020-08-05 |
| EP2945635A4 (en) | 2016-05-25 |
| WO2014105821A1 (en) | 2014-07-03 |
| CN104994859B (zh) | 2018-10-26 |
| EP2945635A1 (en) | 2015-11-25 |
| AU2013370470B2 (en) | 2018-05-10 |
| JP6336480B2 (ja) | 2018-06-06 |
| BR102013033840A2 (pt) | 2015-10-06 |
| CN104994859A (zh) | 2015-10-21 |
| IL239562B (en) | 2018-02-28 |
| IL239562A0 (en) | 2015-08-31 |
| MX2015008443A (es) | 2015-09-23 |
| US20150342188A1 (en) | 2015-12-03 |
| RU2656101C2 (ru) | 2018-05-31 |
| HK1216147A1 (zh) | 2016-10-21 |
| KR20150103095A (ko) | 2015-09-09 |
| ECSP15032926A (es) | 2015-11-30 |
| JP2016509589A (ja) | 2016-03-31 |
| RU2018118951A (ru) | 2018-11-02 |
| UA117123C2 (uk) | 2018-06-25 |
| BR102013033840B1 (pt) | 2019-09-10 |
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