AU2013370470B2 - 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives - Google Patents

1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Download PDF

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Publication number
AU2013370470B2
AU2013370470B2 AU2013370470A AU2013370470A AU2013370470B2 AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2 AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2
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AU
Australia
Prior art keywords
compound
plant
compounds
methyl
phenyl
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Ceased
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AU2013370470A
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AU2013370470A1 (en
Inventor
Beth Lorsbach
W. John Owen
Lindsay Stelzer
Chenglin Yao
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2013370470A 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Ceased AU2013370470B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (2)

Publication Number Publication Date
AU2013370470A1 AU2013370470A1 (en) 2015-07-02
AU2013370470B2 true AU2013370470B2 (en) 2018-05-10

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AU2013370470A Ceased AU2013370470B2 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives

Country Status (18)

Country Link
US (1) US9271497B2 (enExample)
EP (2) EP3689142A1 (enExample)
JP (1) JP6336480B2 (enExample)
KR (1) KR20150103095A (enExample)
CN (1) CN104994859B (enExample)
AU (1) AU2013370470B2 (enExample)
BR (1) BR102013033840B1 (enExample)
CA (1) CA2893776A1 (enExample)
CL (1) CL2015001861A1 (enExample)
EC (1) ECSP15032926A (enExample)
GT (1) GT201500196A (enExample)
HK (1) HK1214518A1 (enExample)
IL (1) IL239562B (enExample)
MX (1) MX2015008443A (enExample)
RU (2) RU2656101C2 (enExample)
UA (1) UA117123C2 (enExample)
WO (1) WO2014105821A1 (enExample)
ZA (1) ZA201504195B (enExample)

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CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
HUE038806T2 (hu) 2012-12-28 2018-11-28 Dow Agrosciences Llc Szinergisztikus fungicid keverékek gombás fertõzések megfékezésére gabonákban
JP2016503816A (ja) 2012-12-31 2016-02-08 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての３−アルキル−５−フルオロ−４置換イミノ−３，４−ジヒドロピリミジン−２（１ｈ）−オン誘導体
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
JP6585057B2 (ja) 2013-12-31 2019-10-02 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
NZ732573A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
RU2702697C2 (ru) 2014-12-30 2019-10-09 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Использование пиколинамидных соединений с фунгицидной активностью
AU2015374380B2 (en) 2014-12-30 2018-01-18 Dow Agrosciences Llc Use of picolinamides as fungicides
KR102805798B1 (ko) 2014-12-30 2025-05-15 코르테바 애그리사이언스 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
WO2016109300A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamides with fungicidal activity
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
WO2018204438A1 (en) 2017-05-02 2018-11-08 Dow Agrosciences Llc Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
CA3115684A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
WO2020095181A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

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US20110263627A1 (en) * 2010-04-26 2011-10-27 Dow Agrosciences Llc N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

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Also Published As

Publication number Publication date
RU2015131110A (ru) 2017-02-03
RU2018118951A3 (enExample) 2019-02-26
RU2656101C2 (ru) 2018-05-31
JP2016509589A (ja) 2016-03-31
UA117123C2 (uk) 2018-06-25
GT201500196A (es) 2016-03-02
WO2014105821A1 (en) 2014-07-03
IL239562A0 (en) 2015-08-31
EP2945635A4 (en) 2016-05-25
HK1216147A1 (zh) 2016-10-21
MX2015008443A (es) 2015-09-23
CN104994859B (zh) 2018-10-26
CA2893776A1 (en) 2014-07-03
US9271497B2 (en) 2016-03-01
RU2018118951A (ru) 2018-11-02
BR102013033840A2 (pt) 2015-10-06
IL239562B (en) 2018-02-28
JP6336480B2 (ja) 2018-06-06
EP3689142A1 (en) 2020-08-05
KR20150103095A (ko) 2015-09-09
AU2013370470A1 (en) 2015-07-02
US20150342188A1 (en) 2015-12-03
ECSP15032926A (es) 2015-11-30
EP2945635A1 (en) 2015-11-25
HK1214518A1 (zh) 2016-07-29
CN104994859A (zh) 2015-10-21
ZA201504195B (en) 2017-08-30
CL2015001861A1 (es) 2015-10-02
BR102013033840B1 (pt) 2019-09-10

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