AU2013370470B2 - 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives - Google Patents

1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Download PDF

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Publication number
AU2013370470B2
AU2013370470B2 AU2013370470A AU2013370470A AU2013370470B2 AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2 AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 A AU2013370470 A AU 2013370470A AU 2013370470 B2 AU2013370470 B2 AU 2013370470B2
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AU
Australia
Prior art keywords
compound
plant
compounds
methyl
phenyl
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Ceased
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AU2013370470A
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AU2013370470A1 (en
Inventor
Beth Lorsbach
W. John Owen
Lindsay Stelzer
Chenglin Yao
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2013370470A 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives Ceased AU2013370470B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261747128P 2012-12-28 2012-12-28
US61/747,128 2012-12-28
PCT/US2013/077478 WO2014105821A1 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives

Publications (2)

Publication Number Publication Date
AU2013370470A1 AU2013370470A1 (en) 2015-07-02
AU2013370470B2 true AU2013370470B2 (en) 2018-05-10

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AU2013370470A Ceased AU2013370470B2 (en) 2012-12-28 2013-12-23 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives

Country Status (18)

Country Link
US (1) US9271497B2 (enExample)
EP (2) EP2945635A4 (enExample)
JP (1) JP6336480B2 (enExample)
KR (1) KR20150103095A (enExample)
CN (1) CN104994859B (enExample)
AU (1) AU2013370470B2 (enExample)
BR (1) BR102013033840B1 (enExample)
CA (1) CA2893776A1 (enExample)
CL (1) CL2015001861A1 (enExample)
EC (1) ECSP15032926A (enExample)
GT (1) GT201500196A (enExample)
HK (1) HK1214518A1 (enExample)
IL (1) IL239562B (enExample)
MX (1) MX2015008443A (enExample)
RU (2) RU2018118951A (enExample)
UA (1) UA117123C2 (enExample)
WO (1) WO2014105821A1 (enExample)
ZA (1) ZA201504195B (enExample)

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EP2938191B1 (en) 2012-12-28 2018-01-31 Dow AgroSciences LLC Synergistic fungicidal mixtures for fungal control in cereals
CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
CN112094262A (zh) 2012-12-31 2020-12-18 阿达玛马克西姆股份有限公司 作为杀真菌剂的化合物
UA129860C2 (uk) 2013-12-31 2025-08-27 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
CR20160344A (es) 2013-12-31 2016-12-19 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas para el control fúngico en cereales
US10173971B2 (en) 2014-12-30 2019-01-08 Dow Agrosciences Llc Picolinamides with fungicidal activity
UA121561C2 (uk) 2014-12-30 2020-06-25 Дау Аґросаєнсиз Елелсі Застосування сполук аміду як фунгіцидів
AU2015374379B2 (en) 2014-12-30 2018-10-04 Dow Agrosciences Llc Picolinamides as fungicides
KR20170100549A (ko) 2014-12-30 2017-09-04 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
CN107426999B (zh) 2014-12-30 2023-01-20 美国陶氏益农公司 具有杀真菌活性的吡啶酰胺化合物
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
EP3618626A4 (en) 2017-05-02 2020-12-02 Dow Agrosciences LLC USE OF ACYCLIC PICOLINAMIDE COMPOUND AS A FUNGICIDE FOR THE CONTROL OF FUNGAL DISEASES ON TURF
CN107192785B (zh) * 2017-06-09 2019-10-15 西南大学 放线菌jy-22抗真菌成分分离方法及其在复配剂中的应用
IL271950B2 (en) 2017-07-17 2024-06-01 Adama Makhteshim Ltd Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
WO2020081382A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
CA3118729A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound
CN114554848A (zh) 2019-10-18 2022-05-27 科迪华农业科技有限责任公司 用于合成吡啶酰胺的方法

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US20110263627A1 (en) * 2010-04-26 2011-10-27 Dow Agrosciences Llc N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

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Also Published As

Publication number Publication date
MX2015008443A (es) 2015-09-23
JP6336480B2 (ja) 2018-06-06
JP2016509589A (ja) 2016-03-31
EP2945635A4 (en) 2016-05-25
HK1216147A1 (zh) 2016-10-21
IL239562A0 (en) 2015-08-31
HK1214518A1 (zh) 2016-07-29
UA117123C2 (uk) 2018-06-25
CA2893776A1 (en) 2014-07-03
US9271497B2 (en) 2016-03-01
ECSP15032926A (es) 2015-11-30
BR102013033840A2 (pt) 2015-10-06
IL239562B (en) 2018-02-28
US20150342188A1 (en) 2015-12-03
EP2945635A1 (en) 2015-11-25
RU2656101C2 (ru) 2018-05-31
CN104994859B (zh) 2018-10-26
RU2018118951A3 (enExample) 2019-02-26
WO2014105821A1 (en) 2014-07-03
BR102013033840B1 (pt) 2019-09-10
RU2015131110A (ru) 2017-02-03
ZA201504195B (en) 2017-08-30
EP3689142A1 (en) 2020-08-05
CN104994859A (zh) 2015-10-21
RU2018118951A (ru) 2018-11-02
AU2013370470A1 (en) 2015-07-02
GT201500196A (es) 2016-03-02
KR20150103095A (ko) 2015-09-09
CL2015001861A1 (es) 2015-10-02

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