JP2014523445A5 - - Google Patents

Download PDF

Info

Publication number
JP2014523445A5
JP2014523445A5 JP2014521743A JP2014521743A JP2014523445A5 JP 2014523445 A5 JP2014523445 A5 JP 2014523445A5 JP 2014521743 A JP2014521743 A JP 2014521743A JP 2014521743 A JP2014521743 A JP 2014521743A JP 2014523445 A5 JP2014523445 A5 JP 2014523445A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
compound
solid dispersion
composition according
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2014521743A
Other languages
English (en)
Japanese (ja)
Other versions
JP2014523445A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2012/047253 external-priority patent/WO2013012959A1/en
Publication of JP2014523445A publication Critical patent/JP2014523445A/ja
Publication of JP2014523445A5 publication Critical patent/JP2014523445A5/ja
Pending legal-status Critical Current

Links

JP2014521743A 2011-07-18 2012-07-18 前立腺癌を処置するための新規な組成物及び方法 Pending JP2014523445A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161508823P 2011-07-18 2011-07-18
US61/508,823 2011-07-18
PCT/US2012/047253 WO2013012959A1 (en) 2011-07-18 2012-07-18 Novel compositions and methods for treating prostate cancer

Publications (2)

Publication Number Publication Date
JP2014523445A JP2014523445A (ja) 2014-09-11
JP2014523445A5 true JP2014523445A5 (enExample) 2015-09-03

Family

ID=47558457

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014521743A Pending JP2014523445A (ja) 2011-07-18 2012-07-18 前立腺癌を処置するための新規な組成物及び方法

Country Status (8)

Country Link
US (3) US20140288037A1 (enExample)
EP (1) EP2734207A4 (enExample)
JP (1) JP2014523445A (enExample)
CN (1) CN103813794A (enExample)
AU (1) AU2012284053A1 (enExample)
BR (1) BR112014001440A2 (enExample)
CA (1) CA2841960A1 (enExample)
WO (1) WO2013012959A1 (enExample)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100047338A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens, In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
KR20180099916A (ko) 2007-02-09 2018-09-05 메타베이시스 테라퓨틱스, 인크. 글루카곤 수용체의 길항제
EP3153501B1 (en) 2008-08-13 2018-11-28 Metabasis Therapeutics, Inc. Glucagon antagonists
WO2010091306A1 (en) 2009-02-05 2010-08-12 Tokai Pharmaceuticals Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens
KR20150015021A (ko) 2012-06-04 2015-02-09 파마시클릭스, 인코포레이티드 브루톤 타이로신 키나아제 저해제의 결정 형태
CA2902971A1 (en) 2013-03-12 2014-09-18 Patheon, Inc. Drug delivery system
AU2014236135A1 (en) 2013-03-14 2015-09-10 Thomas Jefferson University Androgen receptor down-regulating agents and uses thereof
EP2969227B1 (en) * 2013-03-15 2019-05-08 Iceutica Inc. Abiraterone acetate formulation
WO2014165815A2 (en) * 2013-04-04 2014-10-09 University Of Maryland, Baltimore Nonsteroidal and steroidal compounds with potent androgen receptor down-regulation and anti prostate cancer activity
KR20160058774A (ko) * 2013-08-12 2016-05-25 토카이 파마슈티컬, 아이엔씨. 안드로겐-표적 치료제를 이용하는 종양 질환 치료를 위한 바이오마커
US10045998B2 (en) 2013-12-12 2018-08-14 Basf Se Solid form of abiraterone acetate
JP2017519000A (ja) 2014-06-12 2017-07-13 リガンド・ファーマシューティカルズ・インコーポレイテッド グルカゴンアンタゴニスト
US9937259B2 (en) * 2014-06-27 2018-04-10 Zhuhai Beihai Biotech Co., Ltd. Abiraterone derivatives and non-covalent complexes with albumin
US9545407B2 (en) 2014-08-07 2017-01-17 Pharmacyclics Llc Formulations of a bruton's tyrosine kinase inhibitor
WO2016057839A1 (en) * 2014-10-08 2016-04-14 Boston Biopharm, Inc. Compositions and methods for increasing the bioavailability of one or more compounds
CN105616365B (zh) * 2014-11-08 2019-04-05 山东新时代药业有限公司 一种依维莫司片剂
WO2016119742A1 (zh) * 2015-01-29 2016-08-04 苏州晶云药物科技有限公司 (3β)-17-(1H-苯并咪唑-1-基)雄甾-5,16-二烯-3-醇的盐及其制备方法
IL315294A (en) 2015-03-03 2024-10-01 Pharmacyclics Llc Pharmaceutical formulations of bruton's tyrosine kinase inhibitor
EP3824908A1 (en) 2015-04-10 2021-05-26 Capsugel Belgium NV Abiraterone acetate lipid formulations
WO2016172517A1 (en) * 2015-04-24 2016-10-27 Tokai Pharmaceuticals, Inc. Methods of treating prostate cancer
US10550107B2 (en) 2015-05-18 2020-02-04 Msn Laboratories Private Limited Process for the preparation of N-[4-[(3-chloro-4-fluoro phenyl) amino]-7-[[(3s-tetrahydro-3-furanyl]oxy]-6-quinazolinyl]-4-(dimethyl amino)-(2E)-2-butenamide (2Z)-2-butenedioate (1:2) and its polymorphs thereof
JP6796083B2 (ja) 2015-06-09 2020-12-02 カプスゲル・ベルギウム・ナムローゼ・フェンノートシャップCapsugel Belgium NV カプセル中の薬剤の噴霧乾燥ディスパーションからの迅速な溶解を達成するための製剤
CN106692051B (zh) * 2015-08-18 2021-01-12 南京诺瑞特医药科技有限公司 17-(3-吡啶)雄甾-4,6-二烯-3-酮的制剂
CN105055314A (zh) * 2015-09-28 2015-11-18 杭州安德科技有限公司 一种阿比特龙的口腔喷雾剂及其使用和制备方法
US10682362B2 (en) 2015-10-14 2020-06-16 Wayne State University Treatments and diagnostics for cancers
CN109125276A (zh) * 2017-06-19 2019-01-04 齐鲁制药有限公司 一种醋酸阿比特龙片剂的药物组合物及其制备方法
CN110636837B (zh) * 2017-08-28 2022-05-24 江苏恒瑞医药股份有限公司 一种cyp17抑制剂的药物组合物及其制备方法
CA3075095A1 (en) * 2017-09-22 2019-03-28 Dispersol Technologies, Llc Abiraterone-cyclic oligomer pharmaceutical formulations and methods of formation and administration thereof
CN109718198A (zh) * 2017-10-30 2019-05-07 浙江京新药业股份有限公司 一种治疗前列腺癌的注射剂及其制备方法
CN109956990B (zh) * 2017-12-22 2023-02-17 四川科瑞德制药股份有限公司 一种干燥哌库溴铵的方法
TW202003453A (zh) 2018-02-13 2020-01-16 美商利根德製藥公司 升糖素受體拮抗劑
PL247245B1 (pl) * 2019-01-31 2025-06-02 Gdanski Univ Medyczny Samoemulgująca kompozycja farmaceutyczna w postaci ciekłej zawierająca jako substancję aktywną substancję leczniczą nietrwałą w środowisku wodnym
CN110917152B (zh) * 2019-02-01 2021-07-02 鲁南制药集团股份有限公司 一种cyp17抑制剂片及其制备方法
CZ2019168A3 (cs) 2019-03-20 2020-09-30 Zentiva, K.S. Farmaceutická kompozice obsahující abirateron acetát
CN110538150A (zh) * 2019-09-26 2019-12-06 湖南瑞林医药科技有限公司 一种含有醋酸阿比特龙的药物组合物及其制备方法和应用
WO2021094992A1 (en) * 2019-11-14 2021-05-20 Suven Life Sciences Limited Amorphous pharmaceutical compositions of abiraterone acetate
BR112022021040A2 (pt) * 2020-04-16 2022-12-06 Tavanta Therapeutics Hungary Incorporated Métodos e composições para o tratamento de câncer de próstata
JP7320903B2 (ja) 2021-12-15 2023-08-04 湖南慧▲澤▼生物医▲薬▼科技有限公司 アビラテロン酢酸エステルを含む組成物及び使用
WO2024091899A1 (en) * 2022-10-25 2024-05-02 University Of Maryland, Baltimore Salts of galeterone and salts of next generation galeterone analogs, and uses thereof

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69837903T2 (de) * 1997-08-11 2008-02-14 Pfizer Products Inc., Groton Feste pharmazeutische Dispersionen mit erhöhter Bioverfügbarkeit
US20030059471A1 (en) * 1997-12-15 2003-03-27 Compton Bruce Jon Oral delivery formulation
DE69942721D1 (de) * 1998-04-10 2010-10-14 Mitsubishi Chem Corp Sialsäure-derivate enthaltende feste dispersion
UA80393C2 (uk) * 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0103424D0 (sv) * 2001-10-15 2001-10-15 Astrazeneca Ab Pharmaceutical formulation
WO2005053660A2 (en) * 2003-12-03 2005-06-16 Lifecycle Pharma A/S Pharmaceutical compositions comprising danazol
US20060013873A1 (en) * 2004-07-16 2006-01-19 Chih-Chiang Yang Bioadhesive dosage form of steroids
MX2007010593A (es) * 2005-03-02 2008-02-20 Univ Maryland Inhibidores de cyp17/antiandrogenos esteroideos de heteroailo de c-17 novedosos: sintesis, actividades biologicas in vitro, farmacocinetica y actividad antitumoral.
US20060204588A1 (en) * 2005-03-10 2006-09-14 Elan Pharma International Limited Formulations of a nanoparticulate finasteride, dutasteride or tamsulosin hydrochloride, and mixtures thereof
DE102005011786A1 (de) * 2005-03-11 2006-09-14 Pharmasol Gmbh Verfahren zur Herstellung ultrafeiner Submicron-Suspensionen
WO2010089763A2 (en) * 2008-06-30 2010-08-12 Reliance Life Sciences Pvt. Ltd. Poly(n-vinyl caprolactam-co-acrylamide) microparticles for controlled release applications
WO2010091306A1 (en) * 2009-02-05 2010-08-12 Tokai Pharmaceuticals Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens
WO2011017534A2 (en) * 2009-08-07 2011-02-10 Tokai Pharmaceuticals, Inc. Treatment of prostate cancer

Similar Documents

Publication Publication Date Title
JP2014523445A5 (enExample)
JP6368242B2 (ja) 40−o−(2−ヒドロキシ)エチル−ラパマイシンを含む医薬組成物
JP2009530415A5 (enExample)
EP2040704A2 (en) Pharmaceutical compositions comprising implitapide and methods of using same
KR20160093611A (ko) 경구 투여를 위한 약물 제제의 제조 방법
JP6355645B2 (ja) 活性成分としてテトラゾール誘導体を含む、溶解性が改善された固体分散体
US20170129869A1 (en) Amorphous form of eliglustat hemitartarate
RU2012131158A (ru) Фармацевтическая композиция с контролируемым высвобождением лекарственного средства
US20170319539A1 (en) Amorphous Empagliflozin
WO2016038532A1 (en) Amorphous treprostinil diethanolamine
TW201446286A (zh) 抗病毒化合物之固態分散調製劑
JP2014525449A5 (enExample)
WO2015132708A1 (en) Pharmaceutical composition of roflumilast
CN105188676A (zh) 包括葡糖激酶活化剂的固体组合物及其制备和使用方法
JP2011507838A5 (enExample)
JP2023026417A (ja) フマル酸ジメチルを含有する腸溶性錠剤
JP2025026876A (ja) 5-ブロモピリジン-3-イル3-デオキシ-3-[4-(3,4,5-トリフルオロフェニル)-1H-1,2,3-トリアゾール-1-イル]-1-チオ-α-D-ガラクトピラノシドの非晶質形態
JP2011500811A5 (enExample)
EP3302438A1 (en) Oral pharmaceutical composition of isotretinoin
JP2019516765A5 (enExample)
JP2009510027A (ja) ベンラファキシン塩酸塩の制御放出性の医薬組成物、及びその調製方法
WO2011113320A1 (zh) 包含决奈达隆的药物组合物
CN101579337A (zh) 氯吡格雷组合物及其制备方法
TWI837095B (zh) 一種醫藥組成物及其製備方法
JP2009506027A (ja) 初期溶解率が改善されたプランルカスト固体分散体の薬剤学的組成物およびその製造方法