SE0103424D0 - Pharmaceutical formulation - Google Patents

Pharmaceutical formulation

Info

Publication number
SE0103424D0
SE0103424D0 SE0103424A SE0103424A SE0103424D0 SE 0103424 D0 SE0103424 D0 SE 0103424D0 SE 0103424 A SE0103424 A SE 0103424A SE 0103424 A SE0103424 A SE 0103424A SE 0103424 D0 SE0103424 D0 SE 0103424D0
Authority
SE
Sweden
Prior art keywords
drug
sub
alpha
relates
pharmaceutical formulation
Prior art date
Application number
SE0103424A
Other languages
English (en)
Inventor
Nicola Bateman
Julie Cahill
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0103424A priority Critical patent/SE0103424D0/sv
Publication of SE0103424D0 publication Critical patent/SE0103424D0/sv
Priority to IL16130602A priority patent/IL161306A0/xx
Priority to CNA028203747A priority patent/CN1571658A/zh
Priority to PCT/GB2002/004621 priority patent/WO2003032950A1/en
Priority to HU0401369A priority patent/HUP0401369A3/hu
Priority to ARP020103826A priority patent/AR036877A1/es
Priority to BR0213248-6A priority patent/BR0213248A/pt
Priority to JP2003535754A priority patent/JP3639587B2/ja
Priority to US10/492,629 priority patent/US20060058381A1/en
Priority to CA002462219A priority patent/CA2462219A1/en
Priority to PL02368226A priority patent/PL368226A1/xx
Priority to EP02770069A priority patent/EP1439823A1/en
Priority to MXPA04003520A priority patent/MXPA04003520A/es
Priority to RU2004115023/15A priority patent/RU2004115023A/ru
Priority to KR1020047005493A priority patent/KR20050035163A/ko
Priority to ZA200402729A priority patent/ZA200402729B/xx
Priority to NO20041485A priority patent/NO20041485L/no
Priority to IS7219A priority patent/IS7219A/is
Priority to CO04043957A priority patent/CO5580755A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SE0103424A 2001-10-15 2001-10-15 Pharmaceutical formulation SE0103424D0 (sv)

Priority Applications (19)

Application Number Priority Date Filing Date Title
SE0103424A SE0103424D0 (sv) 2001-10-15 2001-10-15 Pharmaceutical formulation
KR1020047005493A KR20050035163A (ko) 2001-10-15 2002-10-11 (r)-비칼루타미드를 포함하는 약학적 제제
US10/492,629 US20060058381A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalitamide
PL02368226A PL368226A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r) -bicalutamide
PCT/GB2002/004621 WO2003032950A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r) -bicalutamide
HU0401369A HUP0401369A3 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalutamide, process for its preparation and use thereof
ARP020103826A AR036877A1 (es) 2001-10-15 2002-10-11 Formulacion farmaceutica
BR0213248-6A BR0213248A (pt) 2001-10-15 2002-10-11 Formulação farmacêutica, dose farmacêutica, dispersão sólida de um polìmero entérico, métodos para o tratamento de cãncer de próstata e/ou para a redução do risco de cancer de próstata em um paciente, para aumentara biodisponibilidade e a estabilidade em armazenamento de 4'-ciano-alfa',alfa',alfa' -trifluoro-3-(4-fluorofenilsilfonil)-2-hidróxi-2-metil propiono-m-toluidida, e para a preparação de uma formulação farmacêutica, e, usos de 4'-ciano-alfa',alfa',alfa'-trifluoro-3-(4-fluorofenilsu lfonil -2-hidróxi-2-metilpropiono-m-toluidida e de um polìmero entérico
JP2003535754A JP3639587B2 (ja) 2001-10-15 2002-10-11 医薬製剤
IL16130602A IL161306A0 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalutamide
CA002462219A CA2462219A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r) -bicalutamide
CNA028203747A CN1571658A (zh) 2001-10-15 2002-10-11 包含(r)-比卡鲁胺的药物制剂
EP02770069A EP1439823A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalutamide
MXPA04003520A MXPA04003520A (es) 2001-10-15 2002-10-11 Formulacion farmaceutica que comprende (r)-bicalutamida.
RU2004115023/15A RU2004115023A (ru) 2001-10-15 2002-10-11 Фапмацевтическая композиция, содержащая (r)-бикалутамид
ZA200402729A ZA200402729B (en) 2001-10-15 2004-04-07 Pharmaceutical formulation comprising (R) -bicalutamide.
NO20041485A NO20041485L (no) 2001-10-15 2004-04-13 Farmasoytisk formulering omfattende (R)-bicalutamid
IS7219A IS7219A (is) 2001-10-15 2004-04-14 Lyfjablanda sem inniheldur (R) -bíkalútamíð
CO04043957A CO5580755A2 (es) 2001-10-15 2004-05-12 Formulacion farmaceutica comprendiendo (r)-bicalutamida

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0103424A SE0103424D0 (sv) 2001-10-15 2001-10-15 Pharmaceutical formulation

Publications (1)

Publication Number Publication Date
SE0103424D0 true SE0103424D0 (sv) 2001-10-15

Family

ID=20285650

Family Applications (1)

Application Number Title Priority Date Filing Date
SE0103424A SE0103424D0 (sv) 2001-10-15 2001-10-15 Pharmaceutical formulation

Country Status (19)

Country Link
US (1) US20060058381A1 (sv)
EP (1) EP1439823A1 (sv)
JP (1) JP3639587B2 (sv)
KR (1) KR20050035163A (sv)
CN (1) CN1571658A (sv)
AR (1) AR036877A1 (sv)
BR (1) BR0213248A (sv)
CA (1) CA2462219A1 (sv)
CO (1) CO5580755A2 (sv)
HU (1) HUP0401369A3 (sv)
IL (1) IL161306A0 (sv)
IS (1) IS7219A (sv)
MX (1) MXPA04003520A (sv)
NO (1) NO20041485L (sv)
PL (1) PL368226A1 (sv)
RU (1) RU2004115023A (sv)
SE (1) SE0103424D0 (sv)
WO (1) WO2003032950A1 (sv)
ZA (1) ZA200402729B (sv)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0302847A3 (en) * 2001-02-27 2005-05-30 Astrazeneca Ab Pharmaceutical formulation comprising bicalutamide
NZ578743A (en) 2004-01-20 2011-04-29 Novartis Ag Direct compression formulation and process
CN101128195A (zh) * 2005-02-23 2008-02-20 阿斯利康(瑞典)有限公司 用于递送增加的稳态血浆水平的比卡鲁胺
US20080045600A1 (en) * 2006-08-17 2008-02-21 Gawande Rahul S Bicalutamide compositions
US20100048912A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens, In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
EP2393827B1 (en) 2009-02-05 2015-10-07 Tokai Pharmaceuticals, Inc. Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens
CN101987086B (zh) * 2009-08-03 2012-07-18 北京化工大学 一种超细比卡鲁胺口服片剂及其制备方法
AU2012284053A1 (en) * 2011-07-18 2014-01-23 Tokai Pharmaceuticals, Inc. Novel compositions and methods for treating prostate cancer
RS62676B1 (sr) 2012-09-11 2021-12-31 Medivation Prostate Therapeutics Llc Formulacije enzalutamida
RU2015137617A (ru) 2013-03-14 2017-04-18 Юниверсити Оф Мэриленд, Балтимор Офис Оф Текнолоджи Трансфер Агенты, подавляющие андрогенные рецепторы, и их применение
KR20160058774A (ko) 2013-08-12 2016-05-25 토카이 파마슈티컬, 아이엔씨. 안드로겐-표적 치료제를 이용하는 종양 질환 치료를 위한 바이오마커
JP6830892B2 (ja) 2014-12-05 2021-02-17 アラゴン ファーマシューティカルズ,インコーポレイテッド 抗癌性組成物
CN114886852A (zh) * 2014-12-05 2022-08-12 阿拉贡药品公司 抗癌组合物

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3629237A (en) * 1968-09-12 1971-12-21 Shinetsu Chemical Co Compositions useful as enteric coatings and method for preparing acid phthalates of cellulose ethers for them
US4309405A (en) * 1979-08-09 1982-01-05 American Home Products Corporation Sustained release pharmaceutical compositions
EP0100172B1 (en) * 1982-07-23 1987-08-12 Imperial Chemical Industries Plc Amide derivatives
US4946686A (en) * 1987-09-24 1990-08-07 Merck & Co., Inc. Solubility modulated drug delivery system
ES2111065T5 (es) * 1991-04-16 2005-06-16 Nippon Shinyaku Company, Limited Procedimiento para producir una dispersion solida.
WO1995019770A1 (en) * 1994-01-21 1995-07-27 Sepracor, Inc. Methods and compositions for treating androgen-dependent diseases using optically pure r-(-)-casodex
HUP0302847A3 (en) * 2001-02-27 2005-05-30 Astrazeneca Ab Pharmaceutical formulation comprising bicalutamide
DE60211139T2 (de) * 2001-04-02 2007-03-01 Astrazeneca Ab Feste arzneizusammensetzung enthaltend 4'-cyano-trifluoro-3-(4-fluorophenylsulphonyl) -2-hydroxy-2-methylpropiono- m toluidide und pvp

Also Published As

Publication number Publication date
JP3639587B2 (ja) 2005-04-20
CN1571658A (zh) 2005-01-26
BR0213248A (pt) 2004-09-28
HUP0401369A2 (hu) 2004-11-29
RU2004115023A (ru) 2005-04-10
CO5580755A2 (es) 2005-11-30
WO2003032950A1 (en) 2003-04-24
HUP0401369A3 (en) 2006-05-29
KR20050035163A (ko) 2005-04-15
CA2462219A1 (en) 2003-04-24
MXPA04003520A (es) 2004-07-23
NO20041485L (no) 2004-04-13
IL161306A0 (en) 2004-09-27
ZA200402729B (en) 2005-01-13
US20060058381A1 (en) 2006-03-16
EP1439823A1 (en) 2004-07-28
PL368226A1 (en) 2005-03-21
JP2004521963A (ja) 2004-07-22
AR036877A1 (es) 2004-10-13
IS7219A (is) 2004-04-14

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