JP2014505696A5 - - Google Patents

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Publication number
JP2014505696A5
JP2014505696A5 JP2013551000A JP2013551000A JP2014505696A5 JP 2014505696 A5 JP2014505696 A5 JP 2014505696A5 JP 2013551000 A JP2013551000 A JP 2013551000A JP 2013551000 A JP2013551000 A JP 2013551000A JP 2014505696 A5 JP2014505696 A5 JP 2014505696A5
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JP
Japan
Prior art keywords
morpholin
methyl
indol
purine
purin
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JP2013551000A
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English (en)
Japanese (ja)
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JP2014505696A (ja
JP5963777B2 (ja
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Priority claimed from PCT/IB2012/050428 external-priority patent/WO2012104776A1/en
Publication of JP2014505696A publication Critical patent/JP2014505696A/ja
Publication of JP2014505696A5 publication Critical patent/JP2014505696A5/ja
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Publication of JP5963777B2 publication Critical patent/JP5963777B2/ja
Expired - Fee Related legal-status Critical Current
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JP2013551000A 2011-01-31 2012-01-30 新規ヘテロ環誘導体 Expired - Fee Related JP5963777B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201161437956P 2011-01-31 2011-01-31
US61/437,956 2011-01-31
US201161552905P 2011-10-28 2011-10-28
US61/552,905 2011-10-28
PCT/IB2012/050428 WO2012104776A1 (en) 2011-01-31 2012-01-30 Novel heterocyclic derivatives

Publications (3)

Publication Number Publication Date
JP2014505696A JP2014505696A (ja) 2014-03-06
JP2014505696A5 true JP2014505696A5 (https=) 2015-03-05
JP5963777B2 JP5963777B2 (ja) 2016-08-03

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ID=45607319

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JP2013551000A Expired - Fee Related JP5963777B2 (ja) 2011-01-31 2012-01-30 新規ヘテロ環誘導体

Country Status (25)

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US (2) US8987257B2 (https=)
EP (1) EP2670753B1 (https=)
JP (1) JP5963777B2 (https=)
KR (1) KR101928116B1 (https=)
CN (1) CN103476777B (https=)
AP (1) AP2013007043A0 (https=)
AR (1) AR085039A1 (https=)
AU (1) AU2012213080B2 (https=)
BR (1) BR112013019509A2 (https=)
CA (1) CA2825605C (https=)
CL (1) CL2013002177A1 (https=)
CO (1) CO6781507A2 (https=)
CR (1) CR20130369A (https=)
EA (1) EA025011B1 (https=)
ES (1) ES2611885T3 (https=)
IL (1) IL227664A0 (https=)
MX (1) MX343706B (https=)
PE (1) PE20140293A1 (https=)
PH (1) PH12013501600A1 (https=)
PL (1) PL2670753T3 (https=)
PT (1) PT2670753T (https=)
SG (1) SG192193A1 (https=)
TW (1) TW201309700A (https=)
UY (1) UY33883A (https=)
WO (1) WO2012104776A1 (https=)

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GB201007286D0 (en) 2010-04-30 2010-06-16 Astex Therapeutics Ltd New compounds
GB201020179D0 (en) 2010-11-29 2011-01-12 Astex Therapeutics Ltd New compounds
JP5963777B2 (ja) 2011-01-31 2016-08-03 ノバルティス アーゲー 新規ヘテロ環誘導体
GB201118654D0 (en) 2011-10-28 2011-12-07 Astex Therapeutics Ltd New compounds
GB201118675D0 (en) 2011-10-28 2011-12-14 Astex Therapeutics Ltd New compounds
GB201118652D0 (en) 2011-10-28 2011-12-07 Astex Therapeutics Ltd New compounds
GB201118656D0 (en) 2011-10-28 2011-12-07 Astex Therapeutics Ltd New compounds
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GB201209613D0 (en) 2012-05-30 2012-07-11 Astex Therapeutics Ltd New compounds
GB201209609D0 (en) 2012-05-30 2012-07-11 Astex Therapeutics Ltd New compounds
GB201307577D0 (en) 2013-04-26 2013-06-12 Astex Therapeutics Ltd New compounds
JP6606428B2 (ja) * 2013-10-11 2019-11-13 国立大学法人 東京医科歯科大学 脊髄小脳変性症を予防又は治療するための薬剤
JO3512B1 (ar) 2014-03-26 2020-07-05 Astex Therapeutics Ltd مشتقات كينوكسالين مفيدة كمعدلات لإنزيم fgfr كيناز
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JP6752715B2 (ja) 2014-03-26 2020-09-09 アステックス、セラピューティックス、リミテッドAstex Therapeutics Limited 組合せ
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DK3353177T3 (da) 2015-09-23 2020-08-24 Janssen Pharmaceutica Nv Tricykliske heterocykler til behandling af cancer
AU2016328693B2 (en) 2015-09-23 2021-03-11 Janssen Pharmaceutica Nv Bi-heteroaryl substituted 1,4-benzodiazepines and uses thereof for the treatment of cancer
JP7068186B2 (ja) 2016-12-02 2022-05-16 第一三共株式会社 新規エンド-β-N-アセチルグルコサミニダーゼ
CZ308800B6 (cs) * 2019-02-12 2021-05-26 Univerzita Palackého v Olomouci Heterocyklické dusíkaté deriváty purinu, farmaceutické přípravky obsahující tyto deriváty a jejich použití při neuroprotekci
EP4161519A4 (en) * 2020-06-03 2024-07-17 Yumanity Therapeutics, Inc. PURINES AND METHODS OF USE
US12405265B2 (en) * 2020-06-12 2025-09-02 Arizona Board Of Regents On Behalf Of Arizona State University Transient reporters and methods for base editing enrichment
AU2022406926A1 (en) * 2021-12-08 2024-07-25 Kineta, Inc. Purines and methods of their use
CN115181100A (zh) * 2022-07-27 2022-10-14 广西大学 一种以嘌呤及吡咯并嘧啶母核的磺酰胺类小分子抑制剂

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