JP2013525490A5 - - Google Patents
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- Publication number
- JP2013525490A5 JP2013525490A5 JP2013509201A JP2013509201A JP2013525490A5 JP 2013525490 A5 JP2013525490 A5 JP 2013525490A5 JP 2013509201 A JP2013509201 A JP 2013509201A JP 2013509201 A JP2013509201 A JP 2013509201A JP 2013525490 A5 JP2013525490 A5 JP 2013525490A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- hydroxyl
- optionally substituted
- halo
- het
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33197410P | 2010-05-06 | 2010-05-06 | |
| US61/331,974 | 2010-05-06 | ||
| PCT/US2011/035091 WO2011140164A1 (en) | 2010-05-06 | 2011-05-04 | Aza-indole derivatives useful as modulators of faah |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013525490A JP2013525490A (ja) | 2013-06-20 |
| JP2013525490A5 true JP2013525490A5 (enExample) | 2014-06-05 |
Family
ID=44904047
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013509201A Pending JP2013525490A (ja) | 2010-05-06 | 2011-05-04 | Ｆａａｈのモジュレータとして有用なアザインドール誘導体 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20130059850A1 (enExample) |
| EP (1) | EP2566481A4 (enExample) |
| JP (1) | JP2013525490A (enExample) |
| CN (1) | CN102917707A (enExample) |
| AU (1) | AU2011248175A1 (enExample) |
| BR (1) | BR112012028055A2 (enExample) |
| CA (1) | CA2797281A1 (enExample) |
| WO (1) | WO2011140164A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201411236D0 (en) | 2014-06-25 | 2014-08-06 | Takeda Pharmaceutical | Novel compounds |
| ES2885474T3 (es) | 2015-10-13 | 2021-12-13 | Inst Nat Sante Rech Med | Derivados de sibirilina para la utilización en la prevención y/o tratamiento de trastornos asociados a la necroptosis celular |
| KR20190045216A (ko) * | 2016-09-16 | 2019-05-02 | 수미토모 케미칼 컴퍼니 리미티드 | 복소환 화합물 및 그것을 함유하는 유해 절족 동물 방제제 |
| CN109589325B (zh) * | 2019-02-19 | 2019-11-26 | 牡丹江医学院 | 一种用于治疗肠炎的药物组合物及其制备方法 |
| WO2020254289A1 (en) * | 2019-06-17 | 2020-12-24 | Ucb Pharma Gmbh | N-(phenyl)-indole-3-sulfonamide derivatives and related compounds as gpr17 modulators for treating cns disorders such as multiple sclerosis |
| CN111743864B (zh) * | 2020-08-05 | 2022-04-01 | 牡丹江医学院 | 一种体育外伤喷雾剂及其制备方法 |
| CN112159423A (zh) * | 2020-11-03 | 2021-01-01 | 凯美克(上海)医药科技有限公司 | 1H-吡咯并[2,3-b]吡啶-2-硼酸频哪醇酯的合成方法 |
| WO2022157392A1 (en) * | 2021-01-25 | 2022-07-28 | Seabelife | Use of indole, 6- and 7-azaindole derivatives as inhibitors of ferroptosis regulated cell death |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH574441A5 (enExample) * | 1973-06-14 | 1976-04-15 | Ciba Geigy Ag | |
| JPS5239672A (en) * | 1975-09-26 | 1977-03-28 | Sankyo Co Ltd | Process for preparing indole-2-allyl-3- thioeter compounds |
| NZ222878A (en) * | 1986-12-17 | 1991-02-26 | Merck Frosst Canada Inc | 3-hetero-substituted-n-benzyl-indole derivatives, and pharmaceutical compositions |
| US5095031A (en) * | 1990-08-20 | 1992-03-10 | Abbott Laboratories | Indole derivatives which inhibit leukotriene biosynthesis |
| US5527819A (en) * | 1991-09-06 | 1996-06-18 | Merck & Co., Inc. | Inhibitors of HIV reverse transcriptase |
| CN1119856A (zh) * | 1993-02-24 | 1996-04-03 | 麦克公司 | Hiv逆转录酶抑制剂 |
| FR2705346B1 (fr) * | 1993-05-18 | 1995-08-11 | Union Pharma Scient Appl | Nouveaux dérivés de pipéridinyl thio indole, leurs procédés de préparation, compositions pharmaceutiques les contenant, utiles notamment comme antalgiques . |
| RU2337909C2 (ru) * | 2002-02-01 | 2008-11-10 | Ф.Хоффманн-Ля Рош Аг | Замещенные индолы и фармацевтическая композиция, обладающая агонистической активностью в отношении альфа-1a/l адренорецептора |
| UA78999C2 (en) * | 2002-06-04 | 2007-05-10 | Wyeth Corp | 1-(aminoalkyl)-3-sulfonylazaindoles as ligands of 5-hydroxytryptamine-6 |
| TW200403243A (en) * | 2002-07-18 | 2004-03-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylazaindole or-azaindazole derivatives as 5-hydroxytryptamine-6 ligands |
| US6800655B2 (en) * | 2002-08-20 | 2004-10-05 | Sri International | Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents |
| WO2004074286A1 (en) * | 2003-02-14 | 2004-09-02 | Wyeth | Heterocyclyl-3-sulfonylazaindole or -azaindazole derivatives as 5-hydroxytryptamine-6 ligands |
| WO2006015123A1 (en) * | 2004-07-27 | 2006-02-09 | Sgx Pharmaceuticals, Inc. | Pyrrolo-pyridine kinase modulators |
| ATE445396T1 (de) * | 2004-08-19 | 2009-10-15 | Aventis Pharma Inc | 3-arylthioindol-2-carbonsäureamidderivate und ihre analoge als hemmer von caseinkinase i |
| GB2422831A (en) * | 2005-02-04 | 2006-08-09 | Oxagen Ltd | Pyrrolopyridines and their use in the treatment of diseases mediated by PGD2 at the CRTH2 receptor |
| UA95244C2 (ru) * | 2005-06-22 | 2011-07-25 | Плексикон, Инк. | Соединения и способ модулирования активности киназ, и показания для их применения |
| US7960544B2 (en) * | 2005-12-16 | 2011-06-14 | Ironwood Pharmaceuticals, Inc. | Useful indole compounds |
| US20090118503A1 (en) * | 2007-06-20 | 2009-05-07 | Kevin Sprott | Faah inhibitors |
| BRPI0908851A2 (pt) * | 2008-02-22 | 2017-05-30 | Irm Llc | compostos e composições como moduladores da atividades de gpr119 |
| HUE025471T2 (hu) * | 2008-04-16 | 2016-03-29 | Karobio Ab | Új ösztrogén receptor ligandumok |
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2011
- 2011-05-04 AU AU2011248175A patent/AU2011248175A1/en not_active Abandoned
- 2011-05-04 BR BR112012028055A patent/BR112012028055A2/pt not_active IP Right Cessation
- 2011-05-04 JP JP2013509201A patent/JP2013525490A/ja active Pending
- 2011-05-04 US US13/696,520 patent/US20130059850A1/en not_active Abandoned
- 2011-05-04 EP EP11778226.8A patent/EP2566481A4/en not_active Withdrawn
- 2011-05-04 CN CN2011800228440A patent/CN102917707A/zh active Pending
- 2011-05-04 CA CA2797281A patent/CA2797281A1/en not_active Abandoned
- 2011-05-04 WO PCT/US2011/035091 patent/WO2011140164A1/en not_active Ceased