JP2013520413A5 - - Google Patents

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Publication number
JP2013520413A5
JP2013520413A5 JP2012553849A JP2012553849A JP2013520413A5 JP 2013520413 A5 JP2013520413 A5 JP 2013520413A5 JP 2012553849 A JP2012553849 A JP 2012553849A JP 2012553849 A JP2012553849 A JP 2012553849A JP 2013520413 A5 JP2013520413 A5 JP 2013520413A5
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formula
compound
reacting
activator
reducing agent
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JP2012553849A
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Japanese (ja)
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JP2013520413A (ja
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Priority claimed from PCT/SE2011/050171 external-priority patent/WO2011102794A1/en
Publication of JP2013520413A publication Critical patent/JP2013520413A/ja
Publication of JP2013520413A5 publication Critical patent/JP2013520413A5/ja
Ceased legal-status Critical Current

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JP2012553849A 2010-02-18 2011-02-17 シクロプロピルアミド誘導体及びそれに関連する中間体の製造方法 Ceased JP2013520413A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US30558310P 2010-02-18 2010-02-18
US61/305,583 2010-02-18
PCT/SE2011/050171 WO2011102794A1 (en) 2010-02-18 2011-02-17 Processes for making cyclopropyl amide derivatives and intermediates associated therewith

Publications (2)

Publication Number Publication Date
JP2013520413A JP2013520413A (ja) 2013-06-06
JP2013520413A5 true JP2013520413A5 (https=) 2014-03-20

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ID=44370080

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2012553849A Ceased JP2013520413A (ja) 2010-02-18 2011-02-17 シクロプロピルアミド誘導体及びそれに関連する中間体の製造方法
JP2012553850A Pending JP2013520414A (ja) 2010-02-18 2011-02-17 シクロプロピルベンズアミド誘導体の新規な結晶形態
JP2015160029A Pending JP2016006103A (ja) 2010-02-18 2015-08-14 シクロプロピルベンズアミド誘導体の新規な結晶形態

Family Applications After (2)

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JP2012553850A Pending JP2013520414A (ja) 2010-02-18 2011-02-17 シクロプロピルベンズアミド誘導体の新規な結晶形態
JP2015160029A Pending JP2016006103A (ja) 2010-02-18 2015-08-14 シクロプロピルベンズアミド誘導体の新規な結晶形態

Country Status (19)

Country Link
US (2) US20110201623A1 (https=)
EP (2) EP2536702A4 (https=)
JP (3) JP2013520413A (https=)
KR (2) KR20130002316A (https=)
CN (2) CN103168027B (https=)
AR (2) AR080204A1 (https=)
AU (2) AU2011218491C1 (https=)
BR (2) BR112012020782A2 (https=)
CA (2) CA2788444A1 (https=)
CL (2) CL2012002259A1 (https=)
CO (1) CO6592109A2 (https=)
ES (1) ES2541857T3 (https=)
IL (1) IL221431A (https=)
MX (2) MX336333B (https=)
NZ (2) NZ602110A (https=)
RU (2) RU2012139082A (https=)
SG (3) SG10201501226VA (https=)
TW (2) TWI520945B (https=)
WO (2) WO2011102795A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SA08290520B1 (ar) 2007-08-22 2012-02-22 استرازينيكا ايه بي مشتقات سيكلو بروبيل أميد وتركيبات صيدلية تحتوي عليها لعلاج حالة مرضية سببها مستقبلات هيستامين h3
TW201039825A (en) * 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
JP5746718B2 (ja) * 2010-02-18 2015-07-08 アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag シクロプロピルアミド誘導体からなる固体形態
RU2012139082A (ru) * 2010-02-18 2014-03-27 Астразенека Аб Способы получения производных циклопропиламида и связанных с ними промежуточных соединений
FR3003466B1 (fr) * 2013-03-22 2015-08-07 Servier Lab Utilisation du 4-{3-[cis-hexahydrocyclopenta[c]pyrrol-2(1h)-yl]propoxy}benzamide pour le traitement des douleurs neuropathiques
EP2976322B1 (de) * 2013-03-22 2019-11-20 Merck Patent GmbH Synthesebausteine für die herstellung von materialien für organische elektrolumineszenzvorrichtungen
CN103342655A (zh) * 2013-07-02 2013-10-09 扬州大学 取代乙二酮双苯胺希夫碱合成取代酰胺的新方法
JP2026000886A (ja) 2024-06-18 2026-01-06 イーライ リリー アンド カンパニー Gip受容体アゴニスト化合物

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RU2012139082A (ru) 2010-02-18 2014-03-27 Астразенека Аб Способы получения производных циклопропиламида и связанных с ними промежуточных соединений

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