JP2011513402A5 - - Google Patents

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JP2011513402A5
JP2011513402A5 JP2010549649A JP2010549649A JP2011513402A5 JP 2011513402 A5 JP2011513402 A5 JP 2011513402A5 JP 2010549649 A JP2010549649 A JP 2010549649A JP 2010549649 A JP2010549649 A JP 2010549649A JP 2011513402 A5 JP2011513402 A5 JP 2011513402A5
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chlorophenyl
reacting
process according
ethanol
item
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JP2010549649A
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JP5491421B2 (ja
JP2011513402A (ja
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Priority claimed from PCT/US2009/001340 external-priority patent/WO2009111004A1/en
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JP2010549649A 2008-03-04 2009-03-03 ５−ｈｔ２ｃアゴニストである（ｒ）−８−クロロ−１−メチル−２，３，４，５−テトラヒドロ−１ｈ−３−ベンゾアゼピンに関連する中間体の調製のためのプロセス Expired - Fee Related JP5491421B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US6810208P 2008-03-04 2008-03-04
US61/068,102 2008-03-04
PCT/US2009/001340 WO2009111004A1 (en) 2008-03-04 2009-03-03 Processes for the preparation of intermediates related to the 5-ht2c agonist (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine

Publications (3)

Publication Number Publication Date
JP2011513402A JP2011513402A (ja) 2011-04-28
JP2011513402A5 true JP2011513402A5 (https=) 2013-03-21
JP5491421B2 JP5491421B2 (ja) 2014-05-14

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JP2010549649A Expired - Fee Related JP5491421B2 (ja) 2008-03-04 2009-03-03 ５−ｈｔ２ｃアゴニストである（ｒ）−８−クロロ−１−メチル−２，３，４，５−テトラヒドロ−１ｈ−３−ベンゾアゼピンに関連する中間体の調製のためのプロセス

Country Status (5)

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US (1) US8822727B2 (https=)
EP (1) EP2288585A1 (https=)
JP (1) JP5491421B2 (https=)
CN (1) CN102015591B (https=)
WO (1) WO2009111004A1 (https=)

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CN107673949B (zh) * 2017-10-25 2021-02-23 南京恒旺生物医药有限公司 一种1-氯-3-甲基-2-丁烯的制备方法
CN112358406A (zh) * 2020-10-28 2021-02-12 山东省药学科学院 一种氯卡色林中间体的制备方法
CN115784911A (zh) * 2022-10-19 2023-03-14 山东省药学科学院 一种1-[2-(4-氯苯基)-乙基氨基]-2-丙醇的合成方法

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