JP2010540556A5 - - Google Patents

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Publication number
JP2010540556A5
JP2010540556A5 JP2010527140A JP2010527140A JP2010540556A5 JP 2010540556 A5 JP2010540556 A5 JP 2010540556A5 JP 2010527140 A JP2010527140 A JP 2010527140A JP 2010527140 A JP2010527140 A JP 2010527140A JP 2010540556 A5 JP2010540556 A5 JP 2010540556A5
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JP
Japan
Prior art keywords
pharmaceutical composition
compound
compound according
pharmaceutical
integer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010527140A
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English (en)
Japanese (ja)
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JP2010540556A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/077673 external-priority patent/WO2009042767A1/en
Publication of JP2010540556A publication Critical patent/JP2010540556A/ja
Publication of JP2010540556A5 publication Critical patent/JP2010540556A5/ja
Pending legal-status Critical Current

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JP2010527140A 2007-09-26 2008-09-25 アザシチジン類似体およびその使用 Pending JP2010540556A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US97543707P 2007-09-26 2007-09-26
PCT/US2008/077673 WO2009042767A1 (en) 2007-09-26 2008-09-25 Azacytidine analogues and uses thereof

Publications (2)

Publication Number Publication Date
JP2010540556A JP2010540556A (ja) 2010-12-24
JP2010540556A5 true JP2010540556A5 (enExample) 2011-08-11

Family

ID=40511851

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2010527140A Pending JP2010540556A (ja) 2007-09-26 2008-09-25 アザシチジン類似体およびその使用
JP2010527139A Pending JP2010540555A (ja) 2007-09-26 2008-09-25 アザシチジン類似体およびその使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010527139A Pending JP2010540555A (ja) 2007-09-26 2008-09-25 アザシチジン類似体およびその使用

Country Status (15)

Country Link
US (2) US8399420B2 (enExample)
EP (2) EP2205073A4 (enExample)
JP (2) JP2010540556A (enExample)
KR (2) KR20100072230A (enExample)
CN (2) CN101815437A (enExample)
AU (2) AU2008304380A1 (enExample)
BR (2) BRPI0817269A2 (enExample)
CA (2) CA2700267A1 (enExample)
IL (1) IL204690A0 (enExample)
MX (2) MX2010003261A (enExample)
NZ (2) NZ583824A (enExample)
RU (1) RU2488591C2 (enExample)
UA (2) UA99308C2 (enExample)
WO (2) WO2009042766A1 (enExample)
ZA (1) ZA201001660B (enExample)

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DK3692983T3 (da) 2008-05-15 2021-09-20 Celgene Corp Orale formuleringer af cytidinanaloger og fremgangsmåder til anvendelse deraf
EP2321302B1 (en) 2008-08-01 2014-10-29 Dr. Reddy's Laboratories Ltd. Azacitidine process and polymorphs
WO2010129211A2 (en) * 2009-04-27 2010-11-11 Dr. Reddy's Laboratories Ltd. Preparation of decitabine
EP2670396A1 (en) 2011-01-31 2013-12-11 Celgene Corporation Pharmaceutical compositions of cytidine analogs and methods of use thereof
US20120264710A1 (en) * 2011-04-15 2012-10-18 Marit Liland Sandvold Systems and Methods for Detecting hENT1 Expression in Hematological Disorders
TW201700103A (zh) 2011-11-01 2017-01-01 西建公司 利用胞嘧啶核苷類似物之口服配方治療癌症的方法
JP6114317B2 (ja) 2012-02-24 2017-04-12 シグナル ファーマシューティカルズ，エルエルシー Ｔｏｒキナーゼ阻害剤の組合せ療法を用いて、非小細胞肺がんを処置する方法
US9493500B2 (en) 2012-07-19 2016-11-15 Richard Daifuku Fluorinated pyrimidine analogs and methods of use thereof
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CA3007357C (en) 2015-12-03 2023-12-05 Epidestiny, Inc. Compositions containing decitabine, 5azacytidine and tetrahydrouridine and uses thereof
CN110446504B (zh) 2017-03-20 2024-07-26 瓦西尼斯公司 用脑信号蛋白-4d抗体联合表观遗传调节剂治疗癌症
MX2019015731A (es) 2017-06-22 2020-08-03 Celgene Corp Tratamiento de carcinoma hepatocelular caracterizado por infeccion por virus de hepatitis b.
WO2019204637A1 (en) * 2018-04-19 2019-10-24 Southern Research Institute 4'-thio-nucleotide and -nucleoside prodrugs for the treatment of cancer
US20230416294A1 (en) * 2020-08-10 2023-12-28 The Johns Hopkins University Decitabine analogs for immunological and oncological therapy

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