JP2008535902A5 - - Google Patents

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Publication number
JP2008535902A5
JP2008535902A5 JP2008505964A JP2008505964A JP2008535902A5 JP 2008535902 A5 JP2008535902 A5 JP 2008535902A5 JP 2008505964 A JP2008505964 A JP 2008505964A JP 2008505964 A JP2008505964 A JP 2008505964A JP 2008535902 A5 JP2008535902 A5 JP 2008535902A5
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JP
Japan
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group
compound according
optionally substituted
treatment
attached
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2008505964A
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English (en)
Japanese (ja)
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JP2008535902A (ja
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Publication date
Priority claimed from GB0507831A external-priority patent/GB0507831D0/en
Application filed filed Critical
Priority claimed from PCT/GB2006/001369 external-priority patent/WO2006109081A1/en
Publication of JP2008535902A publication Critical patent/JP2008535902A/ja
Publication of JP2008535902A5 publication Critical patent/JP2008535902A5/ja
Pending legal-status Critical Current

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JP2008505964A 2005-04-15 2006-04-13 Ｄｎａ−ｐｋ阻害剤 Pending JP2008535902A (ja)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US67188605P 2005-04-15 2005-04-15
US67183005P 2005-04-15 2005-04-15
GB0507831A GB0507831D0 (en) 2005-04-18 2005-04-18 DNA-PK inhibitors
US69606405P 2005-07-01 2005-07-01
US71890405P 2005-09-20 2005-09-20
PCT/GB2006/001369 WO2006109081A1 (en) 2005-04-15 2006-04-13 Dna-pk inhibitors

Publications (2)

Publication Number Publication Date
JP2008535902A JP2008535902A (ja) 2008-09-04
JP2008535902A5 true JP2008535902A5 (enExample) 2009-04-30

Family

ID=36579227

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2008505966A Pending JP2008535903A (ja) 2005-04-15 2006-04-13 Ｄｎａ−ｐｋ阻害剤
JP2008505964A Pending JP2008535902A (ja) 2005-04-15 2006-04-13 Ｄｎａ−ｐｋ阻害剤

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2008505966A Pending JP2008535903A (ja) 2005-04-15 2006-04-13 Ｄｎａ−ｐｋ阻害剤

Country Status (13)

Country Link
US (2) US20060264623A1 (enExample)
EP (2) EP1869021A1 (enExample)
JP (2) JP2008535903A (enExample)
KR (1) KR20080002963A (enExample)
AR (2) AR053358A1 (enExample)
AU (1) AU2006235731A1 (enExample)
CA (1) CA2603637A1 (enExample)
IL (1) IL186445A0 (enExample)
MX (1) MX2007012696A (enExample)
NO (1) NO20075809L (enExample)
TW (2) TW200720274A (enExample)
UY (1) UY29479A1 (enExample)
WO (2) WO2006109081A1 (enExample)

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WO2011001115A1 (fr) 2009-07-02 2011-01-06 Sanofi-Aventis Nouveaux derives de 6-morpholin-4-yl-pyrimidin-4- ( 3h ) -one, leur preparation pharmaceutique comme inhibiteurs de phos phorylat i on d ' akt ( pkb )
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US8815853B2 (en) 2010-12-23 2014-08-26 Sanofi Pyrimidinone derivatives, preparation thereof and pharmaceutical use thereof
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SI3459942T1 (sl) 2012-04-24 2021-05-31 Vertex Pharmaceuticals Incorporated Inhibitorji DNA-PK
WO2013186726A2 (en) * 2012-06-15 2013-12-19 Basf Se Multicomponent crystals comprising dasatinib and selected cocrystal formers
FR2992314B1 (fr) 2012-06-22 2015-10-16 Sanofi Sa Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one et 1,2,3,4-tetrahydro-pyrimido{1,2-a}pyrimidin-6-one comportant une morpholine substituee, leur preparation et leur utilisation pharmaceutique
FR2992316A1 (fr) 2012-06-22 2013-12-27 Sanofi Sa Derives de pyrimidinones, leur preparation et leur application en therapeutique
HUE041544T2 (hu) 2013-03-12 2019-05-28 Vertex Pharma DNS-PK inhibitorok
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JP2019529475A (ja) 2016-09-27 2019-10-17 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ Ｄｎａ損傷剤とｄｎａ−ｐｋ阻害剤との組合せ物を使用する、がんを処置するための方法
CN109232476B (zh) * 2018-11-06 2020-06-26 常州大学 一种制备n-苯基-3-吗啡啉丙酰胺的方法
WO2021184014A1 (en) * 2020-03-13 2021-09-16 Arizona Board Of Regetns On Behalf Of The University Of Arizona Stable reactive compositions for bioconjugation, probes, and protein labeling
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