JP2010505940A5 - - Google Patents

Download PDF

Info

Publication number
JP2010505940A5
JP2010505940A5 JP2009531969A JP2009531969A JP2010505940A5 JP 2010505940 A5 JP2010505940 A5 JP 2010505940A5 JP 2009531969 A JP2009531969 A JP 2009531969A JP 2009531969 A JP2009531969 A JP 2009531969A JP 2010505940 A5 JP2010505940 A5 JP 2010505940A5
Authority
JP
Japan
Prior art keywords
phenyl
piperazine
carbonyl
amino
butyryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009531969A
Other languages
English (en)
Japanese (ja)
Other versions
JP5341763B2 (ja
JP2010505940A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2007/054155 external-priority patent/WO2008044217A2/en
Publication of JP2010505940A publication Critical patent/JP2010505940A/ja
Publication of JP2010505940A5 publication Critical patent/JP2010505940A5/ja
Application granted granted Critical
Publication of JP5341763B2 publication Critical patent/JP5341763B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009531969A 2006-10-13 2007-10-12 2−アミノカルボニル−ピリジン誘導体 Expired - Fee Related JP5341763B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IB2006053773 2006-10-13
IBPCT/IB2006/053773 2006-10-13
IB2006053817 2006-10-17
IBPCT/IB2006/053817 2006-10-17
PCT/IB2007/054155 WO2008044217A2 (en) 2006-10-13 2007-10-12 2-aminocarbonyl-pyridine derivatives

Publications (3)

Publication Number Publication Date
JP2010505940A JP2010505940A (ja) 2010-02-25
JP2010505940A5 true JP2010505940A5 (enExample) 2013-07-11
JP5341763B2 JP5341763B2 (ja) 2013-11-13

Family

ID=39167796

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009531969A Expired - Fee Related JP5341763B2 (ja) 2006-10-13 2007-10-12 2−アミノカルボニル−ピリジン誘導体

Country Status (17)

Country Link
US (1) US8093250B2 (enExample)
EP (1) EP2081903B1 (enExample)
JP (1) JP5341763B2 (enExample)
KR (1) KR101525260B1 (enExample)
AR (1) AR063258A1 (enExample)
AU (1) AU2007305925A1 (enExample)
BR (1) BRPI0720193A2 (enExample)
CA (1) CA2664579C (enExample)
CL (1) CL2007002920A1 (enExample)
ES (1) ES2473609T3 (enExample)
IL (1) IL198059A0 (enExample)
MA (1) MA30868B1 (enExample)
MX (1) MX2009003724A (enExample)
NO (1) NO20091838L (enExample)
RU (1) RU2009117705A (enExample)
TW (1) TW200823190A (enExample)
WO (1) WO2008044217A2 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200640877A (en) 2005-04-28 2006-12-01 Actelion Pharmaceuticals Ltd Pyrimidine derivatives
CL2007002920A1 (es) 2006-10-13 2008-06-06 Actelion Pharmaceuticals Ltd Compuestos derivados de 2-aminocarbonilpiridina; composicion farmaceutica; y uso para el tratamiento de trastornos vasculares oclusivos.
CL2007003038A1 (es) 2006-10-25 2008-06-06 Actelion Pharmaceuticals Ltd Compuestos derivados de 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y uso en el tratamiento de trastornos vasculares oclusivos.
HRP20120735T1 (hr) 2007-11-29 2012-10-31 Actelion Pharmaceuticals Ltd. Derivati fosfonske kiseline i njihova uporaba kao antagonista p2y12 receptora
US8946439B2 (en) 2008-02-29 2015-02-03 Evotec Ag Amide compounds, compositions and uses thereof
AR071652A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2- fenil-piridina substituidos
AR071653A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2-fenil-4-ciclopropil-pirimidina
US20110237578A1 (en) * 2008-09-18 2011-09-29 Zhi-Liang Wei Amide compounds, compositions and uses thereof
NZ596213A (en) 2009-04-08 2013-05-31 Actelion Pharmaceuticals Ltd 6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines as adenosine 5'-diphosphate (ADP) receptor antagonists
CA2756654C (en) 2009-04-22 2017-08-22 Actelion Pharmaceuticals Ltd Thiazole derivatives and their use as p2y12 receptor antagonists
US9120752B2 (en) 2010-07-16 2015-09-01 Purdue Pharma, L.P. Pyridine compounds as sodium channel blockers
US9539246B2 (en) 2011-08-30 2017-01-10 University Of Utah Research Foundation Methods and compositions for treating nephrogenic diabetes insipidus
US9206127B2 (en) 2012-03-16 2015-12-08 Purdue Pharm, L.P. Substituted pyridines as sodium channel blockers
EP2935257B1 (en) 2012-12-20 2018-02-07 Purdue Pharma LP Cyclic sulfonamides as sodium channel blockers
US10730866B2 (en) 2014-04-07 2020-08-04 Purdue Pharma L.P. Indole derivatives and use thereof
TWI752086B (zh) 2016-09-22 2022-01-11 瑞士商愛杜西亞製藥有限公司 結晶型式
KR102510832B1 (ko) 2017-03-15 2023-03-15 이도르시아 파마슈티컬스 리미티드 P2y12 수용체 안타고니스트의 피하 투여

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5373586A (en) 1976-12-09 1978-06-30 Mitsubishi Chem Ind Ltd New penicillin derivatives
CA2020437A1 (en) 1989-07-05 1991-01-06 Yoshihide Fuse Cinnamamide derivative
IL123986A (en) * 1997-04-24 2011-10-31 Organon Nv Medicinal compounds
KR100565701B1 (ko) * 1997-07-31 2006-03-29 우베 고산 가부시키가이샤 N-아실아미노산 아미드 화합물 및 그의 제조 중간체
EP1192132B1 (en) * 1999-06-14 2005-09-07 Eli Lilly And Company Serine protease inhibitors
US6861424B2 (en) 2001-06-06 2005-03-01 Schering Aktiengesellschaft Platelet adenosine diphosphate receptor antagonists
US7056923B2 (en) * 2002-12-11 2006-06-06 Schering Aktiengesellschaft Platelet adenosine diphosphate receptor antagonists
TW200640877A (en) * 2005-04-28 2006-12-01 Actelion Pharmaceuticals Ltd Pyrimidine derivatives
MY147373A (en) 2005-10-21 2012-11-30 Actelion Pharmaceuticals Ltd Piperazine derivatives as antimalarial agents
CL2007002920A1 (es) 2006-10-13 2008-06-06 Actelion Pharmaceuticals Ltd Compuestos derivados de 2-aminocarbonilpiridina; composicion farmaceutica; y uso para el tratamiento de trastornos vasculares oclusivos.
CL2007003038A1 (es) 2006-10-25 2008-06-06 Actelion Pharmaceuticals Ltd Compuestos derivados de 2-fenil-6-aminocarbonil-pirimidina; composicion farmaceutica; y uso en el tratamiento de trastornos vasculares oclusivos.
HRP20120735T1 (hr) 2007-11-29 2012-10-31 Actelion Pharmaceuticals Ltd. Derivati fosfonske kiseline i njihova uporaba kao antagonista p2y12 receptora
AR071653A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2-fenil-4-ciclopropil-pirimidina
AR071652A1 (es) 2008-04-11 2010-07-07 Actelion Pharmaceuticals Ltd Derivados 2- fenil-piridina substituidos
NZ596213A (en) 2009-04-08 2013-05-31 Actelion Pharmaceuticals Ltd 6-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-phenyl-pyrimidines as adenosine 5'-diphosphate (ADP) receptor antagonists
CA2756654C (en) 2009-04-22 2017-08-22 Actelion Pharmaceuticals Ltd Thiazole derivatives and their use as p2y12 receptor antagonists

Similar Documents

Publication Publication Date Title
JP2010505940A5 (enExample)
RU2483072C2 (ru) Производные фосфоновой кислоты и их применение в качестве антагонистов рецептора p2y12
JP5341763B2 (ja) 2−アミノカルボニル−ピリジン誘導体
CA2720552C (en) Acylthiourea compound or salt thereof, and use thereof
JP2012522847A5 (enExample)
TR201806882T4 (tr) Selektif östrojen reseptörü yıkıcıları olarak benzotiofen türevleri ve bunların bileşimleri.
JP2014525937A5 (enExample)
JP2012530765A5 (enExample)
JP2015533782A (ja) スルファモイル−アリールアミド及びb型肝炎の治療のための薬剤としてのその使用
JP6257787B2 (ja) Egfr−t790mキナーゼ阻害剤として置換されたピリミジニウム類化合物
JP2017533968A5 (enExample)
JP2016525075A5 (enExample)
RU2010145463A (ru) Производные замещенного 2-фенилпиридина
JP2011518811A5 (enExample)
JP2012511588A5 (enExample)
JP2012513398A5 (enExample)
EP4323350A1 (en) Isoindolinone compounds
JPWO2019143678A5 (enExample)
RU2009119421A (ru) Производные 2-фенил-6-аминокарбонилпиримидина и их применение в качестве антагонистов тромбоцитарного рецептора адф (p2y12 рецептора)
JPWO2019148044A5 (enExample)
JP2012527487A5 (enExample)
JP2015524843A5 (enExample)
US9266864B2 (en) VEGFR3 inhibitors
WO2014026243A1 (en) Vegfr3 inhibitors
JP2006519221A (ja) 化合物並びに細胞増殖性疾患、網膜症及び関節炎を処置する方法