JP2010502759A - タンパク質物質の経口または直腸投与のための医薬組成物 - Google Patents
タンパク質物質の経口または直腸投与のための医薬組成物 Download PDFInfo
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/282—Organic compounds, e.g. fats
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Immunology (AREA)
- Inorganic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Transplantation (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI20061741 ITMI20061741A1 (it) | 2006-09-12 | 2006-09-12 | Composizioni farmaceutiche per la somministrazione orale di sostanze proteiche |
| ITMI20071205 ITMI20071205A1 (it) | 2007-06-15 | 2007-06-15 | Composizioni farmaceutiche per la somministrazione orale o rettale di sostanze proteiche |
| PCT/EP2007/059378 WO2008031770A2 (en) | 2006-09-12 | 2007-09-07 | Pharmaceutical compositions for the oral or rectal administration of protein substances |
Publications (2)
| Publication Number | Publication Date |
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| JP2010502759A true JP2010502759A (ja) | 2010-01-28 |
| JP2010502759A5 JP2010502759A5 (cg-RX-API-DMAC10.html) | 2010-10-21 |
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| JP2009527791A Pending JP2010502759A (ja) | 2006-09-12 | 2007-09-07 | タンパク質物質の経口または直腸投与のための医薬組成物 |
Country Status (8)
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| US (1) | US20100004157A1 (cg-RX-API-DMAC10.html) |
| EP (1) | EP2081555A2 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2010502759A (cg-RX-API-DMAC10.html) |
| KR (1) | KR20090086060A (cg-RX-API-DMAC10.html) |
| CA (1) | CA2663548A1 (cg-RX-API-DMAC10.html) |
| MX (1) | MX2009002756A (cg-RX-API-DMAC10.html) |
| RU (1) | RU2009113557A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2008031770A2 (cg-RX-API-DMAC10.html) |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017521479A (ja) * | 2014-05-15 | 2017-08-03 | ラニ セラピューティクス， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の薬学的組成物およびそれを製造するための方法 |
| JP2018514563A (ja) * | 2015-05-01 | 2018-06-07 | インキューブ ラブズ， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の製作のための薬学的組成物および方法 |
| JP2019514855A (ja) * | 2016-03-31 | 2019-06-06 | ブイエイチスクエアード リミテッド | 組成物 |
| JP2021506894A (ja) * | 2017-12-22 | 2021-02-22 | コスモ・テクノロジーズ・リミテツド | 固体送達組成物 |
| US11548940B2 (en) | 2014-05-15 | 2023-01-10 | Rani Therapeutics, Llc | Anti-interleukin antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| US12018090B2 (en) | 2014-05-15 | 2024-06-25 | Rani Therapeutics, Llc | PCSK9 antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8809392B2 (en) | 2008-03-28 | 2014-08-19 | Ecolab Usa Inc. | Sulfoperoxycarboxylic acids, their preparation and methods of use as bleaching and antimicrobial agents |
| US12203056B2 (en) | 2008-03-28 | 2025-01-21 | Ecolab Usa Inc. | Sulfoperoxycarboxylic acids, their preparation and methods of use as bleaching and antimicrobial agents |
| GB201017048D0 (en) * | 2010-10-08 | 2010-11-24 | Ucl Business Plc | Composition |
| US10946091B2 (en) * | 2012-06-04 | 2021-03-16 | Gaurav Agrawal | Compositions and methods for treating Crohn's disease and related conditions and infections |
| AU2016239949A1 (en) | 2015-03-31 | 2017-09-07 | Sorriso Pharmaceuticals, Inc. | Peptide construct having a protease-cleavable linker |
| WO2016156468A1 (en) | 2015-03-31 | 2016-10-06 | Vhsquared Limited | Polypeptides |
| EP3294273A4 (en) * | 2015-05-08 | 2018-12-05 | Incube Labs, LLC | Anti-interleukin antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| US11491114B2 (en) | 2016-10-12 | 2022-11-08 | Curioralrx, Llc | Formulations for enteric delivery of therapeutic agents |
| CA3045310A1 (en) * | 2016-12-14 | 2018-06-21 | Progenity, Inc. | Treatment of a disease of the gastrointestinal tract with a chemokine/chemokine receptor inhibitor |
| CA3144566A1 (en) | 2019-06-21 | 2020-12-24 | Sorriso Pharmaceuticals, Inc. | Polypeptides |
| JP7692844B2 (ja) | 2019-06-21 | 2025-06-16 | ソリッソ ファーマシューティカルズ，インク． | ポリペプチド |
| US12570736B2 (en) | 2019-06-21 | 2026-03-10 | Sorriso Pharmaceuticals, Inc. | Compositions |
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| JPH07145068A (ja) * | 1991-08-07 | 1995-06-06 | Yeda Res & Dev Co Ltd | 溶解型ｔｎｆ受容体のマルチマー、その製造方法、およびそれを含有する医薬組成物 |
| JPH10503179A (ja) * | 1994-06-24 | 1998-03-24 | イミュネックス・コーポレーション | 放出制御性ポリペプチド組成物および炎症性腸疾患の治療方法 |
| JP2003501457A (ja) * | 1999-06-14 | 2003-01-14 | コスモ ソシエタ ペル アチオニ | 制御放出および味感遮蔽経口医薬組成物 |
| WO2005027878A1 (en) * | 2003-09-19 | 2005-03-31 | Penwest Pharmaceuticals Co. | Delayed released dosage forms |
| WO2006009764A1 (en) * | 2004-06-17 | 2006-01-26 | Amano Enzyme Usa., Ltd. | Controlled release formulations of enzymes, microorganisms, and antibodies with mucoadhesive polymers |
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| AU2002341321A1 (en) * | 2001-11-30 | 2003-06-10 | Pfizer Products Inc. | Combination of an il-1/18 inhibitor with a tnf inhibitor for the treatment of inflammation |
| ITMI20012599A1 (it) * | 2001-12-11 | 2003-06-11 | Cosmo Spa | Composizioni farmaceutiche per la somministrazione orale di eparina osuoi derivati, utili per la terapia di malattie infiammatorie dell'int |
| US7879361B2 (en) * | 2005-01-04 | 2011-02-01 | Gp Medical, Inc. | Nanoparticles for drug delivery |
| DE602006020123D1 (de) * | 2005-05-04 | 2011-03-31 | Zealand Pharma As | Glucagon-like-peptide-2- (glp-2-) analoga |
-
2007
- 2007-09-07 EP EP07803323A patent/EP2081555A2/en not_active Withdrawn
- 2007-09-07 MX MX2009002756A patent/MX2009002756A/es not_active Application Discontinuation
- 2007-09-07 CA CA002663548A patent/CA2663548A1/en not_active Abandoned
- 2007-09-07 RU RU2009113557/15A patent/RU2009113557A/ru not_active Application Discontinuation
- 2007-09-07 US US12/441,112 patent/US20100004157A1/en not_active Abandoned
- 2007-09-07 WO PCT/EP2007/059378 patent/WO2008031770A2/en not_active Ceased
- 2007-09-07 JP JP2009527791A patent/JP2010502759A/ja active Pending
- 2007-09-07 KR KR1020097007396A patent/KR20090086060A/ko not_active Withdrawn
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| JPH07145068A (ja) * | 1991-08-07 | 1995-06-06 | Yeda Res & Dev Co Ltd | 溶解型ｔｎｆ受容体のマルチマー、その製造方法、およびそれを含有する医薬組成物 |
| JPH10503179A (ja) * | 1994-06-24 | 1998-03-24 | イミュネックス・コーポレーション | 放出制御性ポリペプチド組成物および炎症性腸疾患の治療方法 |
| JP2003501457A (ja) * | 1999-06-14 | 2003-01-14 | コスモ ソシエタ ペル アチオニ | 制御放出および味感遮蔽経口医薬組成物 |
| WO2005027878A1 (en) * | 2003-09-19 | 2005-03-31 | Penwest Pharmaceuticals Co. | Delayed released dosage forms |
| WO2006009764A1 (en) * | 2004-06-17 | 2006-01-26 | Amano Enzyme Usa., Ltd. | Controlled release formulations of enzymes, microorganisms, and antibodies with mucoadhesive polymers |
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| US11026998B2 (en) | 2014-05-15 | 2021-06-08 | Rani Therapeutics, Llc | Shaped mass composition comprising exenatide |
| JP7565688B2 (ja) | 2014-05-15 | 2024-10-11 | ラニ セラピューティクス， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の薬学的組成物およびそれを製造するための方法 |
| JP2020063301A (ja) * | 2014-05-15 | 2020-04-23 | インキューブ ラブズ， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の薬学的組成物およびそれを製造するための方法 |
| US12018090B2 (en) | 2014-05-15 | 2024-06-25 | Rani Therapeutics, Llc | PCSK9 antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| US10953075B2 (en) | 2014-05-15 | 2021-03-23 | Incube Labs, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising anti-interleukin antibodies |
| US11718665B2 (en) | 2014-05-15 | 2023-08-08 | Rani Therapeutics, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising polypeptides and/or proteins |
| JP2021102660A (ja) * | 2014-05-15 | 2021-07-15 | インキューブ ラブズ， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の薬学的組成物およびそれを製造するための方法 |
| US11291709B2 (en) | 2014-05-15 | 2022-04-05 | Rani Therapeutics, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising TNF-inhibiting antibodies |
| US11304993B2 (en) | 2014-05-15 | 2022-04-19 | Rani Therapeutics, Llc | Pharmaceutical compositions and methods for fabrication of solid masses comprising polypeptides and/or proteins |
| US11548940B2 (en) | 2014-05-15 | 2023-01-10 | Rani Therapeutics, Llc | Anti-interleukin antibody preparations for delivery into a lumen of the intestinal tract using a swallowable drug delivery device |
| JP2017521479A (ja) * | 2014-05-15 | 2017-08-03 | ラニ セラピューティクス， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の薬学的組成物およびそれを製造するための方法 |
| JP2018514563A (ja) * | 2015-05-01 | 2018-06-07 | インキューブ ラブズ， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の製作のための薬学的組成物および方法 |
| JP7202070B2 (ja) | 2015-05-01 | 2023-01-11 | ラニ セラピューティクス， エルエルシー | ポリペプチドおよび／またはタンパク質を含む固体塊の製作のための薬学的組成物および方法 |
| JP7224917B2 (ja) | 2016-03-31 | 2023-02-20 | ソリッソ ファーマシューティカルズ，インク． | 組成物 |
| JP2023058591A (ja) * | 2016-03-31 | 2023-04-25 | ソリッソ ファーマシューティカルズ，インク． | 組成物 |
| JP7496906B2 (ja) | 2016-03-31 | 2024-06-07 | ソリッソ ファーマシューティカルズ，インク． | 組成物 |
| JP2019514855A (ja) * | 2016-03-31 | 2019-06-06 | ブイエイチスクエアード リミテッド | 組成物 |
| JP2021506894A (ja) * | 2017-12-22 | 2021-02-22 | コスモ・テクノロジーズ・リミテツド | 固体送達組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20100004157A1 (en) | 2010-01-07 |
| WO2008031770A3 (en) | 2008-09-12 |
| KR20090086060A (ko) | 2009-08-10 |
| CA2663548A1 (en) | 2008-03-20 |
| RU2009113557A (ru) | 2010-10-20 |
| EP2081555A2 (en) | 2009-07-29 |
| WO2008031770A2 (en) | 2008-03-20 |
| MX2009002756A (es) | 2009-05-25 |
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