JP2009533423A5 - - Google Patents

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Publication number
JP2009533423A5
JP2009533423A5 JP2009505314A JP2009505314A JP2009533423A5 JP 2009533423 A5 JP2009533423 A5 JP 2009533423A5 JP 2009505314 A JP2009505314 A JP 2009505314A JP 2009505314 A JP2009505314 A JP 2009505314A JP 2009533423 A5 JP2009533423 A5 JP 2009533423A5
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JP
Japan
Prior art keywords
diol
oxadiazol
nitrobenzene
pharmaceutical composition
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2009505314A
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English (en)
Japanese (ja)
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JP5442434B2 (ja
JP2009533423A (ja
Filing date
Publication date
Priority claimed from EP06007534A external-priority patent/EP1845097A1/en
Application filed filed Critical
Publication of JP2009533423A publication Critical patent/JP2009533423A/ja
Publication of JP2009533423A5 publication Critical patent/JP2009533423A5/ja
Application granted granted Critical
Publication of JP5442434B2 publication Critical patent/JP5442434B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009505314A 2006-04-10 2007-04-10 新規医薬化合物 Active JP5442434B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06007534.8 2006-04-10
EP06007534A EP1845097A1 (en) 2006-04-10 2006-04-10 Oxadiazole derivatives as COMT inhibitors
PCT/PT2007/000016 WO2007117165A1 (en) 2006-04-10 2007-04-10 New pharmaceutical compounds

Publications (3)

Publication Number Publication Date
JP2009533423A JP2009533423A (ja) 2009-09-17
JP2009533423A5 true JP2009533423A5 (enExample) 2010-05-27
JP5442434B2 JP5442434B2 (ja) 2014-03-12

Family

ID=37188829

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009505314A Active JP5442434B2 (ja) 2006-04-10 2007-04-10 新規医薬化合物

Country Status (15)

Country Link
US (2) US8536203B2 (enExample)
EP (3) EP1845097A1 (enExample)
JP (1) JP5442434B2 (enExample)
KR (1) KR20080108327A (enExample)
CN (1) CN101454285B (enExample)
AR (1) AR060421A1 (enExample)
AU (1) AU2007235755A1 (enExample)
BR (1) BRPI0711538A2 (enExample)
CA (1) CA2648914C (enExample)
ES (1) ES2565019T3 (enExample)
MX (1) MX2008013020A (enExample)
NO (1) NO20084712L (enExample)
RU (1) RU2008143670A (enExample)
WO (1) WO2007117165A1 (enExample)
ZA (1) ZA200809479B (enExample)

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EP3303283B1 (en) * 2015-06-23 2021-04-21 National Institute Of Biological Sciences, Beijing Fto inhibitors
US10532976B2 (en) * 2015-06-23 2020-01-14 National Institute Of Biological Sciences, Beijing FTO inhibitors
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US12097193B2 (en) 2018-10-05 2024-09-24 Bial—Portela & Ca, S.A. Methods for the administration of COMT inhibitors
CN112375014A (zh) * 2020-12-17 2021-02-19 重庆柳江医药科技有限公司 一种奥匹卡朋工艺杂质及制备方法和用途
CN116283664B (zh) * 2023-01-12 2025-05-16 中国药科大学 一种硝基儿茶酚衍生物、包含其的药物组合物及其应用
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TR201906117T4 (tr) 2008-07-29 2019-05-21 Bial Portela & Ca Sa Nitrokatesollere yönelik uygulama rejimi.
US20100256194A1 (en) 2009-04-01 2010-10-07 Bial - Portela & Ca, S.A. Pharmaceutical formulations comprising nitrocatechol derivatives and methods of making the same
US9132094B2 (en) 2009-04-01 2015-09-15 Bial—Portela & Ca, S.A. Pharmaceutical formulations comprising nitrocatechol derivatives and methods of making thereof
CN102781424B (zh) 2010-03-04 2016-03-30 奥赖恩公司 左旋多巴、卡比多巴和恩他卡朋用于治疗帕金森病的应用
US20140045900A1 (en) 2011-02-11 2014-02-13 Bial-Portela & Ca, S.A. Administration regime for nitrocatechols
PT2791134T (pt) 2011-12-13 2019-12-18 BIAL PORTELA & Cª S A Composto químico útil como intermediário para a preparação de um inibidor de catecol-o-metiltransferase

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