JP2007532546A5 - - Google Patents

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Publication number
JP2007532546A5
JP2007532546A5 JP2007507409A JP2007507409A JP2007532546A5 JP 2007532546 A5 JP2007532546 A5 JP 2007532546A5 JP 2007507409 A JP2007507409 A JP 2007507409A JP 2007507409 A JP2007507409 A JP 2007507409A JP 2007532546 A5 JP2007532546 A5 JP 2007532546A5
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JP
Japan
Prior art keywords
oxo
oct
amide
isopropyl
azabicyclo
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JP2007507409A
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English (en)
Japanese (ja)
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JP2007532546A (ja
JP4944012B2 (ja
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Priority claimed from PCT/US2005/011393 external-priority patent/WO2005100350A1/en
Publication of JP2007532546A publication Critical patent/JP2007532546A/ja
Publication of JP2007532546A5 publication Critical patent/JP2007532546A5/ja
Application granted granted Critical
Publication of JP4944012B2 publication Critical patent/JP4944012B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2007507409A 2004-04-07 2005-04-06 ５−ｈｔ４レセプターアゴニストとしてのキノリノン−カルボキサミド化合物 Expired - Lifetime JP4944012B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US56007604P 2004-04-07 2004-04-07
US60/560,076 2004-04-07
PCT/US2005/011393 WO2005100350A1 (en) 2004-04-07 2005-04-06 Quinolinone-carboxamide compounds as 5-ht4 receptor agonists

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2008076685A Division JP2008174569A (ja) 2004-04-07 2008-03-24 ５−ｈｔ４レセプターアゴニストとしてのキノリノン−カルボキサミド化合物

Publications (3)

Publication Number Publication Date
JP2007532546A JP2007532546A (ja) 2007-11-15
JP2007532546A5 true JP2007532546A5 (https=) 2008-05-15
JP4944012B2 JP4944012B2 (ja) 2012-05-30

Family

ID=34964334

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2007507409A Expired - Lifetime JP4944012B2 (ja) 2004-04-07 2005-04-06 ５−ｈｔ４レセプターアゴニストとしてのキノリノン−カルボキサミド化合物
JP2008076685A Withdrawn JP2008174569A (ja) 2004-04-07 2008-03-24 ５−ｈｔ４レセプターアゴニストとしてのキノリノン−カルボキサミド化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2008076685A Withdrawn JP2008174569A (ja) 2004-04-07 2008-03-24 ５−ｈｔ４レセプターアゴニストとしてのキノリノン−カルボキサミド化合物

Country Status (28)

Country Link
US (9) US7375114B2 (https=)
EP (1) EP1735304B1 (https=)
JP (2) JP4944012B2 (https=)
KR (1) KR101167296B1 (https=)
CN (1) CN100569771C (https=)
AR (1) AR050407A1 (https=)
AT (1) ATE420088T1 (https=)
AU (1) AU2005233560B2 (https=)
BR (1) BRPI0509761B8 (https=)
CA (1) CA2561558C (https=)
CY (1) CY1108908T1 (https=)
DE (1) DE602005012249D1 (https=)
DK (1) DK1735304T3 (https=)
ES (1) ES2320907T3 (https=)
HR (1) HRP20090162T1 (https=)
IL (1) IL178086A (https=)
MA (1) MA28559B1 (https=)
MX (1) MXPA06011398A (https=)
MY (1) MY155036A (https=)
NO (1) NO337126B1 (https=)
NZ (1) NZ549941A (https=)
PL (1) PL1735304T3 (https=)
PT (1) PT1735304E (https=)
RU (1) RU2394033C2 (https=)
SI (1) SI1735304T1 (https=)
TW (1) TWI351282B (https=)
WO (1) WO2005100350A1 (https=)
ZA (1) ZA200608363B (https=)

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TWI415850B (zh) 2007-07-20 2013-11-21 Theravance Inc 製備ｍｕ類鴉片受體拮抗劑之中間物的方法
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AR086554A1 (es) 2011-05-27 2014-01-08 Novartis Ag Derivados de la piperidina 3-espirociclica como agonistas de receptores de la ghrelina
JP2015525202A (ja) 2012-05-03 2015-09-03 ノバルティス アーゲー グレリン受容体アゴニストとしての２，７−ジアザ−スピロ［４，５］デカ−７−イル誘導体のｌ−リンゴ酸塩およびその結晶形態
KR102692887B1 (ko) * 2017-07-31 2024-08-08 알파시그마 에스.피.에이. 벨루세트라그를 사용하여 위마비 증상을 치료하는 방법
MX2020003242A (es) 2017-09-22 2020-09-18 Jubilant Epipad LLC Compuestos heterociclicos como inhibidores de pad.
AU2018352142B2 (en) 2017-10-18 2022-08-25 Jubilant Epipad LLC Imidazo-pyridine compounds as PAD inhibitors
KR20200085836A (ko) 2017-11-06 2020-07-15 주빌런트 프로델 엘엘씨 Pd1/pd-l1 활성화 억제제로서의 피리미딘 유도체
BR112020010322A2 (pt) 2017-11-24 2020-11-17 Jubilant Episcribe Llc composto da fórmula i; composto da fórmula ia; composto da fórmula ib; processo de preparação de compostos da fórmula i; composição farmacêutica; método para o tratamento e/ou prevenção de várias doenças; uso dos compostos; método para o tratamento de câncer; e método para o tratamento e/ou prevenção de uma afecção mediada por prmt5 ou um distúrbio proliferativo ou câncer
SG11202008950PA (en) 2018-03-13 2020-10-29 Jubilant Prodel LLC Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation
IL314038A (en) 2022-01-11 2024-09-01 Suven Life Sciences Ltd Pyrrolo[1,2-b]-2-pyridazinone compounds as 5-HT4 receptor agonists
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