JP2007514746A5 - - Google Patents

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JP2007514746A5
JP2007514746A5 JP2006545364A JP2006545364A JP2007514746A5 JP 2007514746 A5 JP2007514746 A5 JP 2007514746A5 JP 2006545364 A JP2006545364 A JP 2006545364A JP 2006545364 A JP2006545364 A JP 2006545364A JP 2007514746 A5 JP2007514746 A5 JP 2007514746A5
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group
composition
compound
substituted
disease
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JP2006545364A
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Japanese (ja)
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JP4939229B2 (ja
JP2007514746A (ja
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Priority claimed from PCT/US2004/042060 external-priority patent/WO2005066147A1/en
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Publication of JP2007514746A5 publication Critical patent/JP2007514746A5/ja
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JP2006545364A 2003-12-19 2004-12-16 Cxc−ケモカインレセプターリガンドおよびcc−ケモカインレセプターリガンドとしてのチアジアゾール Expired - Fee Related JP4939229B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53131103P 2003-12-19 2003-12-19
US60/531,311 2003-12-19
US53171303P 2003-12-22 2003-12-22
US60/531,713 2003-12-22
PCT/US2004/042060 WO2005066147A1 (en) 2003-12-19 2004-12-16 Thiadiazoles as cxc- and cc- chemokine receptor ligands

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011030301A Division JP2011093943A (ja) 2003-12-19 2011-02-15 Cxc−ケモカインレセプターリガンドおよびcc−ケモカインレセプターリガンドとしてのチアジアゾール

Publications (3)

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JP2007514746A JP2007514746A (ja) 2007-06-07
JP2007514746A5 true JP2007514746A5 (https=) 2008-02-07
JP4939229B2 JP4939229B2 (ja) 2012-05-23

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JP2006545364A Expired - Fee Related JP4939229B2 (ja) 2003-12-19 2004-12-16 Cxc−ケモカインレセプターリガンドおよびcc−ケモカインレセプターリガンドとしてのチアジアゾール
JP2011030301A Withdrawn JP2011093943A (ja) 2003-12-19 2011-02-15 Cxc−ケモカインレセプターリガンドおよびcc−ケモカインレセプターリガンドとしてのチアジアゾール

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JP2011030301A Withdrawn JP2011093943A (ja) 2003-12-19 2011-02-15 Cxc−ケモカインレセプターリガンドおよびcc−ケモカインレセプターリガンドとしてのチアジアゾール

Country Status (13)

Country Link
US (2) US7338968B2 (https=)
EP (1) EP1694659B8 (https=)
JP (2) JP4939229B2 (https=)
CN (1) CN1918138B (https=)
AR (1) AR046791A1 (https=)
AT (1) ATE406356T1 (https=)
CA (1) CA2550189A1 (https=)
DE (1) DE602004016211D1 (https=)
ES (1) ES2308299T3 (https=)
MX (1) MXPA06007076A (https=)
MY (1) MY139808A (https=)
TW (1) TW200528450A (https=)
WO (1) WO2005066147A1 (https=)

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WO2012068440A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
CA2818542A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
MY165963A (en) 2011-06-20 2018-05-18 Incyte Holdings Corp Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
TW201313721A (zh) 2011-08-18 2013-04-01 Incyte Corp 作為jak抑制劑之環己基氮雜環丁烷衍生物
UA111854C2 (uk) 2011-09-07 2016-06-24 Інсайт Холдінгс Корпорейшн Способи і проміжні сполуки для отримання інгібіторів jak
TW201406761A (zh) 2012-05-18 2014-02-16 Incyte Corp 做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
US8865723B2 (en) 2012-10-25 2014-10-21 Tetra Discovery Partners Llc Selective PDE4 B inhibition and improvement in cognition in subjects with brain injury
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WO2014138168A1 (en) 2013-03-06 2014-09-12 Incyte Corporation Processes and intermediates for making a jak inhibitor
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AR113922A1 (es) 2017-12-08 2020-07-01 Incyte Corp Terapia de combinación de dosis baja para el tratamiento de neoplasias mieloproliferativas
EA202091830A1 (ru) 2018-01-30 2020-12-29 Инсайт Корпорейшн Способы и промежуточные соединения для получения ингибитора jak
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