JP2005527587A5 - - Google Patents

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Publication number
JP2005527587A5
JP2005527587A5 JP2003584051A JP2003584051A JP2005527587A5 JP 2005527587 A5 JP2005527587 A5 JP 2005527587A5 JP 2003584051 A JP2003584051 A JP 2003584051A JP 2003584051 A JP2003584051 A JP 2003584051A JP 2005527587 A5 JP2005527587 A5 JP 2005527587A5
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JP
Japan
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JP2003584051A
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English (en)
Japanese (ja)
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JP2005527587A (ja
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Priority claimed from US10/116,117 external-priority patent/US20030028018A1/en
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Publication of JP2005527587A publication Critical patent/JP2005527587A/ja
Publication of JP2005527587A5 publication Critical patent/JP2005527587A5/ja
Pending legal-status Critical Current

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JP2003584051A 2002-04-05 2003-04-04 キノリノン誘導体 Pending JP2005527587A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/116,117 US20030028018A1 (en) 2000-09-11 2002-04-05 Quinolinone derivatives
PCT/US2003/010463 WO2003087095A1 (en) 2002-04-05 2003-04-04 Quinolinone derivatives

Publications (2)

Publication Number Publication Date
JP2005527587A JP2005527587A (ja) 2005-09-15
JP2005527587A5 true JP2005527587A5 (https=) 2006-06-22

Family

ID=29248193

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003584051A Pending JP2005527587A (ja) 2002-04-05 2003-04-04 キノリノン誘導体

Country Status (24)

Country Link
US (3) US20030028018A1 (https=)
EP (1) EP1497287B1 (https=)
JP (1) JP2005527587A (https=)
KR (1) KR101035894B1 (https=)
CN (1) CN1659165A (https=)
AP (1) AP2070A (https=)
AT (1) ATE489092T1 (https=)
AU (1) AU2003226275B2 (https=)
BR (1) BR0308996A (https=)
CA (1) CA2481055C (https=)
DE (1) DE60335096D1 (https=)
EA (1) EA010393B1 (https=)
EC (1) ECSP045411A (https=)
ES (1) ES2357289T3 (https=)
HR (1) HRP20041031B1 (https=)
IL (2) IL164324A0 (https=)
MA (1) MA28122A1 (https=)
MX (1) MXPA04009739A (https=)
NO (1) NO331021B1 (https=)
NZ (1) NZ536068A (https=)
PL (1) PL209412B1 (https=)
PT (1) PT1497287E (https=)
SG (1) SG143985A1 (https=)
WO (1) WO2003087095A1 (https=)

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JP2015505562A (ja) 2012-01-31 2015-02-23 ノバルティス アーゲー Ｒｔｋ阻害剤と抗エストロゲン剤との組合せ、およびがん治療のためのその使用
US20150202203A1 (en) 2012-07-11 2015-07-23 Novartis Ag Method of Treating Gastrointestinal Stromal Tumors
WO2014058785A1 (en) 2012-10-10 2014-04-17 Novartis Ag Combination therapy
JP6223563B2 (ja) 2013-10-14 2017-11-01 エーザイ・アール・アンド・ディー・マネジメント株式会社 選択的に置換されたキノリン化合物
CN105636945B (zh) 2013-10-14 2017-11-17 卫材R&D管理有限公司 选择性取代的喹啉化合物
LT3157566T (lt) 2014-06-17 2019-08-12 Vertex Pharmaceuticals Incorporated Vėžio gydymo būdas, panaudojant chk1 ir atr inhibitorių derinį
EP2977374A1 (en) 2014-07-21 2016-01-27 Université de Strasbourg Molecules presenting dual emission properties
HK1258570A1 (zh) 2015-09-30 2019-11-15 Vertex Pharmaceuticals Inc. 使用dna损伤剂及atr抑制剂的组合治疗癌症的方法
CN108003150A (zh) * 2016-10-31 2018-05-08 河南工业大学 4-杂芳基喹啉酮衍生物的制备方法及其应用
EP3645526B1 (en) * 2017-06-27 2024-09-04 Janssen Pharmaceutica NV New quinolinone compounds
KR102723359B1 (ko) 2017-11-24 2024-10-28 얀센 파마슈티카 엔브이 피라졸로피리디논 화합물
EP3713941B1 (en) 2017-11-24 2022-06-22 Janssen Pharmaceutica NV Pyrazolopyridinone compounds
CN108516973A (zh) * 2018-03-30 2018-09-11 广西师范大学 3-苯并噻唑-1-(3-二甲氨基)丙基喹啉-4-酮衍生物及其制备方法和应用
MX2021007853A (es) 2018-12-26 2021-08-11 Janssen Pharmaceutica Nv Compuestos de tienopiridinona.

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