JP2005507400A5 - - Google Patents
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- Publication number
- JP2005507400A5 JP2005507400A5 JP2003537607A JP2003537607A JP2005507400A5 JP 2005507400 A5 JP2005507400 A5 JP 2005507400A5 JP 2003537607 A JP2003537607 A JP 2003537607A JP 2003537607 A JP2003537607 A JP 2003537607A JP 2005507400 A5 JP2005507400 A5 JP 2005507400A5
- Authority
- JP
- Japan
- Prior art keywords
- composition
- dosage form
- gabapentin
- composition according
- stomach
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000203 mixture Substances 0.000 claims 45
- UGJMXCAKCUNAIE-UHFFFAOYSA-N Gabapentin Chemical compound OC(=O)CC1(CN)CCCCC1 UGJMXCAKCUNAIE-UHFFFAOYSA-N 0.000 claims 26
- 239000002552 dosage form Substances 0.000 claims 25
- 229960002870 gabapentin Drugs 0.000 claims 13
- 210000002784 stomach Anatomy 0.000 claims 7
- 239000008194 pharmaceutical composition Substances 0.000 claims 5
- 150000003839 salts Chemical class 0.000 claims 5
- 229920003171 Poly (ethylene oxide) Polymers 0.000 claims 2
- 239000003795 chemical substances by application Substances 0.000 claims 2
- 210000001198 duodenum Anatomy 0.000 claims 2
- 235000012054 meals Nutrition 0.000 claims 2
- 210000000813 small intestine Anatomy 0.000 claims 2
- WTDRDQBEARUVNC-LURJTMIESA-N L-DOPA Chemical compound OC(=O)[C@@H](N)CC1=CC=C(O)C(O)=C1 WTDRDQBEARUVNC-LURJTMIESA-N 0.000 claims 1
- WTDRDQBEARUVNC-UHFFFAOYSA-N L-Dopa Natural products OC(=O)C(N)CC1=CC=C(O)C(O)=C1 WTDRDQBEARUVNC-UHFFFAOYSA-N 0.000 claims 1
- 241000124008 Mammalia Species 0.000 claims 1
- 208000019695 Migraine disease Diseases 0.000 claims 1
- 208000016285 Movement disease Diseases 0.000 claims 1
- 239000000853 adhesive Substances 0.000 claims 1
- 230000001070 adhesive effect Effects 0.000 claims 1
- 125000000217 alkyl group Chemical group 0.000 claims 1
- 230000002921 anti-spasmodic effect Effects 0.000 claims 1
- 229940124575 antispasmodic agent Drugs 0.000 claims 1
- 239000002775 capsule Substances 0.000 claims 1
- 239000001913 cellulose Substances 0.000 claims 1
- 229920002678 cellulose Polymers 0.000 claims 1
- 238000004821 distillation Methods 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 206010015037 epilepsy Diseases 0.000 claims 1
- 238000013265 extended release Methods 0.000 claims 1
- 229920001477 hydrophilic polymer Polymers 0.000 claims 1
- 239000001866 hydroxypropyl methyl cellulose Substances 0.000 claims 1
- 229920003088 hydroxypropyl methyl cellulose Polymers 0.000 claims 1
- UFVKGYZPFZQRLF-UHFFFAOYSA-N hydroxypropyl methyl cellulose Chemical compound OC1C(O)C(OC)OC(CO)C1OC1C(O)C(O)C(OC2C(C(O)C(OC3C(C(O)C(O)C(CO)O3)O)C(CO)O2)O)C(CO)O1 UFVKGYZPFZQRLF-UHFFFAOYSA-N 0.000 claims 1
- 235000010979 hydroxypropyl methyl cellulose Nutrition 0.000 claims 1
- 229960004502 levodopa Drugs 0.000 claims 1
- 239000000463 material Substances 0.000 claims 1
- 239000011159 matrix material Substances 0.000 claims 1
- 206010027599 migraine Diseases 0.000 claims 1
- 208000004296 neuralgia Diseases 0.000 claims 1
- 208000021722 neuropathic pain Diseases 0.000 claims 1
- 229940005483 opioid analgesics Drugs 0.000 claims 1
- 229940126701 oral medication Drugs 0.000 claims 1
- 229920000642 polymer Polymers 0.000 claims 1
- 230000002035 prolonged effect Effects 0.000 claims 1
- 238000011321 prophylaxis Methods 0.000 claims 1
- 208000020016 psychiatric disease Diseases 0.000 claims 1
- 239000007939 sustained release tablet Substances 0.000 claims 1
- 239000003826 tablet Substances 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
- 239000003029 tricyclic antidepressant agent Substances 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33524801P | 2001-10-25 | 2001-10-25 | |
| US60/335,248 | 2001-10-25 | ||
| PCT/IB2002/005440 WO2003035040A1 (en) | 2001-10-25 | 2002-10-25 | Methods of treatment using a gastric retained gabapentin dosage |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010179064A Division JP2010254713A (ja) | 2001-10-25 | 2010-08-09 | 胃に留まるガバペンチン投薬を使用する処置方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005507400A JP2005507400A (ja) | 2005-03-17 |
| JP2005507400A5 true JP2005507400A5 (OSRAM) | 2006-01-05 |
| JP5421511B2 JP5421511B2 (ja) | 2014-02-19 |
Family
ID=23310919
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003537607A Expired - Fee Related JP5421511B2 (ja) | 2001-10-25 | 2002-10-25 | 胃に留まるガバペンチン投薬を使用する処置方法 |
| JP2010179064A Pending JP2010254713A (ja) | 2001-10-25 | 2010-08-09 | 胃に留まるガバペンチン投薬を使用する処置方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010179064A Pending JP2010254713A (ja) | 2001-10-25 | 2010-08-09 | 胃に留まるガバペンチン投薬を使用する処置方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (10) | US7438927B2 (OSRAM) |
| EP (2) | EP1439825B2 (OSRAM) |
| JP (2) | JP5421511B2 (OSRAM) |
| AU (1) | AU2002348828B2 (OSRAM) |
| CA (1) | CA2464322C (OSRAM) |
| DK (1) | DK1439825T4 (OSRAM) |
| MX (1) | MXPA04003946A (OSRAM) |
| TW (1) | TWI312285B (OSRAM) |
| WO (1) | WO2003035040A1 (OSRAM) |
Families Citing this family (154)
| Publication number | Priority date | Publication date | Assignee | Title |
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2002
- 2002-10-24 TW TW091124777A patent/TWI312285B/zh not_active IP Right Cessation
- 2002-10-25 EP EP02781665.1A patent/EP1439825B2/en not_active Expired - Lifetime
- 2002-10-25 WO PCT/IB2002/005440 patent/WO2003035040A1/en not_active Ceased
- 2002-10-25 EP EP10179051A patent/EP2266539A3/en not_active Withdrawn
- 2002-10-25 MX MXPA04003946A patent/MXPA04003946A/es active IP Right Grant
- 2002-10-25 DK DK02781665.1T patent/DK1439825T4/en active
- 2002-10-25 JP JP2003537607A patent/JP5421511B2/ja not_active Expired - Fee Related
- 2002-10-25 CA CA2464322A patent/CA2464322C/en not_active Expired - Lifetime
- 2002-10-25 AU AU2002348828A patent/AU2002348828B2/en not_active Ceased
-
2003
- 2003-01-22 US US10/280,309 patent/US7438927B2/en not_active Expired - Lifetime
-
2008
- 2008-09-26 US US12/239,591 patent/US7731989B2/en not_active Expired - Fee Related
-
2010
- 2010-03-29 US US12/749,101 patent/US8252332B2/en not_active Expired - Fee Related
- 2010-08-09 JP JP2010179064A patent/JP2010254713A/ja active Pending
-
2011
- 2011-05-19 US US13/111,575 patent/US8192756B2/en not_active Expired - Fee Related
- 2011-11-21 US US13/301,644 patent/US8231905B2/en not_active Expired - Fee Related
-
2012
- 2012-02-14 US US13/396,441 patent/US8409613B2/en not_active Expired - Fee Related
- 2012-07-19 US US13/553,622 patent/US8333991B2/en not_active Expired - Fee Related
- 2012-07-27 US US13/560,938 patent/US8333992B2/en not_active Expired - Fee Related
-
2013
- 2013-04-01 US US13/854,433 patent/US8580303B2/en not_active Expired - Fee Related
- 2013-11-08 US US14/075,965 patent/US20140072623A1/en not_active Abandoned
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