JP2004517037A - 修飾された形の薬理活性薬物およびそれらの用途 - Google Patents

修飾された形の薬理活性薬物およびそれらの用途 Download PDF

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JP2004517037A
JP2004517037A JP2002504950A JP2002504950A JP2004517037A JP 2004517037 A JP2004517037 A JP 2004517037A JP 2002504950 A JP2002504950 A JP 2002504950A JP 2002504950 A JP2002504950 A JP 2002504950A JP 2004517037 A JP2004517037 A JP 2004517037A
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compound
nsaid
sulfur
subject
disease
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JP2004517037A5 (https=
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− サン ライ、チン
ワン、ティンミン
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メデイノックス,インコーポレイテッド
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/555Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound pre-targeting systems involving an organic compound, other than a peptide, protein or antibody, for targeting specific cells
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63Esters of sulfonic acids
    • C07C309/72Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/73Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton to carbon atoms of non-condensed six-membered aromatic rings
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JP2002504950A 2000-06-23 2001-06-19 修飾された形の薬理活性薬物およびそれらの用途 Pending JP2004517037A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US09/602,688 US6355666B1 (en) 2000-06-23 2000-06-23 Protected forms of pharmacologically active agents and uses therefor
US09/715,767 US6429223B1 (en) 2000-06-23 2000-11-17 Modified forms of pharmacologically active agents and uses therefor
PCT/US2001/019750 WO2002000167A2 (en) 2000-06-23 2001-06-19 Modified forms of pharmacologically active agents and uses therefor

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JP2004517037A true JP2004517037A (ja) 2004-06-10
JP2004517037A5 JP2004517037A5 (https=) 2012-02-23

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US (2) US6429223B1 (https=)
EP (2) EP2261200A3 (https=)
JP (1) JP2004517037A (https=)
KR (2) KR100898646B1 (https=)
CN (1) CN1441770B (https=)
AT (1) ATE486840T1 (https=)
AU (2) AU2001270010C1 (https=)
CA (1) CA2414150A1 (https=)
DE (1) DE60143393D1 (https=)
ES (1) ES2355708T3 (https=)
TW (1) TWI309166B (https=)
WO (1) WO2002000167A2 (https=)

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JP2009280595A (ja) * 2006-06-27 2009-12-03 Takeda Chem Ind Ltd 縮合環化合物
JP2010529101A (ja) * 2007-06-04 2010-08-26 テックフィールズ インコーポレイテッド 非常に速い皮膚及び膜浸透速度を有するnsaiaプロドラッグ及びその新規医薬使用
JP2013147515A (ja) * 2013-05-08 2013-08-01 Techfields Inc 非常に速い皮膚及び膜浸透速度を有するnsaiaプロドラッグ及びその新規医薬使用
JP2015120703A (ja) * 2015-01-05 2015-07-02 テックフィールズ インコーポレイテッド 非常に速い皮膚及び膜浸透速度を有するnsaiaプロドラッグ及びその新規医薬使用
JP2015527309A (ja) * 2012-07-03 2015-09-17 セリックスビオ プライヴェート リミテッド 中等度から重度の疼痛の治療のための組成物及び方法
JP2019011336A (ja) * 2018-09-05 2019-01-24 テックフィールズ インコーポレイテッド 非常に速い皮膚及び膜浸透速度を有するnsaiaプロドラッグ及びその新規医薬使用
JP2019524814A (ja) * 2016-08-12 2019-09-05 オレゴン ヘルス アンド サイエンス ユニバーシティ アミド化合物、その医薬組成物、及びその使用方法
JP2021513547A (ja) * 2018-02-14 2021-05-27 オレゴン ヘルス アンド サイエンス ユニバーシティ ソベチロムの誘導体
US11667606B2 (en) 2019-03-01 2023-06-06 Autobahn Therapeutics, Inc. Thyromimetics
US11827596B2 (en) 2018-12-12 2023-11-28 Autobahn Therapeutics, Inc. Thyromimetics
US12466781B2 (en) 2019-11-29 2025-11-11 Autobahn Therapeutics, Inc. Thyromimetics
US12528761B2 (en) 2020-06-17 2026-01-20 Autobahn Therapeutics, Inc. Thyromimetics
US12590072B2 (en) 2020-06-17 2026-03-31 Autobahn Therapeutics, Inc. Thyromimetics

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