KR20080071628A - 변형된 형태의 약학상 활성 제제 및 그의 용도 - Google Patents

변형된 형태의 약학상 활성 제제 및 그의 용도 Download PDF

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KR20080071628A
KR20080071628A KR1020087017854A KR20087017854A KR20080071628A KR 20080071628 A KR20080071628 A KR 20080071628A KR 1020087017854 A KR1020087017854 A KR 1020087017854A KR 20087017854 A KR20087017854 A KR 20087017854A KR 20080071628 A KR20080071628 A KR 20080071628A
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compound
mmol
substituted
nsaid
scheme
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Korean (ko)
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칭-산 레이
팅민 왕
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메디녹스, 인크.
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Priority claimed from US09/602,688 external-priority patent/US6355666B1/en
Application filed by 메디녹스, 인크. filed Critical 메디녹스, 인크.
Publication of KR20080071628A publication Critical patent/KR20080071628A/ko
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    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63Esters of sulfonic acids
    • C07C309/72Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/73Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton to carbon atoms of non-condensed six-membered aromatic rings
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
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  • Epidemiology (AREA)
  • Cardiology (AREA)
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KR1020087017854A 2000-06-23 2001-06-19 변형된 형태의 약학상 활성 제제 및 그의 용도 Ceased KR20080071628A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US09/602,688 US6355666B1 (en) 2000-06-23 2000-06-23 Protected forms of pharmacologically active agents and uses therefor
US09/602,688 2000-06-23
US09/715,767 2000-11-17
US09/715,767 US6429223B1 (en) 2000-06-23 2000-11-17 Modified forms of pharmacologically active agents and uses therefor

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020027017468A Division KR100898646B1 (ko) 2000-06-23 2001-06-19 변형된 형태의 약학상 활성 제제 및 그의 용도

Publications (1)

Publication Number Publication Date
KR20080071628A true KR20080071628A (ko) 2008-08-04

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Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020087017854A Ceased KR20080071628A (ko) 2000-06-23 2001-06-19 변형된 형태의 약학상 활성 제제 및 그의 용도
KR1020027017468A Expired - Fee Related KR100898646B1 (ko) 2000-06-23 2001-06-19 변형된 형태의 약학상 활성 제제 및 그의 용도

Family Applications After (1)

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KR1020027017468A Expired - Fee Related KR100898646B1 (ko) 2000-06-23 2001-06-19 변형된 형태의 약학상 활성 제제 및 그의 용도

Country Status (12)

Country Link
US (2) US6429223B1 (https=)
EP (2) EP2261200A3 (https=)
JP (1) JP2004517037A (https=)
KR (2) KR20080071628A (https=)
CN (1) CN1441770B (https=)
AT (1) ATE486840T1 (https=)
AU (2) AU7001001A (https=)
CA (1) CA2414150A1 (https=)
DE (1) DE60143393D1 (https=)
ES (1) ES2355708T3 (https=)
TW (1) TWI309166B (https=)
WO (1) WO2002000167A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024177378A1 (ko) * 2023-02-24 2024-08-29 애니머스큐어 주식회사 디플루니살 또는 이의 약학적으로 허용가능한 염을 포함하는 암 악액질 치용 조성물

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US6716452B1 (en) * 2000-08-22 2004-04-06 New River Pharmaceuticals Inc. Active agent delivery systems and methods for protecting and administering active agents
KR20030046389A (ko) * 2000-09-01 2003-06-12 그리폰 테라퓨틱스, 인코포레이티드 친핵체에 안정한 티오에스테르 발생 화합물, 제조 및 사용방법
US8394813B2 (en) 2000-11-14 2013-03-12 Shire Llc Active agent delivery systems and methods for protecting and administering active agents
US7169752B2 (en) 2003-09-30 2007-01-30 New River Pharmaceuticals Inc. Compounds and compositions for prevention of overdose of oxycodone
US20060014697A1 (en) 2001-08-22 2006-01-19 Travis Mickle Pharmaceutical compositions for prevention of overdose or abuse
AU2002365372A1 (en) * 2001-11-27 2003-06-10 Astrazeneca Ab New process
TW200400963A (en) 2002-05-21 2004-01-16 Wyeth Corp R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease
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