CN1441770B - 药学活性剂的修饰型及其应用 - Google Patents

药学活性剂的修饰型及其应用 Download PDF

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Publication number
CN1441770B
CN1441770B CN018115721A CN01811572A CN1441770B CN 1441770 B CN1441770 B CN 1441770B CN 018115721 A CN018115721 A CN 018115721A CN 01811572 A CN01811572 A CN 01811572A CN 1441770 B CN1441770 B CN 1441770B
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substituted
compound
purposes
inflammatory drug
nonsteroidal anti
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Expired - Fee Related
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CN018115721A
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Chinese (zh)
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CN1441770A (zh
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赖青山
T·王
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Medinox Inc
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Medinox Inc
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    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
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CN018115721A 2000-06-23 2001-06-19 药学活性剂的修饰型及其应用 Expired - Fee Related CN1441770B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US09/602,688 2000-06-23
US09/602,688 US6355666B1 (en) 2000-06-23 2000-06-23 Protected forms of pharmacologically active agents and uses therefor
US09/715,767 2000-11-17
US09/715,767 US6429223B1 (en) 2000-06-23 2000-11-17 Modified forms of pharmacologically active agents and uses therefor
PCT/US2001/019750 WO2002000167A2 (en) 2000-06-23 2001-06-19 Modified forms of pharmacologically active agents and uses therefor

Publications (2)

Publication Number Publication Date
CN1441770A CN1441770A (zh) 2003-09-10
CN1441770B true CN1441770B (zh) 2012-03-21

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US (2) US6429223B1 (https=)
EP (2) EP2261200A3 (https=)
JP (1) JP2004517037A (https=)
KR (2) KR100898646B1 (https=)
CN (1) CN1441770B (https=)
AT (1) ATE486840T1 (https=)
AU (2) AU2001270010C1 (https=)
CA (1) CA2414150A1 (https=)
DE (1) DE60143393D1 (https=)
ES (1) ES2355708T3 (https=)
TW (1) TWI309166B (https=)
WO (1) WO2002000167A2 (https=)

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US8394813B2 (en) 2000-11-14 2013-03-12 Shire Llc Active agent delivery systems and methods for protecting and administering active agents
US7169752B2 (en) 2003-09-30 2007-01-30 New River Pharmaceuticals Inc. Compounds and compositions for prevention of overdose of oxycodone
US20060014697A1 (en) 2001-08-22 2006-01-19 Travis Mickle Pharmaceutical compositions for prevention of overdose or abuse
WO2003045896A1 (en) * 2001-11-27 2003-06-05 Astrazeneca Ab New process
TW200400963A (en) * 2002-05-21 2004-01-16 Wyeth Corp R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease
CA2491127A1 (en) * 2002-07-03 2004-01-15 Nitromed, Inc. Nitrosated nonsteroidal antiinflammatory compounds, compositions and methods of use
AU2003261281A1 (en) * 2002-07-29 2004-02-16 Nicox S.A. Cyclooxygenase- 2 selective inhibitors, compositions and methods of use
ITMI20021861A1 (it) * 2002-08-29 2004-02-29 Nicox Sa Procedimento di sintesi di nitrossialchilesteri di acidi carbossilici, intermedi impiegabili in detto procedimento e loro preparazione.
KR20050074493A (ko) * 2002-10-21 2005-07-18 라모트 앳 텔-아비브 유니버시티 리미티드 칼륨 채널 및/또는 피질 뉴우런 작용 조절제로서 유용한n-페닐안트라닐산 및/또는 2-벤즈이미다졸론의 유도체
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