JP2003531173A5 - - Google Patents
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- Publication number
- JP2003531173A5 JP2003531173A5 JP2001577956A JP2001577956A JP2003531173A5 JP 2003531173 A5 JP2003531173 A5 JP 2003531173A5 JP 2001577956 A JP2001577956 A JP 2001577956A JP 2001577956 A JP2001577956 A JP 2001577956A JP 2003531173 A5 JP2003531173 A5 JP 2003531173A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19929800P | 2000-04-24 | 2000-04-24 | |
| US60/199,298 | 2000-04-24 | ||
| US20602500P | 2000-05-22 | 2000-05-22 | |
| US60/206,025 | 2000-05-22 | ||
| US22536400P | 2000-08-14 | 2000-08-14 | |
| US60/225,364 | 2000-08-14 | ||
| PCT/US2001/013175 WO2001080857A1 (en) | 2000-04-24 | 2001-04-24 | Zolpidem hemitartrate |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006033099A Division JP2006137778A (ja) | 2000-04-24 | 2006-02-09 | ゾルピデムヘミタートレイト |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2003531173A JP2003531173A (ja) | 2003-10-21 |
| JP2003531173A5 true JP2003531173A5 (https=) | 2005-12-22 |
Family
ID=27394001
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001577956A Withdrawn JP2003531173A (ja) | 2000-04-24 | 2001-04-24 | ゾルピデムヘミタートレイト |
| JP2006033099A Pending JP2006137778A (ja) | 2000-04-24 | 2006-02-09 | ゾルピデムヘミタートレイト |
| JP2006177160A Pending JP2006249105A (ja) | 2000-04-24 | 2006-06-27 | ゾルピデムヘミタートレイト |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006033099A Pending JP2006137778A (ja) | 2000-04-24 | 2006-02-09 | ゾルピデムヘミタートレイト |
| JP2006177160A Pending JP2006249105A (ja) | 2000-04-24 | 2006-06-27 | ゾルピデムヘミタートレイト |
Country Status (21)
| Country | Link |
|---|---|
| US (8) | US20020077332A1 (https=) |
| EP (1) | EP1292304B1 (https=) |
| JP (3) | JP2003531173A (https=) |
| KR (1) | KR20030069796A (https=) |
| AT (4) | ATE335481T1 (https=) |
| AU (2) | AU5721301A (https=) |
| CA (1) | CA2406982A1 (https=) |
| CZ (1) | CZ20023775A3 (https=) |
| DE (7) | DE04010651T1 (https=) |
| DK (1) | DK1292304T3 (https=) |
| ES (4) | ES2238941T3 (https=) |
| HR (1) | HRP20020909A2 (https=) |
| HU (1) | HUP0300701A2 (https=) |
| IL (1) | IL152411A0 (https=) |
| NZ (1) | NZ522015A (https=) |
| PL (1) | PL358548A1 (https=) |
| PT (3) | PT1541146E (https=) |
| SE (1) | SE5292304T3 (https=) |
| SK (1) | SK16372002A3 (https=) |
| WO (1) | WO2001080857A1 (https=) |
| YU (1) | YU79402A (https=) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2001284322A1 (en) | 2000-08-29 | 2002-03-13 | Ranbaxy Laboratories Limited | Synthesis of n,n-dimethyl-3-(4-methyl) benzoyl propionamide, a key intermediate of zolpidem |
| US6869970B2 (en) | 2002-02-04 | 2005-03-22 | Novartis Ag | Crystalline salt forms of valsartan |
| EP1575952B1 (en) | 2002-12-18 | 2009-02-18 | Mallinckrodt Inc. | Synthesis of heteroaryl acetamides |
| WO2004087703A1 (en) * | 2003-03-12 | 2004-10-14 | Sun Pharmaceutical Industries Limited | Process for the preparation of n,n,6-trimethyl-2-(4-methylphenyl)-imidazo[1,2-a]pyridine-3-acetamide |
| WO2005010002A1 (en) * | 2003-07-31 | 2005-02-03 | Ranbaxy Laboratories Limited | Process for the synthesis of zolpidem |
| JP5179757B2 (ja) * | 2004-02-17 | 2013-04-10 | トランセプト ファーマシューティカルズ， インコーポレイティド | 口腔粘膜を介して催眠剤をデリバリーするための組成物及びその使用方法 |
| WO2006008636A2 (en) * | 2004-07-16 | 2006-01-26 | Ranbaxy Laboratories Limited | Processes for the preparation of zolpidem and its hemitartrate |
| US20070287740A1 (en) * | 2005-05-25 | 2007-12-13 | Transcept Pharmaceuticals, Inc. | Compositions and methods of treating middle-of-the night insomnia |
| US20070225322A1 (en) * | 2005-05-25 | 2007-09-27 | Transoral Pharmaceuticals, Inc. | Compositions and methods for treating middle-of-the night insomnia |
| EP1883408A4 (en) * | 2005-05-25 | 2009-11-11 | Transcept Pharmaceuticals Inc | SOLID COMPOSITIONS AND METHODS FOR TREATMENT OF INSOMNIA IN THE NIGHT |
| KR20080038416A (ko) * | 2005-08-19 | 2008-05-06 | 아벤티스 파마슈티칼스 인크. | 수면제와 치환된 비스 아릴 및 헤테로아릴 화합물의 배합물및 이의 치료요법적 용도 |
| AU2006283702A1 (en) * | 2005-08-19 | 2007-03-01 | Aventis Pharmaceuticals Inc. | Comination of a hypnotic agent and R(+)-alpha-(2,3-dimethoxy-phenyl)-1-(2-(4-fluorophenl)ethyl)-4-piperidinemethanol and therapeutic application thereof |
| EP1948655A1 (en) * | 2005-10-03 | 2008-07-30 | Mallinckrodt, Inc. | Process for preparing zolpidem hemitartrate and tartrate polymorphs |
| WO2007047047A2 (en) * | 2005-10-17 | 2007-04-26 | Mallinckrodt Inc. | Polymorph transformation of zolpidem in tablet matrix |
| US20070098788A1 (en) * | 2005-10-28 | 2007-05-03 | Gore Subhash P | Non-benzodiazepine hypnotic compositions |
| WO2007117399A2 (en) | 2006-03-31 | 2007-10-18 | Janssen Pharmaceutica N.V. | Benzoimidazol-2-yl pyrimidines and pyrazines as modulators of the histamine h4 receptor |
| WO2008067549A2 (en) * | 2006-11-30 | 2008-06-05 | Transcept Pharmaceuticals, Inc. | Stabilized zolpidem pharmaceutical compositions |
| US20080145425A1 (en) * | 2006-12-15 | 2008-06-19 | Pliva Research & Development Limited | Pharmaceutical composition of zolpidem |
| US9371311B2 (en) | 2008-06-30 | 2016-06-21 | Janssen Pharmaceutica Nv | Benzoimidazol-2-yl pyrimidine derivatives |
| SG192446A1 (en) * | 2008-06-30 | 2013-08-30 | Janssen Pharmaceutica Nv | Process for the preparation of benzoimidazol-2-yl pyrimidine derivatives |
| WO2011066352A1 (en) | 2009-11-27 | 2011-06-03 | Genzyme Corporation | An amorphous and a crystalline form of genz 112638 hemitartrat as inhibitor of glucosylceramide synthase |
| WO2011115069A1 (ja) * | 2010-03-19 | 2011-09-22 | 第一三共株式会社 | 結晶の網羅的探索 |
| PT2964229T (pt) | 2013-03-06 | 2020-03-23 | Janssen Pharmaceutica Nv | Moduladores de piridina benzimidazol-2-ilo do recetor h4 de histamina |
| CN116283957A (zh) * | 2021-12-03 | 2023-06-23 | 山东新时代药业有限公司 | 唑吡坦水合物及其制备方法 |
| CN116283958B (zh) * | 2021-12-03 | 2026-02-24 | 山东新时代药业有限公司 | 唑吡坦共晶体及其制备方法 |
| CN117907368A (zh) * | 2024-01-27 | 2024-04-19 | 鲁南贝特制药有限公司 | 一种酒石酸唑吡坦药用晶型d中晶型a、e的定量测定方法 |
| CN118750459B (zh) * | 2024-07-22 | 2025-04-01 | 常州市武进中医医院 | 一种酒石酸唑吡坦片及其制备方法 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4151273A (en) * | 1974-10-31 | 1979-04-24 | The Regents Of The University Of California | Increasing the absorption rate of insoluble drugs |
| FR2408345A1 (fr) * | 1976-11-30 | 1979-06-08 | Besins Jean Louis | Nouvelle composition a action anti-conceptionnelle |
| US4302446A (en) * | 1979-10-02 | 1981-11-24 | Bristol-Myers Company | Pharmaceutical compositions |
| IT1130924B (it) * | 1980-03-06 | 1986-06-18 | Secifarma Spa | Procedimento per la preparazione di spironolattone micronizzato |
| DE3018940A1 (de) * | 1980-05-17 | 1981-11-26 | Hoechst Ag, 6000 Frankfurt | Verwendung eines vinylchlorid-pfropf-copolymerisates in der plastisolverarbeitung |
| FR2492382A1 (fr) * | 1980-10-22 | 1982-04-23 | Synthelabo | Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique |
| FR2525601A1 (fr) * | 1982-04-21 | 1983-10-28 | Synthelabo | Derives d'imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique |
| US4675323A (en) * | 1985-08-06 | 1987-06-23 | Synthelabo | Imidazo(1,2-a)quinoline derivatives useful as anxiolytic agents |
| SE457326B (sv) * | 1986-02-14 | 1988-12-19 | Lejus Medical Ab | Foerfarande foer framstaellning av en snabbt soenderfallande kaerna innehaallande bl a mikrokristallin cellulosa |
| FR2600650B1 (fr) * | 1986-06-27 | 1988-09-09 | Synthelabo | Procede de preparation d'imidazopyridines et composes intermediaires |
| FR2606410B1 (fr) * | 1986-11-07 | 1989-02-24 | Synthelabo | Imidazopyridines, leur preparation et leur application en therapeutique |
| EP0289371B1 (fr) * | 1987-03-27 | 1991-09-25 | Synthelabo | Dérivés d'imidazopyridines, leur préparation et leur application en thérapeutique |
| US5271944A (en) * | 1991-04-05 | 1993-12-21 | Biofor, Ltd. | Pharmacologically enhanced formulations |
| IT1276522B1 (it) * | 1995-04-07 | 1997-10-31 | Elena Benincasa | Uso dello zolpidem per il trattamento terapeudico di sindromi neuropsichiatriche associate a disfunsione e di circuiti neurali dei |
| PT1038875E (pt) * | 1999-03-25 | 2003-10-31 | Synthon Bv | Derivados de imidazopiridina e processo para os preparar |
| ATE297924T1 (de) * | 1999-03-25 | 2005-07-15 | Synthon Bv | Zolpidem salze |
| WO2001042239A1 (en) * | 1999-12-13 | 2001-06-14 | Sumika Fine Chemicals Co., Ltd. | Process for the preparation of a pyridinemethanol compound |
-
2001
- 2001-04-24 CZ CZ20023775A patent/CZ20023775A3/cs unknown
- 2001-04-24 SK SK1637-2002A patent/SK16372002A3/sk not_active Application Discontinuation
- 2001-04-24 DE DE04010651T patent/DE04010651T1/de active Pending
- 2001-04-24 DE DE04010435T patent/DE04010435T1/de active Pending
- 2001-04-24 WO PCT/US2001/013175 patent/WO2001080857A1/en not_active Ceased
- 2001-04-24 AT AT04010435T patent/ATE335481T1/de not_active IP Right Cessation
- 2001-04-24 ES ES04010435T patent/ES2238941T3/es not_active Expired - Lifetime
- 2001-04-24 ES ES05001922T patent/ES2277301T3/es not_active Expired - Lifetime
- 2001-04-24 DE DE60122216T patent/DE60122216T2/de not_active Expired - Fee Related
- 2001-04-24 DE DE60114617T patent/DE60114617T2/de not_active Expired - Fee Related
- 2001-04-24 DE DE20122435U patent/DE20122435U1/de not_active Expired - Lifetime
- 2001-04-24 HU HU0300701A patent/HUP0300701A2/hu unknown
- 2001-04-24 AT AT01930705T patent/ATE308324T1/de not_active IP Right Cessation
- 2001-04-24 AU AU5721301A patent/AU5721301A/xx active Pending
- 2001-04-24 DE DE60125429T patent/DE60125429T2/de not_active Expired - Fee Related
- 2001-04-24 AU AU2001257213A patent/AU2001257213B2/en not_active Ceased
- 2001-04-24 CA CA002406982A patent/CA2406982A1/en not_active Abandoned
- 2001-04-24 US US09/841,025 patent/US20020077332A1/en not_active Abandoned
- 2001-04-24 YU YU79402A patent/YU79402A/sh unknown
- 2001-04-24 NZ NZ522015A patent/NZ522015A/en unknown
- 2001-04-24 PT PT05001922T patent/PT1541146E/pt unknown
- 2001-04-24 DE DE60122944T patent/DE60122944T2/de not_active Expired - Fee Related
- 2001-04-24 JP JP2001577956A patent/JP2003531173A/ja not_active Withdrawn
- 2001-04-24 ES ES04010651T patent/ES2239558T3/es not_active Expired - Lifetime
- 2001-04-24 PT PT04010651T patent/PT1475093E/pt unknown
- 2001-04-24 PL PL01358548A patent/PL358548A1/xx not_active Application Discontinuation
- 2001-04-24 DK DK01930705T patent/DK1292304T3/da active
- 2001-04-24 ES ES01930705T patent/ES2248321T3/es not_active Expired - Lifetime
- 2001-04-24 IL IL15241101A patent/IL152411A0/xx unknown
- 2001-04-24 KR KR1020027014220A patent/KR20030069796A/ko not_active Ceased
- 2001-04-24 EP EP01930705A patent/EP1292304B1/en not_active Revoked
- 2001-04-24 AT AT05001922T patent/ATE348613T1/de not_active IP Right Cessation
- 2001-04-24 AT AT04010651T patent/ATE338550T1/de not_active IP Right Cessation
- 2001-04-24 PT PT04010435T patent/PT1473036E/pt unknown
- 2001-04-24 SE SE01930705T patent/SE5292304T3/xx unknown
- 2001-04-24 HR HR20020909A patent/HRP20020909A2/hr not_active Application Discontinuation
-
2004
- 2004-05-24 US US10/853,345 patent/US20040220213A1/en not_active Abandoned
- 2004-05-24 US US10/852,912 patent/US20040214858A1/en not_active Abandoned
- 2004-05-24 US US10/853,031 patent/US20040220210A1/en not_active Abandoned
- 2004-05-24 US US10/853,033 patent/US20040220211A1/en not_active Abandoned
- 2004-05-24 US US10/853,640 patent/US20040214859A1/en not_active Abandoned
- 2004-05-24 US US10/853,338 patent/US20040220212A1/en not_active Abandoned
-
2006
- 2006-02-09 JP JP2006033099A patent/JP2006137778A/ja active Pending
- 2006-06-27 JP JP2006177160A patent/JP2006249105A/ja active Pending
- 2006-10-25 US US11/588,122 patent/US20070037843A1/en not_active Abandoned