IN2012DN04949A - - Google Patents

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Publication number
IN2012DN04949A
IN2012DN04949A IN4949DEN2012A IN2012DN04949A IN 2012DN04949 A IN2012DN04949 A IN 2012DN04949A IN 4949DEN2012 A IN4949DEN2012 A IN 4949DEN2012A IN 2012DN04949 A IN2012DN04949 A IN 2012DN04949A
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India
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hif
activity
conditions
syndromes related
diseases
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English (en)
Inventor
Robert Shalwitz
Joseph H Gardner
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Aerpio Therapeutics Inc
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Publication of IN2012DN04949A publication Critical patent/IN2012DN04949A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/92—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with a hetero atom directly attached to the ring nitrogen atom
    • C07D211/96—Sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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US20150157617A1 (en) 2015-06-11
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ZA201204104B (en) 2013-02-27
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IL219610A0 (en) 2012-07-31
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CA2774046A1 (en) 2011-05-12
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HK1190334A1 (en) 2014-07-04
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US10562854B2 (en) 2020-02-18
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US8999971B2 (en) 2015-04-07
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