IL92055A - 3-(cycloalkyl substituted 1,2,4-oxadiazolyl)-4,5-dihydro-4-oxo-5- tertbutyl-imidaz (1,5-a) quinoxalines - Google Patents

3-(cycloalkyl substituted 1,2,4-oxadiazolyl)-4,5-dihydro-4-oxo-5- tertbutyl-imidaz (1,5-a) quinoxalines

Info

Publication number
IL92055A
IL92055A IL9205589A IL9205589A IL92055A IL 92055 A IL92055 A IL 92055A IL 9205589 A IL9205589 A IL 9205589A IL 9205589 A IL9205589 A IL 9205589A IL 92055 A IL92055 A IL 92055A
Authority
IL
Israel
Prior art keywords
oxo
dihydro
compound
tert
binding
Prior art date
Application number
IL9205589A
Other languages
English (en)
Other versions
IL92055A0 (en
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of IL92055A0 publication Critical patent/IL92055A0/xx
Publication of IL92055A publication Critical patent/IL92055A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL9205589A 1988-11-10 1989-10-19 3-(cycloalkyl substituted 1,2,4-oxadiazolyl)-4,5-dihydro-4-oxo-5- tertbutyl-imidaz (1,5-a) quinoxalines IL92055A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK626288A DK626288D0 (da) 1988-11-10 1988-11-10 Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen

Publications (2)

Publication Number Publication Date
IL92055A0 IL92055A0 (en) 1990-07-12
IL92055A true IL92055A (en) 1994-01-25

Family

ID=8148369

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9205589A IL92055A (en) 1988-11-10 1989-10-19 3-(cycloalkyl substituted 1,2,4-oxadiazolyl)-4,5-dihydro-4-oxo-5- tertbutyl-imidaz (1,5-a) quinoxalines

Country Status (17)

Country Link
US (1) US4999353A (el)
EP (1) EP0368652B1 (el)
JP (1) JPH02178285A (el)
AT (1) ATE119162T1 (el)
AU (1) AU622941B2 (el)
CA (1) CA2002624A1 (el)
DE (1) DE68921418T2 (el)
DK (1) DK626288D0 (el)
ES (1) ES2068903T3 (el)
FI (1) FI92931C (el)
GR (1) GR3015718T3 (el)
IE (1) IE68939B1 (el)
IL (1) IL92055A (el)
NO (1) NO173827C (el)
NZ (1) NZ231321A (el)
PT (1) PT92279B (el)
ZA (1) ZA898051B (el)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK588489D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
AU657986B2 (en) * 1991-06-14 1995-03-30 Pharmacia & Upjohn Company Imidazo(1,5-a)quinoxalines
WO1993012113A1 (en) * 1991-12-17 1993-06-24 The Upjohn Company 3-SUBSTITUTED IMIDAZO (1,5-a) AND IMIDAZO (1,5-a)-TRIAZOLO (1,5-c) QUINOXALINES AND QUINAZOLINES WITH CNS ACTIVITY
DE4228095A1 (de) * 1992-08-24 1994-03-03 Asta Medica Ag Neue 4,5-Dihydro-4-oxo-pyrrolo[1,2-a]chinoxaline und entsprechende Aza-analoga und Verfahren zu deren Herstellung
FR2696466B1 (fr) * 1992-10-02 1994-11-25 Rhone Poulenc Rorer Sa Dérivés de 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, leur préparation et les médicaments les contenant.
US5792766A (en) 1996-03-13 1998-08-11 Neurogen Corporation Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands
JP4042925B2 (ja) * 1996-11-20 2008-02-06 シスメックス株式会社 幼若白血球の分類計数法
US20040180898A1 (en) * 2003-03-03 2004-09-16 Bang-Chi Chen Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazoquinoxalines and heterocyclic-substituted imidazopyrazines
BR112018010216B1 (pt) 2015-11-20 2024-02-15 Forma Therapeutics, Inc Purinonas como inibidores da protease específica da ubiquitina 1 e composição farmacêutica compreendendo os referidos compostos

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
ES2011448B3 (es) * 1985-10-17 1990-01-16 As Ferrosan Preparacion de un compuesto heterocido y uso del mismo
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
US4999353A (en) 1991-03-12
DE68921418D1 (de) 1995-04-06
ATE119162T1 (de) 1995-03-15
AU622941B2 (en) 1992-04-30
NO894474D0 (no) 1989-11-09
NO173827B (no) 1993-11-01
DK626288D0 (da) 1988-11-10
ES2068903T3 (es) 1995-05-01
IE893374L (en) 1990-05-10
GR3015718T3 (en) 1995-07-31
FI92931B (fi) 1994-10-14
CA2002624A1 (en) 1990-05-10
FI92931C (fi) 1995-01-25
PT92279A (pt) 1990-05-31
EP0368652A1 (en) 1990-05-16
PT92279B (pt) 1995-08-09
JPH02178285A (ja) 1990-07-11
DE68921418T2 (de) 1995-07-13
FI895257A0 (fi) 1989-11-06
NO173827C (no) 1994-02-09
EP0368652B1 (en) 1995-03-01
IE68939B1 (en) 1996-07-24
AU4439389A (en) 1990-05-17
NZ231321A (en) 1991-10-25
ZA898051B (en) 1990-08-29
IL92055A0 (en) 1990-07-12
NO894474L (no) 1990-05-11

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