DK155524C - Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse - Google Patents

Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse

Info

Publication number
DK155524C
DK155524C DK137487A DK137487A DK155524C DK 155524 C DK155524 C DK 155524C DK 137487 A DK137487 A DK 137487A DK 137487 A DK137487 A DK 137487A DK 155524 C DK155524 C DK 155524C
Authority
DK
Denmark
Prior art keywords
alkyl
condensed
pharmaceutical preparations
preparations containing
alkynyl
Prior art date
Application number
DK137487A
Other languages
English (en)
Other versions
DK137487D0 (da
DK137487A (da
DK155524B (da
Inventor
Frank Watjen
Holger Claus Hansen
Original Assignee
Ferrosan As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrosan As filed Critical Ferrosan As
Publication of DK137487D0 publication Critical patent/DK137487D0/da
Priority to DK137487A priority Critical patent/DK155524C/da
Priority to IL85295A priority patent/IL85295A/xx
Priority to PH36480A priority patent/PH24076A/en
Priority to US07/156,363 priority patent/US4873244A/en
Priority to IE43888A priority patent/IE62320B1/en
Priority to ZA881140A priority patent/ZA881140B/xx
Priority to FI880815A priority patent/FI92700C/fi
Priority to AT88301783T priority patent/ATE92926T1/de
Priority to ES88301783T priority patent/ES2058251T3/es
Priority to EP88301783A priority patent/EP0283162B1/en
Priority to DE88301783T priority patent/DE3883033T2/de
Priority to NZ223777A priority patent/NZ223777A/xx
Priority to KR1019880002727A priority patent/KR960010455B1/ko
Priority to CA000561758A priority patent/CA1308712C/en
Priority to NO881191A priority patent/NO169340C/no
Priority to JP63062068A priority patent/JPS6463581A/ja
Priority to AU13259/88A priority patent/AU607469B2/en
Priority to PT87013A priority patent/PT87013B/pt
Priority to PH37235A priority patent/PH24165A/en
Publication of DK137487A publication Critical patent/DK137487A/da
Publication of DK155524B publication Critical patent/DK155524B/da
Priority to US07/340,901 priority patent/US4902686A/en
Application granted granted Critical
Publication of DK155524C publication Critical patent/DK155524C/da
Priority to FI925310A priority patent/FI93837C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Luminescent Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK137487A 1987-03-18 1987-03-18 Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse DK155524C (da)

Priority Applications (21)

Application Number Priority Date Filing Date Title
DK137487A DK155524C (da) 1987-03-18 1987-03-18 Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
IL85295A IL85295A (en) 1987-03-18 1988-02-02 Tricyclic imidazole derivatives,their preparation and pharmaceutical compositions containing them
PH36480A PH24076A (en) 1987-03-18 1988-02-10 Heterocyclic fused derivatives of imidazoles,composition and method of use thereof
US07/156,363 US4873244A (en) 1987-03-18 1988-02-16 Tricyclic heterocyclic compounds as psychopharmaceuticals
IE43888A IE62320B1 (en) 1987-03-18 1988-02-18 Heterocyclic compounds and their preparation and use
ZA881140A ZA881140B (en) 1987-03-18 1988-02-18 Heterocyclic compounds and their preparation and use
FI880815A FI92700C (fi) 1987-03-18 1988-02-22 Menetelmä uusien terapeuttisesti käyttökelpoisten 5-okso-4,5-dihydro-imidatso/1,5-a/kinatsoliinijohdannaisten valmistamiseksi
DE88301783T DE3883033T2 (de) 1987-03-18 1988-03-01 Heterocyclische Verbindungen und ihre Herstellung und Anwendung.
ES88301783T ES2058251T3 (es) 1987-03-18 1988-03-01 Compuestos heterociclicos y su preparacion y uso.
EP88301783A EP0283162B1 (en) 1987-03-18 1988-03-01 Heterocyclic compounds and their preparation and use
AT88301783T ATE92926T1 (de) 1987-03-18 1988-03-01 Heterocyclische verbindungen und ihre herstellung und anwendung.
NZ223777A NZ223777A (en) 1987-03-18 1988-03-07 Heterocyclic derivatives and pharmaceutical compositions
KR1019880002727A KR960010455B1 (ko) 1987-03-18 1988-03-16 헤테로사이클릭 화합물, 이의 제법 및 용도
CA000561758A CA1308712C (en) 1987-03-18 1988-03-17 Heterocyclic compounds and their preparation and use
NO881191A NO169340C (no) 1987-03-18 1988-03-17 Analogifremgangsmaate for fremstilling av terapeutisk aktive, kondenserte, heterocykliske forbindelser som inneholder en imidazolring
JP63062068A JPS6463581A (en) 1987-03-18 1988-03-17 Heterocyclic compound, manufacture and use
AU13259/88A AU607469B2 (en) 1987-03-18 1988-03-18 Imadazo-quinazolines, imidazo (1-5a) pyrido (2,3-e) pyrazines, imidazo quinolines and imidazo quinoxalines
PT87013A PT87013B (pt) 1987-03-18 1988-03-18 Processo de preparacao de compostos heterociclicos derivados da quinazolina e da pirazina e de composicoes farmaceuticas que os contem
PH37235A PH24165A (en) 1987-03-18 1988-07-18 A process for the preparation of heterocyclic fused derivatives of imidazoles
US07/340,901 US4902686A (en) 1987-03-18 1989-04-20 Tricyclic heterocyclic compounds and their use in treating benzodiazepin receptor-related ailments
FI925310A FI93837C (fi) 1987-03-18 1992-11-23 Menetelmä uusien terapeuttisesti käyttökelpoisten 4-okso-4,5-dihydro-imidatso/1,5-a/pyrido/2,3-e/pyratsiinijohdannaisten valmistamiseksi

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK137487A DK155524C (da) 1987-03-18 1987-03-18 Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK137487 1987-03-18

Publications (4)

Publication Number Publication Date
DK137487D0 DK137487D0 (da) 1987-03-18
DK137487A DK137487A (da) 1988-09-19
DK155524B DK155524B (da) 1989-04-17
DK155524C true DK155524C (da) 1989-09-11

Family

ID=8104158

Family Applications (1)

Application Number Title Priority Date Filing Date
DK137487A DK155524C (da) 1987-03-18 1987-03-18 Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse

Country Status (18)

Country Link
US (2) US4873244A (da)
EP (1) EP0283162B1 (da)
JP (1) JPS6463581A (da)
KR (1) KR960010455B1 (da)
AT (1) ATE92926T1 (da)
AU (1) AU607469B2 (da)
CA (1) CA1308712C (da)
DE (1) DE3883033T2 (da)
DK (1) DK155524C (da)
ES (1) ES2058251T3 (da)
FI (1) FI92700C (da)
IE (1) IE62320B1 (da)
IL (1) IL85295A (da)
NO (1) NO169340C (da)
NZ (1) NZ223777A (da)
PH (2) PH24076A (da)
PT (1) PT87013B (da)
ZA (1) ZA881140B (da)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them
DK161148C (da) * 1988-06-14 1991-11-18 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne
DK626288D0 (da) * 1988-11-10 1988-11-10 Ferrosan As Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen
DK588489D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
DK588389D0 (da) * 1989-11-22 1989-11-22 Ferrosan As Heterocykliske forbindelser, deres fremstilling og anvendelse
FR2659329B1 (fr) * 1990-03-09 1994-06-03 Adir Nouveaux derives d'imidazo [1,2-c] quinazoline, leur procede de preparation et les compositions pharmaceutiques les renfermant.
US5276028A (en) * 1990-06-22 1994-01-04 Nordisk A/S Imidazoquinoxaline compounds
US5371080A (en) * 1990-06-22 1994-12-06 Novo Nordisk A/S Imidazoquinazoline compounds and their use
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
DK204291D0 (da) * 1991-12-20 1991-12-20 Novo Nordisk As Heterocykliske forbindelser deres fremstilling og anvendelse
WO1992004350A1 (en) * 1990-09-04 1992-03-19 The Upjohn Company Oxygenated quinoxalines
WO1992022552A1 (en) * 1991-06-14 1992-12-23 The Upjohn Company IMIDAZO[1,5-a]QUINOXALINES
AU4035893A (en) * 1991-12-17 1993-07-19 Upjohn Company, The 3-substituted imidazo (1,5-a) and imidazo (1,5-a)-triazolo (1,5-c) quinoxalines and quinazolines with cns activity
WO1993016082A1 (en) * 1992-02-13 1993-08-19 The Upjohn Company 4-oxo- and 4h-imidazo(5,1-c)(1,4)benzoxazines useful as benzodiazepine receptor-binding agents
WO1993017025A1 (en) * 1992-02-19 1993-09-02 The Upjohn Company 3-substituted imidazo(1,5-a)quinoxalines and quinazolines with cns activity
US5367077A (en) * 1992-04-08 1994-11-22 Neurogen Corporation Certain cycloalkyl and azacycloalkyl pyrrolopyridines; a new class of gaba rain receptor ligands
CA2174106C (en) * 1993-11-19 2005-06-28 Eric Jon Jacobsen Imidazo[1,5-a]quinolines for treatment of anxiety and sleep disorders
JPH09510695A (ja) * 1994-01-03 1997-10-28 エイシア・ファーマシュウティカルズ，インコーポレイテッド ８−アザ、６−アザ、および６，８−ジアザ−１，４−ジヒドロキノキサリン−２，３−ジオン類およびそのグリシン／ｎｍｄａリセプターに対するアンタゴニストとしての使用
FR2799757B1 (fr) * 1999-10-15 2001-12-14 Adir Nouveaux derives polycycliques azaindoliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
IL156813A0 (en) * 2001-01-26 2004-02-08 Bristol Myers Squibb Co Imidazolyl derivatives and pharmaceutical compositions containing the same
WO2017149469A1 (en) 2016-03-03 2017-09-08 Emcure Pharmaceuticals Limited Heterocyclic compounds useful as ido and/or tdo modulators

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
US4771051A (en) * 1985-05-17 1988-09-13 A/S Ferrosan 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
ATE38671T1 (de) * 1985-05-17 1988-12-15 Ferrosan As Oxadiazolylimidazobenzodiazepine, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
ATE80392T1 (de) * 1985-10-17 1992-09-15 Novo Nordisk As Oxadiazolylacetonitrile, ihre herstellung und anwendung.
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar
IL90315A0 (en) * 1988-06-01 1989-12-15 Ferrosan As Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FI92700C (fi) 1994-12-27
IE880438L (en) 1988-09-18
EP0283162A3 (en) 1990-05-30
PT87013B (pt) 1995-03-01
DE3883033T2 (de) 1993-12-16
NZ223777A (en) 1989-09-27
FI880815A0 (fi) 1988-02-22
PT87013A (pt) 1989-03-30
KR960010455B1 (ko) 1996-08-01
DK137487D0 (da) 1987-03-18
IL85295A (en) 1991-12-12
ES2058251T3 (es) 1994-11-01
NO881191D0 (no) 1988-03-17
NO881191L (no) 1988-09-19
ZA881140B (en) 1988-08-15
DK137487A (da) 1988-09-19
ATE92926T1 (de) 1993-08-15
CA1308712C (en) 1992-10-13
PH24165A (en) 1990-03-22
JPS6463581A (en) 1989-03-09
KR880011157A (ko) 1988-10-26
DK155524B (da) 1989-04-17
US4902686A (en) 1990-02-20
NO169340B (no) 1992-03-02
NO169340C (no) 1992-06-10
US4873244A (en) 1989-10-10
FI92700B (fi) 1994-09-15
IE62320B1 (en) 1995-01-25
PH24076A (en) 1990-03-05
AU607469B2 (en) 1991-03-07
EP0283162B1 (en) 1993-08-11
AU1325988A (en) 1988-09-22
EP0283162A2 (en) 1988-09-21
DE3883033D1 (de) 1993-09-16
FI880815A (fi) 1988-09-19

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Legal Events

Date Code Title Description
PBP Patent lapsed