IL90337A0 - Aromatic and heterocyclic carboxamide derivatives as antineoplastic agents - Google Patents
Aromatic and heterocyclic carboxamide derivatives as antineoplastic agentsInfo
- Publication number
- IL90337A0 IL90337A0 IL90337A IL9033789A IL90337A0 IL 90337 A0 IL90337 A0 IL 90337A0 IL 90337 A IL90337 A IL 90337A IL 9033789 A IL9033789 A IL 9033789A IL 90337 A0 IL90337 A0 IL 90337A0
- Authority
- IL
- Israel
- Prior art keywords
- aromatic
- antineoplastic agents
- carboxamide derivatives
- heterocyclic carboxamide
- heterocyclic
- Prior art date
Links
- 239000002246 antineoplastic agent Substances 0.000 title abstract 2
- 229940053202 antiepileptics carboxamide derivative Drugs 0.000 title 1
- 229940034982 antineoplastic agent Drugs 0.000 title 1
- 125000003118 aryl group Chemical group 0.000 title 1
- 125000000623 heterocyclic group Chemical group 0.000 title 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Steroid Compounds (AREA)
- Graft Or Block Polymers (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19803488A | 1988-05-24 | 1988-05-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL90337A0 true IL90337A0 (en) | 1989-12-15 |
Family
ID=22731735
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL90337A IL90337A0 (en) | 1988-05-24 | 1989-05-18 | Aromatic and heterocyclic carboxamide derivatives as antineoplastic agents |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP0343893B1 (enExample) |
| JP (1) | JPH0678331B2 (enExample) |
| KR (1) | KR910006864B1 (enExample) |
| CN (1) | CN1023700C (enExample) |
| AT (1) | ATE79114T1 (enExample) |
| AU (1) | AU601905B2 (enExample) |
| CA (1) | CA1328871C (enExample) |
| DD (1) | DD283815A5 (enExample) |
| DE (1) | DE68902358T2 (enExample) |
| DK (1) | DK249389A (enExample) |
| ES (1) | ES2043012T3 (enExample) |
| FI (1) | FI892498A7 (enExample) |
| GR (1) | GR3005844T3 (enExample) |
| HU (1) | HU202507B (enExample) |
| IE (1) | IE891667L (enExample) |
| IL (1) | IL90337A0 (enExample) |
| MX (1) | MX173140B (enExample) |
| MY (1) | MY106035A (enExample) |
| NO (1) | NO172389C (enExample) |
| NZ (1) | NZ229234A (enExample) |
| PL (1) | PL154875B1 (enExample) |
| PT (1) | PT90622B (enExample) |
| SU (1) | SU1681728A3 (enExample) |
| YU (1) | YU47019B (enExample) |
| ZA (1) | ZA893862B (enExample) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2790299B2 (ja) * | 1989-02-01 | 1998-08-27 | 保土谷化学工業株式会社 | ペンゾチアゾール誘導体 |
| US5262400A (en) * | 1991-06-20 | 1993-11-16 | Merck & Co., Inc. | 4α-substituted avermectin derivatives |
| US6100423A (en) * | 1995-08-30 | 2000-08-08 | G. D. Searle & Co. | Amino benzenepropanoic acid compounds and derivatives thereof |
| CZ293323B6 (cs) * | 1995-08-30 | 2004-04-14 | G. D. Searle & Co. | Meta-guanidinové, močovinové, thiomočovinové nebo azacyklické deriváty aminobenzoové kyseliny jako antagonisty integrinů |
| US5716281A (en) * | 1995-11-27 | 1998-02-10 | Sega Enterprises, Ltd. | Game apparatus using a vehicle with an optical image synthesizing system |
| TW513418B (en) * | 1996-07-31 | 2002-12-11 | Otsuka Pharma Co Ltd | Thiazole derivatives, their production and use |
| CA2309319A1 (en) | 1997-11-10 | 1999-05-20 | Bristol-Myers Squibb Company | Benzothiazole protein tyrosine kinase inhibitors |
| EP0928793B1 (en) * | 1998-01-02 | 2002-05-15 | F. Hoffmann-La Roche Ag | Thiazole derivatives |
| AU3406599A (en) * | 1998-04-09 | 1999-11-01 | Institut Fur Diagnostikforschung Gmbh An Der Freien Universitat Berlin | Novel benzyl guanidine derivatives for therapy and (in-vivo) and (in-vitro) diagnosis |
| NZ522928A (en) | 2000-06-21 | 2005-05-27 | F | Benzothiazole derivatives |
| US6620811B2 (en) * | 2001-11-19 | 2003-09-16 | Hoffmann-La Roche Inc. | Isonicotin- and nicotinamide derivatives of benzothiazoles |
| US6599901B1 (en) * | 2001-11-19 | 2003-07-29 | Hoffman-La Roche Inc. | Pyridone substituted benzothiazole derivatives |
| US6624163B2 (en) * | 2001-11-29 | 2003-09-23 | Hoffman-La Roche Inc. | Benzothiazole derivatives |
| GB0130868D0 (en) | 2001-12-24 | 2002-02-06 | Univ Strathclyde | New compounds |
| CN100357283C (zh) * | 2002-04-02 | 2007-12-26 | 中国科学院上海药物研究所 | 一类甲硫氨酰氨肽酶抑制剂 |
| US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
| DE602004016328D1 (de) * | 2003-05-13 | 2008-10-16 | Hoffmann La Roche | 2-imidazo-benzothiazole als adenosin-rezeptor liganden |
| AU2004251814B2 (en) * | 2003-05-19 | 2009-07-23 | F. Hoffmann-La Roche Ag | Benzothiazole derivatives as adenosine receptor ligands |
| EP1628662B1 (en) * | 2003-05-21 | 2007-02-14 | F. Hoffmann-La Roche Ag | Benzothiazole derivatives and use thereof in the treatment of diseases related to the adenosine a2a receptor |
| MXPA05012772A (es) * | 2003-05-30 | 2006-02-13 | Hoffmann La Roche | Derivados de benzotiazol y uso de los mismos en el tratamiento de enfermedades relacionadas con el receptor a2a de adenosina. |
| PT1660491E (pt) * | 2003-07-28 | 2008-10-10 | Janssen Pharmaceutica Nv | Derivados de benzimidazole, benzotiazole e benzoxazole e a sua utilização como moduladores de lta4h |
| CN1956983B (zh) | 2004-05-24 | 2010-05-26 | 弗·哈夫曼-拉罗切有限公司 | 4-羟基-4-甲基-哌啶-1-甲酸(4-甲氧基-7-吗啉-4-基-苯并噻唑-2-基)-酰胺 |
| EP1773827B1 (en) * | 2004-07-22 | 2010-02-17 | F.Hoffmann-La Roche Ag | Benzothiazole derivatives |
| KR100818028B1 (ko) * | 2004-07-22 | 2008-03-31 | 에프. 호프만-라 로슈 아게 | 치환된 벤조티아졸 |
| CA2586931C (en) | 2004-11-05 | 2013-08-06 | Paul Spurr | Process for preparation of isonicotinic acid derivatives |
| RU2412943C2 (ru) | 2005-03-23 | 2011-02-27 | Ф. Хоффманн-Ля Рош Аг | ПРОИЗВОДНЫЕ АЦЕТИЛЕНИЛ-ПИРАЗОЛО-ПИРИМИДИНА В КАЧЕСТВЕ АНТАГОНИСТОВ mGluR2 |
| ES2340321T3 (es) | 2005-09-27 | 2010-06-01 | F.Hoffmann-La Roche Ag | Oxadiazolilpirazolo-pirimidinas, como antagonistas de mglur2. |
| WO2007104557A2 (en) * | 2006-03-15 | 2007-09-20 | 4Sc Ag | Novel heterocyclic nf-kb inhibitors |
| GB0619325D0 (en) | 2006-09-30 | 2006-11-08 | Univ Strathclyde | New compounds |
| EP2311842A3 (en) * | 2008-06-24 | 2011-07-13 | Takeda Pharmaceutical Company Limited | PI3K/M TOR inhibitors |
| US9499790B2 (en) | 2010-08-26 | 2016-11-22 | Kyoto University | Method for promoting differentiation of pluripotent stem cells into cardiac muscle cells |
| AP2014007595A0 (en) * | 2011-09-30 | 2014-04-30 | Kineta Inc | Anti-viral compounds |
| WO2013111875A1 (ja) | 2012-01-27 | 2013-08-01 | 国立大学法人京都大学 | 多能性幹細胞の心筋分化誘導法 |
| US10196609B2 (en) | 2013-03-08 | 2019-02-05 | Kyoto University | Composition for promoting cardiac differentiation of pluripotent stem cell comprising EGFR inhibitor |
| EP3045451B1 (en) * | 2013-09-13 | 2018-03-28 | Kyoto University | Compound promoting differentiation of pluripotent stem cells into cardiomyocytes |
| WO2015182765A1 (ja) | 2014-05-30 | 2015-12-03 | 国立大学法人京都大学 | 低分子化合物を用いた多能性幹細胞の心筋分化誘導法 |
| CN109776486A (zh) * | 2019-02-26 | 2019-05-21 | 武汉松石科技股份有限公司 | 一种硫酸亚丙酯的制备方法 |
| CN110590735B (zh) * | 2019-09-30 | 2021-07-23 | 江苏国泰超威新材料有限公司 | 一种环状硫酸酯的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS61225168A (ja) * | 1985-03-30 | 1986-10-06 | Nippon Tokushu Noyaku Seizo Kk | 新規ベンズアミド、その製法及び殺虫剤 |
| KR930005004B1 (ko) * | 1985-04-15 | 1993-06-11 | 쟈안센 파아마슈우티카 엔. 부이. | 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법 |
| GB8611606D0 (en) * | 1986-05-13 | 1986-06-18 | Fbc Ltd | Fungicides |
-
1989
- 1989-05-18 IL IL90337A patent/IL90337A0/xx unknown
- 1989-05-22 PT PT90622A patent/PT90622B/pt not_active IP Right Cessation
- 1989-05-22 AT AT89305141T patent/ATE79114T1/de not_active IP Right Cessation
- 1989-05-22 ES ES89305141T patent/ES2043012T3/es not_active Expired - Lifetime
- 1989-05-22 JP JP1128600A patent/JPH0678331B2/ja not_active Expired - Lifetime
- 1989-05-22 DE DE8989305141T patent/DE68902358T2/de not_active Expired - Lifetime
- 1989-05-22 EP EP89305141A patent/EP0343893B1/en not_active Expired - Lifetime
- 1989-05-23 AU AU35098/89A patent/AU601905B2/en not_active Ceased
- 1989-05-23 DK DK249389A patent/DK249389A/da unknown
- 1989-05-23 CA CA000600370A patent/CA1328871C/en not_active Expired - Fee Related
- 1989-05-23 DD DD89328832A patent/DD283815A5/de not_active IP Right Cessation
- 1989-05-23 ZA ZA893862A patent/ZA893862B/xx unknown
- 1989-05-23 MY MYPI89000689A patent/MY106035A/en unknown
- 1989-05-23 NZ NZ229234A patent/NZ229234A/en unknown
- 1989-05-23 MX MX016158A patent/MX173140B/es unknown
- 1989-05-23 FI FI892498A patent/FI892498A7/fi not_active Application Discontinuation
- 1989-05-23 NO NO892059A patent/NO172389C/no unknown
- 1989-05-23 IE IE891667A patent/IE891667L/xx unknown
- 1989-05-23 SU SU894614242A patent/SU1681728A3/ru active
- 1989-05-23 KR KR1019890006889A patent/KR910006864B1/ko not_active Expired
- 1989-05-23 HU HU892578A patent/HU202507B/hu not_active IP Right Cessation
- 1989-05-24 CN CN89103540A patent/CN1023700C/zh not_active Expired - Fee Related
- 1989-05-24 YU YU105989A patent/YU47019B/sh unknown
- 1989-05-24 PL PL1989279613A patent/PL154875B1/pl unknown
-
1992
- 1992-09-30 GR GR920402178T patent/GR3005844T3/el unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ZA893862B (en) | Aromatic and heterocyclic carboxamide derivatives as antineoplastic agents | |
| PT82389A (en) | Heterocyclic amide derivatives | |
| YU123689A (en) | Acyl derivatives | |
| NZ217962A (en) | Heterocyclic carboxamide containing derivatives and pharmaceutical compositions | |
| PH25646A (en) | Acyl derivatives | |
| EG18544A (en) | Six - membred heterocyclic derivatives of n', - substituted - n, n'-diacylhydrazines | |
| ZA872738B (en) | Five-membered heterocyclic derivatives of n'-substituted-n,n'-diacylhydrazines | |
| GB2176185B (en) | N-(3 nitroquinolin-4-yl) guarnidine derivatives | |
| EG19066A (en) | New derivatives of cysteine | |
| IL88427A0 (en) | Disulfide benzylcarbamate and-benzylcarbonate derivatives of anti-tumor drugs | |
| ZA885123B (en) | Pest-combating agents based on derivatives of 2,3-diaminomaleonitrile | |
| ZA884093B (en) | Acyl derivatives | |
| CS693488A1 (en) | Derivatives of sulphonamides | |
| MW3086A1 (en) | Heterocyclic amide derivatives | |
| GB8509882D0 (en) | Heterocyclic amide derivatives | |
| YU54789A (en) | Substituted derivatives of thiourea | |
| YU14889A (en) | Acyl derivatives | |
| ZA885790B (en) | Acyl derivatives | |
| ZA882382B (en) | Acyl derivatives | |
| ZA881182B (en) | Saturated heterocyclic carboxamide derivatives | |
| IE881065L (en) | Acyl derivatives of cephalosporins | |
| IE880619L (en) | 27-halo derivatives of ll-f28249 n of an¹expendable pattern | |
| YU11688A (en) | Derivatives of pyridazodiazepine | |
| IE881760L (en) | Derivatives of n-phenylpyrazoles | |
| IE850020L (en) | Thioxanthene derivatives |