IL157933A0 - Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9] -hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof - Google Patents

Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9] -hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof

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Publication number
IL157933A0
IL157933A0 IL15793302A IL15793302A IL157933A0 IL 157933 A0 IL157933 A0 IL 157933A0 IL 15793302 A IL15793302 A IL 15793302A IL 15793302 A IL15793302 A IL 15793302A IL 157933 A0 IL157933 A0 IL 157933A0
Authority
IL
Israel
Prior art keywords
triazatetracyclo
pentaene
hexadeca
pharmaceutical compositions
tartrate salts
Prior art date
Application number
IL15793302A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23117845&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL157933(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of IL157933A0 publication Critical patent/IL157933A0/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A—HUMAN NECESSITIES
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    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
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    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Neurology (AREA)
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  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
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  • Diabetes (AREA)
  • Nutrition Science (AREA)
  • Psychology (AREA)
  • Virology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
IL15793302A 2001-05-14 2002-04-26 Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9] -hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof IL157933A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29086101P 2001-05-14 2001-05-14
PCT/IB2002/001437 WO2002092089A1 (en) 2001-05-14 2002-04-26 Tartrate salts of 5,8,14-triazatetracyclo {10.3.1.0?2,11.04,9¿}-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof

Publications (1)

Publication Number Publication Date
IL157933A0 true IL157933A0 (en) 2004-03-28

Family

ID=23117845

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15793302A IL157933A0 (en) 2001-05-14 2002-04-26 Tartrate salts of 5,8,14-triazatetracyclo [10.3.1.02,11.04,9] -hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof
IL157933A IL157933A (en) 2001-05-14 2003-09-15 Tetratrate salts of 14,8,5-triazate tetracyclo [9,04.11,02.1.3.10] - Hexadka @ - @@@@@@@@@@@@@ - Penta-An @ and pharmaceuticals containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL157933A IL157933A (en) 2001-05-14 2003-09-15 Tetratrate salts of 14,8,5-triazate tetracyclo [9,04.11,02.1.3.10] - Hexadka @ - @@@@@@@@@@@@@ - Penta-An @ and pharmaceuticals containing them

Country Status (47)

Country Link
US (2) US6890927B2 (pl)
EP (1) EP1392307B1 (pl)
JP (1) JP3779682B2 (pl)
KR (1) KR100551184B1 (pl)
CN (1) CN100370987C (pl)
AP (1) AP1473A (pl)
AR (1) AR033635A1 (pl)
AT (1) ATE302607T1 (pl)
AU (1) AU2002253482B2 (pl)
BG (1) BG66408B1 (pl)
BR (1) BR0209605A (pl)
CA (1) CA2447405C (pl)
CR (1) CR7080A (pl)
CZ (1) CZ304763B6 (pl)
DE (1) DE60205742T2 (pl)
DK (1) DK1392307T3 (pl)
DO (1) DOP2002000392A (pl)
EA (1) EA005528B1 (pl)
EC (2) ECSP034849A (pl)
EE (1) EE05441B1 (pl)
EG (1) EG24228A (pl)
ES (1) ES2246396T3 (pl)
GE (1) GEP20053712B (pl)
GT (1) GT200200084A (pl)
HR (1) HRP20030910B1 (pl)
HU (1) HU229867B1 (pl)
IL (2) IL157933A0 (pl)
IS (1) IS2217B (pl)
MA (1) MA27020A1 (pl)
ME (1) ME00466B (pl)
MX (1) MXPA03010364A (pl)
MY (1) MY127807A (pl)
NO (1) NO326148B1 (pl)
NZ (1) NZ528210A (pl)
OA (1) OA12599A (pl)
PA (1) PA8545101A1 (pl)
PE (1) PE20021065A1 (pl)
PL (1) PL214876B1 (pl)
PT (1) PT1392307E (pl)
RS (1) RS50814B (pl)
SI (1) SI1392307T1 (pl)
SK (1) SK287170B6 (pl)
TN (1) TNSN03113A1 (pl)
TW (1) TWI262078B (pl)
UA (1) UA73422C2 (pl)
WO (1) WO2002092089A1 (pl)
ZA (1) ZA200307235B (pl)

Families Citing this family (48)

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JP2006528237A (ja) * 2003-05-20 2006-12-14 ファイザー・プロダクツ・インク バレニクリンの医薬組成物
WO2005061519A1 (en) * 2003-12-19 2005-07-07 Takeda San Diego, Inc. Kinase inhibitors
EP1763524A1 (en) * 2004-04-23 2007-03-21 Takeda San Diego, Inc. Indole derivatives and use thereof as kinase inhibitors
JP2008505075A (ja) * 2004-06-30 2008-02-21 イーライ リリー アンド カンパニー １−（インドール−６−カルボニル−ｄ−フェニルグリシニル）−４−（１−メチルピペリジン−４−イル）ピペラジンｄ−酒石酸塩
US7550598B2 (en) * 2004-08-18 2009-06-23 Takeda Pharmaceutical Company Limited Kinase inhibitors
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JP2008531540A (ja) * 2005-02-24 2008-08-14 ファイザー・プロダクツ・インク 高純度置換キノキサリンの調製
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US8119655B2 (en) * 2005-10-07 2012-02-21 Takeda Pharmaceutical Company Limited Kinase inhibitors
JP2009508880A (ja) * 2006-02-21 2009-03-05 テバ ファーマシューティカル インダストリーズ リミティド アルモダフィニルの新規な結晶形とその調製方法
EP2223925A1 (en) * 2006-10-09 2010-09-01 Takeda Pharmaceutical Company Limited Kinase inhibitors
SG175609A1 (en) 2006-10-09 2011-11-28 Takeda Pharmaceutical Kinase inhibitors
BRPI0718600A2 (pt) * 2006-11-09 2013-12-10 Pfizer Prod Inc Polimorfos de intermediários nicotínicos.
US20090062257A1 (en) * 2007-08-29 2009-03-05 Protia, Llc Deuterium-enriched varenicline
US20090105346A1 (en) * 2007-10-02 2009-04-23 Alexandr Jegorov Novel crystalline forms of armodafinil and preparation thereof
US20090215787A1 (en) * 2008-02-22 2009-08-27 Mai De Ltd. Preparations of new polymorphic forms of varenicline tartrate
WO2009111623A2 (en) * 2008-03-06 2009-09-11 Dr. Reddy's Laboratories Ltd. Amorphous varenicline tartrate
WO2009109651A1 (en) * 2008-03-06 2009-09-11 Medichem, S.A. SALTS OF A PYRAZINO[2,3-h][3]BENZAZEPINE DERIVATIVE
EP2271344A4 (en) * 2008-03-31 2011-04-27 Univ South Florida METHOD FOR TREATING ILLNESS-RELATED ATAXIA AND NON-ATTACHIC IMBALANCE
WO2009143347A2 (en) * 2008-05-22 2009-11-26 Teva Pharmaceutical Industries Ltd. Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate
US20090318460A1 (en) * 2008-05-26 2009-12-24 Glenmark Amorphous varenicline tartrate and process for the preparation thereof
US20090318695A1 (en) * 2008-06-19 2009-12-24 Vinod Kumar Kansal Processes for the preparation of varenicline and intermediates thereof
US20100010221A1 (en) * 2008-07-10 2010-01-14 Revital Lifshitz-Liron Processes for purifying varenicline l-tartrate salt and preparing crystalline forms of varenicline l-tartrate salt
WO2010023561A1 (en) * 2008-09-01 2010-03-04 Actavis Group Ptc Ehf Process for preparing varenicline, varenicline intermediates, and pharmaceutically acceptable salts thereof
EP2440187A2 (en) 2009-06-10 2012-04-18 Actavis Group PTC ehf. Amorphous varenicline tartrate co-precipitates
RU2012102052A (ru) 2009-06-22 2013-11-20 Тева Фармасьютикал Индастриз Лтд. Твердые формы солей варениклина и способы их получения
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KR101663550B1 (ko) * 2014-06-11 2016-10-07 조선대학교산학협력단 주석산을 유효성분으로 포함하는 고혈압 예방 또는 치료용 약학조성물 및 건강기능식품
KR101724301B1 (ko) 2016-11-22 2017-04-10 주식회사 한서켐 바레니클린 살리실산염의 i형 결정 및 그 제조방법
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KR20230068877A (ko) 2021-11-11 2023-05-18 주식회사 아울바이오 고용량 바레니클린을 포함하는 미립구 및 이의 제조방법 및 이를 포함하는 약학적 조성물
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