IL102574A - Anantiospecific courtship of proxiral oxazolyl quion - Google Patents

Anantiospecific courtship of proxiral oxazolyl quion

Info

Publication number
IL102574A
IL102574A IL10257492A IL10257492A IL102574A IL 102574 A IL102574 A IL 102574A IL 10257492 A IL10257492 A IL 10257492A IL 10257492 A IL10257492 A IL 10257492A IL 102574 A IL102574 A IL 102574A
Authority
IL
Israel
Prior art keywords
process according
borane
methyl
formula
phenyl
Prior art date
Application number
IL10257492A
Other languages
English (en)
Hebrew (he)
Other versions
IL102574A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL102574A0 publication Critical patent/IL102574A0/xx
Publication of IL102574A publication Critical patent/IL102574A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL10257492A 1991-07-22 1992-07-21 Anantiospecific courtship of proxiral oxazolyl quion IL102574A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73356491A 1991-07-22 1991-07-22

Publications (2)

Publication Number Publication Date
IL102574A0 IL102574A0 (en) 1993-01-14
IL102574A true IL102574A (en) 1996-07-23

Family

ID=24948157

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10257492A IL102574A (en) 1991-07-22 1992-07-21 Anantiospecific courtship of proxiral oxazolyl quion

Country Status (21)

Country Link
US (1) US5512689A (fr)
EP (1) EP0595868B1 (fr)
JP (1) JP2671962B2 (fr)
AT (1) ATE173728T1 (fr)
AU (1) AU660701B2 (fr)
CA (1) CA2111445C (fr)
DE (1) DE69227689T2 (fr)
DK (1) DK0595868T3 (fr)
ES (1) ES2123562T3 (fr)
FI (1) FI940306A0 (fr)
HU (1) HUT70412A (fr)
IE (1) IE922359A1 (fr)
IL (1) IL102574A (fr)
MX (1) MX9204278A (fr)
MY (1) MY131277A (fr)
NO (1) NO940227L (fr)
NZ (1) NZ243651A (fr)
PT (1) PT100710B (fr)
TW (1) TW199891B (fr)
WO (1) WO1993002060A1 (fr)
ZA (1) ZA925469B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100214907B1 (ko) * 1991-07-22 1999-08-02 디. 제이. 우드, 스피겔 알렌 제이 당뇨병 치료용 티아졸을 제조하기 위한 키랄 중간체
FR2699172B1 (fr) * 1992-12-11 1995-01-20 Adir Nouveaux dérivés de 4-méthyl-1,3-oxazole, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
TW416958B (en) * 1993-05-14 2001-01-01 Pfizer Enantioselective oxazaborolidine catalysts
US6515003B1 (en) * 1999-08-31 2003-02-04 Maxia Pharmaceuticals, Inc. Heterocyclic derivatives for the treatment of diabetes and other diseases
WO2002072009A2 (fr) 2001-03-07 2002-09-19 Maxia Pharmaceuticals, Inc. Derives heterocycliques pour le traitement du cancer et d'autres maladies proliferatives
WO2002072543A2 (fr) * 2001-03-08 2002-09-19 Maxia Pharmaceuticals, Inc. Molecules activant un recepteur rxr
CA2340824A1 (fr) * 2001-03-14 2002-09-14 Ibm Canada Limited-Ibm Canada Limitee Methode et systeme pour l'analyse du comportement des applications
WO2003016267A1 (fr) * 2001-08-17 2003-02-27 Incyte San Diego Incorporated Derives d'oxime pour le traitement de la dyslipidemie et de l'hypercholesterolemie
WO2003043998A1 (fr) * 2001-11-15 2003-05-30 Incyte San Diego Incorporated Heterocycles n-substitues pour le traitement de l'hypercholesterolemie, de la dyslipidemie et autres troubles du metabolisme, du cancer et de pathologies diverses
US7102000B2 (en) * 2002-03-08 2006-09-05 Incyte San Diego Inc. Heterocyclic amide derivatives for the treatment of diabetes and other diseases
US7196108B2 (en) * 2002-03-08 2007-03-27 Incyte San Diego Inc. Bicyclic heterocycles for the treatment of diabetes and other diseases
US20050014767A1 (en) * 2003-01-29 2005-01-20 Magnus Pfahl Benzoxazole, benzothiazole, and benzimidazole derivatives for the treatment of cancer and other diseases
CA2522759A1 (fr) * 2003-04-18 2004-11-04 Incyte San Diego Incorporated Composes isochromane substitues pour le traitement de troubles metaboliques, du cancer et d'autres maladies

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943635A (en) * 1987-08-27 1990-07-24 President & Fellows Of Harvard College Enantioselective reduction of ketones
US5036079A (en) * 1989-12-07 1991-07-30 Pfizer Inc. Hypoglycemic thiazolidinedione derivatives
TW222626B (fr) * 1991-07-22 1994-04-21 Pfizer

Also Published As

Publication number Publication date
MX9204278A (es) 1994-03-31
FI940306A (fi) 1994-01-21
NO940227D0 (no) 1994-01-21
AU2306292A (en) 1993-02-23
TW199891B (fr) 1993-02-11
EP0595868B1 (fr) 1998-11-25
WO1993002060A1 (fr) 1993-02-04
AU660701B2 (en) 1995-07-06
NZ243651A (en) 1994-01-26
PT100710A (pt) 1993-09-30
IL102574A0 (en) 1993-01-14
CA2111445C (fr) 1997-02-18
DE69227689D1 (de) 1999-01-07
DE69227689T2 (de) 1999-04-22
DK0595868T3 (da) 1999-08-09
EP0595868A1 (fr) 1994-05-11
JPH07502017A (ja) 1995-03-02
CA2111445A1 (fr) 1993-02-04
FI940306A0 (fi) 1994-01-21
HUT70412A (en) 1995-10-30
US5512689A (en) 1996-04-30
JP2671962B2 (ja) 1997-11-05
IE922359A1 (en) 1993-01-27
ZA925469B (en) 1994-01-21
MY131277A (en) 2007-07-31
NO940227L (no) 1994-01-21
ATE173728T1 (de) 1998-12-15
HU9400188D0 (en) 1994-05-30
ES2123562T3 (es) 1999-01-16
PT100710B (pt) 1999-07-30

Similar Documents

Publication Publication Date Title
AU660701B2 (en) Process for the preparation of intermediates in the synthesis of chiral thiazolidine-2,4-dione derivatives
AP776A (en) Benzoxazoles and pyridine derivatives useful in the treatment of the type Ii diabetes.
CA1124245A (fr) Composes du type acide interphenylene-9-thia-11-oxo-12-azaprostanoiques
WO1995017394A1 (fr) Derives heterocycliques et leur utilisation dans des produits pharmaceutiques
CA2299447C (fr) Procede permettant d'obtenir des enantiomeres de cis-olirtine
EP0640089B1 (fr) Catalyseurs a oxazaborolidine enantioselectifs
JP3484200B2 (ja) チアゾリジンジオンの改良製造方法及び新規なチアゾリジンジオン
LU86392A1 (fr) Intermediaires intervenant dans la production d'epipodophyllotoxine et composes apparentes:procedes de preparation et emploi
RU2150472C1 (ru) Способ получения диизопинокамфеилхлорборана в реакционной смеси, способ восстановления прохирального кетона
JP2546559B2 (ja) ジイソピノカンフェイルクロロボランのインシトゥー製造
ARAI et al. Stereoselective reduction of chiral 3-(p-tolylsulfinyl)-2-thienyl ketones. A facile entry to optically active thienylcarbinols
JP2672029B2 (ja) チアゾール系抗糖尿病薬製造用のキラル中間体
US4243817A (en) Prostenoic acids and esters
JPH04352745A (ja) 光学活性アルコールの製法
CA2085716A1 (fr) Carbamates a substituant heterocyclique et methode pour les preparer

Legal Events

Date Code Title Description
FF Patent granted
RH Patent void