PT100710A - Processo para a preparacao de tiazolidina-2,4-diona quirais hipoglicemicas e seus intermediarios - Google Patents

Processo para a preparacao de tiazolidina-2,4-diona quirais hipoglicemicas e seus intermediarios

Info

Publication number
PT100710A
PT100710A PT100710A PT10071092A PT100710A PT 100710 A PT100710 A PT 100710A PT 100710 A PT100710 A PT 100710A PT 10071092 A PT10071092 A PT 10071092A PT 100710 A PT100710 A PT 100710A
Authority
PT
Portugal
Prior art keywords
hypoglycemics
diona
intermediaries
quiet
thiazolidine
Prior art date
Application number
PT100710A
Other languages
English (en)
Other versions
PT100710B (pt
Inventor
George J Quallich
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT100710A publication Critical patent/PT100710A/pt
Publication of PT100710B publication Critical patent/PT100710B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PT100710A 1991-07-22 1992-07-20 Processo para a preparacao de tiazolidina-2,4-diona quirais hipoglicemicas e seus intermediarios PT100710B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73356491A 1991-07-22 1991-07-22

Publications (2)

Publication Number Publication Date
PT100710A true PT100710A (pt) 1993-09-30
PT100710B PT100710B (pt) 1999-07-30

Family

ID=24948157

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100710A PT100710B (pt) 1991-07-22 1992-07-20 Processo para a preparacao de tiazolidina-2,4-diona quirais hipoglicemicas e seus intermediarios

Country Status (21)

Country Link
US (1) US5512689A (pt)
EP (1) EP0595868B1 (pt)
JP (1) JP2671962B2 (pt)
AT (1) ATE173728T1 (pt)
AU (1) AU660701B2 (pt)
CA (1) CA2111445C (pt)
DE (1) DE69227689T2 (pt)
DK (1) DK0595868T3 (pt)
ES (1) ES2123562T3 (pt)
FI (1) FI940306A0 (pt)
HU (1) HUT70412A (pt)
IE (1) IE922359A1 (pt)
IL (1) IL102574A (pt)
MX (1) MX9204278A (pt)
MY (1) MY131277A (pt)
NO (1) NO940227D0 (pt)
NZ (1) NZ243651A (pt)
PT (1) PT100710B (pt)
TW (1) TW199891B (pt)
WO (1) WO1993002060A1 (pt)
ZA (1) ZA925469B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2111446C (en) * 1991-07-22 1997-12-16 George J. Quallich Chiral intermediates for the preparation of antidiabetics thiazoles
FR2699172B1 (fr) * 1992-12-11 1995-01-20 Adir Nouveaux dérivés de 4-méthyl-1,3-oxazole, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
TW416958B (en) * 1993-05-14 2001-01-01 Pfizer Enantioselective oxazaborolidine catalysts
EP1214305A1 (en) * 1999-08-31 2002-06-19 Maxia Pharmaceuticals, Inc. Benzylidene-thiazolidinediones and analogues and their use in the treatment of inflammation
WO2002072009A2 (en) 2001-03-07 2002-09-19 Maxia Pharmaceuticals, Inc. Heterocyclic derivatives for the treatment of cancer and other proliferative diseases
US7265139B2 (en) * 2001-03-08 2007-09-04 Incyte San Diego Inc. RXR activating molecules
CA2340824A1 (en) * 2001-03-14 2002-09-14 Ibm Canada Limited-Ibm Canada Limitee Method and system for application behavior analysis
JP2005500379A (ja) * 2001-08-17 2005-01-06 インサイト サンディエゴ インコーポレーテッド 異脂肪血症および高コレステロール血症を治療するオキシム誘導体
AU2002352706A1 (en) * 2001-11-15 2003-06-10 Maxia Pharmaceuticals, Inc. N-substituted heterocycles for the treatment of hypercholesteremia, dyslipidemia and other metabolic disorders, cancer, and other diseases
US7102000B2 (en) * 2002-03-08 2006-09-05 Incyte San Diego Inc. Heterocyclic amide derivatives for the treatment of diabetes and other diseases
US7196108B2 (en) * 2002-03-08 2007-03-27 Incyte San Diego Inc. Bicyclic heterocycles for the treatment of diabetes and other diseases
US20050014767A1 (en) * 2003-01-29 2005-01-20 Magnus Pfahl Benzoxazole, benzothiazole, and benzimidazole derivatives for the treatment of cancer and other diseases
AU2004232326A1 (en) * 2003-04-18 2004-11-04 Incyte San Diego Incorporated Substituted isochroman compounds for the treatment of metabolic disorders, cancer and other diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943635A (en) * 1987-08-27 1990-07-24 President & Fellows Of Harvard College Enantioselective reduction of ketones
US5036079A (en) * 1989-12-07 1991-07-30 Pfizer Inc. Hypoglycemic thiazolidinedione derivatives
TW222626B (pt) * 1991-07-22 1994-04-21 Pfizer

Also Published As

Publication number Publication date
TW199891B (pt) 1993-02-11
DK0595868T3 (da) 1999-08-09
MY131277A (en) 2007-07-31
DE69227689T2 (de) 1999-04-22
ZA925469B (en) 1994-01-21
FI940306A (fi) 1994-01-21
IL102574A (en) 1996-07-23
PT100710B (pt) 1999-07-30
NO940227L (no) 1994-01-21
EP0595868B1 (en) 1998-11-25
NO940227D0 (no) 1994-01-21
ES2123562T3 (es) 1999-01-16
US5512689A (en) 1996-04-30
JP2671962B2 (ja) 1997-11-05
IL102574A0 (en) 1993-01-14
DE69227689D1 (de) 1999-01-07
AU660701B2 (en) 1995-07-06
NZ243651A (en) 1994-01-26
ATE173728T1 (de) 1998-12-15
IE922359A1 (en) 1993-01-27
MX9204278A (es) 1994-03-31
HUT70412A (en) 1995-10-30
JPH07502017A (ja) 1995-03-02
CA2111445A1 (en) 1993-02-04
AU2306292A (en) 1993-02-23
WO1993002060A1 (en) 1993-02-04
EP0595868A1 (en) 1994-05-11
CA2111445C (en) 1997-02-18
FI940306A0 (fi) 1994-01-21
HU9400188D0 (en) 1994-05-30

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19930527

FG3A Patent granted, date of granting

Effective date: 19990413

MM3A Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20041013