IL101243A - תכשירי רוקחות לטיפול בהיפרפלזיה שפירה של הערמונה המכילים תולדות סטירואיד - Google Patents

תכשירי רוקחות לטיפול בהיפרפלזיה שפירה של הערמונה המכילים תולדות סטירואיד

Info

Publication number
IL101243A
IL101243A IL10124392A IL10124392A IL101243A IL 101243 A IL101243 A IL 101243A IL 10124392 A IL10124392 A IL 10124392A IL 10124392 A IL10124392 A IL 10124392A IL 101243 A IL101243 A IL 101243A
Authority
IL
Israel
Prior art keywords
alkyl
acid
amino
group
methyl
Prior art date
Application number
IL10124392A
Other languages
English (en)
Other versions
IL101243A0 (en
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27100766&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL101243(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of IL101243A0 publication Critical patent/IL101243A0/xx
Publication of IL101243A publication Critical patent/IL101243A/he

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL10124392A 1991-03-20 1992-03-16 תכשירי רוקחות לטיפול בהיפרפלזיה שפירה של הערמונה המכילים תולדות סטירואיד IL101243A (he)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67251191A 1991-03-20 1991-03-20
US84615392A 1992-03-11 1992-03-11

Publications (2)

Publication Number Publication Date
IL101243A0 IL101243A0 (en) 1992-11-15
IL101243A true IL101243A (he) 1999-12-22

Family

ID=27100766

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10124392A IL101243A (he) 1991-03-20 1992-03-16 תכשירי רוקחות לטיפול בהיפרפלזיה שפירה של הערמונה המכילים תולדות סטירואיד

Country Status (18)

Country Link
US (2) US5753641A (he)
EP (1) EP0576603A1 (he)
JP (1) JPH06506227A (he)
AU (1) AU666846B2 (he)
BG (1) BG61798B1 (he)
CA (1) CA2104793C (he)
CZ (1) CZ292712B6 (he)
HU (1) HUT66273A (he)
IE (1) IE920879A1 (he)
IL (1) IL101243A (he)
NO (1) NO305635B1 (he)
NZ (1) NZ241979A (he)
RO (1) RO113613B1 (he)
RU (1) RU2125879C1 (he)
SG (1) SG80530A1 (he)
SK (1) SK284381B6 (he)
UA (1) UA41305C2 (he)
WO (1) WO1992016213A1 (he)

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US5541322A (en) * 1994-10-14 1996-07-30 Glaxo Wellcome Inc. Synthesis of 6-azaandrostenones
US5952351A (en) * 1995-02-23 1999-09-14 Merck & Co., Inc. Alpha 1a adrenergic receptor antagonists
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US6096763A (en) * 1995-02-23 2000-08-01 Merck & Co., Inc. α1a adrenergic receptor antagonists
US5670643A (en) * 1995-03-16 1997-09-23 Glaxo Wellcome Inc. Method for preparing finasteride
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US6001844A (en) * 1995-09-15 1999-12-14 Merck & Co., Inc. 4-Azasteroids for treatment of hyperandrogenic conditions
US6177430B1 (en) 1997-03-27 2001-01-23 Pfizer Inc Use of α1-adrenoreceptor antagonists in the prevention and treatment of benign prostatic hyperplasia
US5922722A (en) * 1996-11-12 1999-07-13 Merck & Co., Inc. Alpha 1a adrenergic receptor antagonists
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US6214832B1 (en) 1997-06-18 2001-04-10 Merck & Co., Inc. Bis-piperidinyl-pyrimidin-2-ones as alpha 1a adrenergic receptor antagonists
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Also Published As

Publication number Publication date
WO1992016213A1 (en) 1992-10-01
EP0576603A1 (en) 1994-01-05
JPH06506227A (ja) 1994-07-14
AU1751492A (en) 1992-10-21
SG80530A1 (en) 2001-05-22
HUT66273A (en) 1994-11-28
NO933327D0 (no) 1993-09-17
US5753641A (en) 1998-05-19
CZ292712B6 (cs) 2003-12-17
SK284381B6 (sk) 2005-02-04
NO933327L (no) 1993-11-17
US6046183A (en) 2000-04-04
IL101243A0 (en) 1992-11-15
RO113613B1 (ro) 1998-09-30
CZ193393A3 (en) 1994-08-17
IE920879A1 (en) 1992-09-23
NO305635B1 (no) 1999-07-05
CA2104793A1 (en) 1992-09-21
AU666846B2 (en) 1996-02-29
BG61798B1 (bg) 1998-06-30
UA41305C2 (uk) 2001-09-17
CA2104793C (en) 2004-06-22
SK100693A3 (en) 1994-11-09
RU2125879C1 (ru) 1999-02-10
NZ241979A (en) 1996-01-26
HU9302624D0 (en) 1993-12-28
BG98113A (bg) 1994-06-30

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