ID27771A - Turunan triazol-piridazin tersubstitusi, komposisi farmasi yang dibuat dari bahan itu - Google Patents

Turunan triazol-piridazin tersubstitusi, komposisi farmasi yang dibuat dari bahan itu

Info

Publication number
ID27771A
ID27771A IDW20002717A ID20002717A ID27771A ID 27771 A ID27771 A ID 27771A ID W20002717 A IDW20002717 A ID W20002717A ID 20002717 A ID20002717 A ID 20002717A ID 27771 A ID27771 A ID 27771A
Authority
ID
Indonesia
Prior art keywords
piridazin
substitutional
triazol
derives
pharmaceutical composition
Prior art date
Application number
IDW20002717A
Other languages
English (en)
Indonesian (id)
Inventor
William Robert Carling
Antony John Davies
Gareth Edward Stephen Pearce
Jose Luis Casiro Pineiro
Andrew Madin
Leslie Joseph Sireet
Cameron John Cowden
James Francis Mccabe
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of ID27771A publication Critical patent/ID27771A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IDW20002717A 1998-06-24 1999-06-15 Turunan triazol-piridazin tersubstitusi, komposisi farmasi yang dibuat dari bahan itu ID27771A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9813576.7A GB9813576D0 (en) 1998-06-24 1998-06-24 Therapeutic agents

Publications (1)

Publication Number Publication Date
ID27771A true ID27771A (id) 2001-04-26

Family

ID=10834265

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW20002717A ID27771A (id) 1998-06-24 1999-06-15 Turunan triazol-piridazin tersubstitusi, komposisi farmasi yang dibuat dari bahan itu

Country Status (35)

Country Link
US (1) US6630471B1 (es)
EP (1) EP1090004B1 (es)
JP (1) JP4749545B2 (es)
KR (1) KR100604108B1 (es)
CN (1) CN1138779C (es)
AR (1) AR018925A1 (es)
AT (1) ATE239730T1 (es)
AU (1) AU757315B2 (es)
BG (1) BG64989B1 (es)
BR (1) BR9911563A (es)
CA (1) CA2335328C (es)
CO (1) CO5031239A1 (es)
CZ (1) CZ291409B6 (es)
DE (1) DE69907675T2 (es)
EA (1) EA003332B1 (es)
EE (1) EE200000767A (es)
ES (1) ES2196824T3 (es)
GB (1) GB9813576D0 (es)
GE (1) GEP20033143B (es)
HR (1) HRP20000879A2 (es)
HU (1) HUP0102894A3 (es)
ID (1) ID27771A (es)
IL (2) IL139775A0 (es)
IS (1) IS2258B (es)
MY (1) MY124341A (es)
NO (1) NO317992B1 (es)
NZ (1) NZ508290A (es)
PE (1) PE20000710A1 (es)
PL (1) PL204650B1 (es)
RS (1) RS49746B (es)
SK (1) SK285307B6 (es)
TR (1) TR200003789T2 (es)
TW (1) TWI222449B (es)
WO (1) WO1999067245A1 (es)
ZA (1) ZA200007485B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2345443A (en) * 1999-01-08 2000-07-12 Merck Sharp & Dohme Use of triazolo-pyridazines for treating premenstrual syndrome
US20050042194A1 (en) 2000-05-11 2005-02-24 A.P. Pharma, Inc. Semi-solid delivery vehicle and pharmaceutical compositions
GB0111191D0 (en) * 2001-05-08 2001-06-27 Merck Sharp & Dohme Therapeutic agents
ATE473980T1 (de) * 2002-12-18 2010-07-15 Vertex Pharma Triazolopyridazine als proteinkinase-inhibitoren
WO2006061428A2 (en) * 2004-12-10 2006-06-15 Universität Zürich Gaba-a alpha 2 and alpha 3 receptor agonists for treating neuropathic, inflammatory and migraine associated pain
WO2011005520A1 (en) 2009-06-23 2011-01-13 Concert Pharmaceuticals, Inc. Deuterium-modified triazolo-pyridazine derivatives as gaba-a receptor modulators
WO2011011712A1 (en) * 2009-07-24 2011-01-27 Concert Pharmaceuticals, Inc. Substituted imidazotriazines
WO2011047315A1 (en) 2009-10-15 2011-04-21 Concert Pharmaceuticals, Inc. Subsitituted benzimidazoles
SG182297A1 (en) 2009-12-31 2012-08-30 Ct Nac Investigaciones Oncologicas Cnio Tricyclic compounds for use as kinase inhibitors
WO2012098387A1 (en) * 2011-01-18 2012-07-26 Centro Nacional De Investigaciones Oncológicas (Cnio) 6, 7-ring-fused triazolo [4, 3 - b] pyridazine derivatives as pim inhibitors
WO2013045519A1 (en) 2011-09-27 2013-04-04 Genfit Derivatives of 6-substituted triazolopyridazines as rev-erb agonists
CA3222584A1 (en) 2016-01-27 2017-08-03 Universitat Zurich Use of gabaa receptor modulators for treatment of itch
MX2020010878A (es) * 2018-04-18 2021-01-29 Neurocycle Therapeutics Inc Compuestos moduladores alostericos positivos gabaa, metodos de preparacion y usos de los mismos.
JP7353663B2 (ja) 2018-09-13 2023-10-02 サニオナ エー/エス Gabaa受容体リガンド
HU231223B1 (hu) 2018-09-28 2022-01-28 Richter Gedeon Nyrt. GABAA A5 receptor modulátor hatású biciklusos vegyületek
US20240043418A1 (en) 2020-03-26 2024-02-08 Richter Gedeon Nyrt. 1,3-dihydro-2h-pyrrolo[3,4-c]pyridine derivatives as gabaa a5 receptor modulators

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ333768A (en) * 1996-07-25 2000-09-29 Merck Sharp & Dohme Substituted triazolo-pyridazine derivatives as ligands for GABA receptors

Also Published As

Publication number Publication date
RS49746B (sr) 2008-04-04
PE20000710A1 (es) 2000-08-14
ZA200007485B (en) 2002-01-07
JP2002518501A (ja) 2002-06-25
NO317992B1 (no) 2005-01-17
KR20010053136A (ko) 2001-06-25
PL204650B1 (pl) 2010-01-29
GEP20033143B (en) 2003-12-25
JP4749545B2 (ja) 2011-08-17
CN1138779C (zh) 2004-02-18
GB9813576D0 (en) 1998-08-19
BG64989B1 (bg) 2006-11-30
AR018925A1 (es) 2001-12-12
KR100604108B1 (ko) 2006-07-26
HUP0102894A3 (en) 2003-03-28
BG105152A (en) 2001-10-31
CZ20004872A3 (cs) 2001-07-11
US6630471B1 (en) 2003-10-07
EA003332B1 (ru) 2003-04-24
HRP20000879A2 (en) 2001-06-30
YU77800A (sh) 2003-10-31
IS2258B (is) 2007-06-15
MY124341A (en) 2006-06-30
DE69907675T2 (de) 2004-03-04
CZ291409B6 (cs) 2003-03-12
HUP0102894A2 (hu) 2001-11-28
AU4630199A (en) 2000-01-10
SK285307B6 (sk) 2006-10-05
EP1090004B1 (en) 2003-05-07
CA2335328A1 (en) 1999-12-29
DE69907675D1 (de) 2003-06-12
AU757315B2 (en) 2003-02-13
TWI222449B (en) 2004-10-21
BR9911563A (pt) 2001-03-20
CN1307579A (zh) 2001-08-08
EA200100071A1 (ru) 2001-06-25
TR200003789T2 (tr) 2001-04-20
CO5031239A1 (es) 2001-04-27
CA2335328C (en) 2007-11-27
IL139775A (en) 2007-02-11
IL139775A0 (en) 2002-02-10
EE200000767A (et) 2002-06-17
NO20006576D0 (no) 2000-12-21
EP1090004A1 (en) 2001-04-11
ES2196824T3 (es) 2003-12-16
SK19552000A3 (sk) 2001-08-06
NO20006576L (no) 2001-02-14
WO1999067245A1 (en) 1999-12-29
IS5730A (is) 2000-11-24
NZ508290A (en) 2003-09-26
PL345332A1 (en) 2001-12-17
ATE239730T1 (de) 2003-05-15

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