ID21775A - Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya - Google Patents

Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya

Info

Publication number
ID21775A
ID21775A IDW990226A ID990226A ID21775A ID 21775 A ID21775 A ID 21775A ID W990226 A IDW990226 A ID W990226A ID 990226 A ID990226 A ID 990226A ID 21775 A ID21775 A ID 21775A
Authority
ID
Indonesia
Prior art keywords
compounds
phenilpirazol
pharmacies
compound
hyperuricacidemia
Prior art date
Application number
IDW990226A
Other languages
English (en)
Inventor
Seigo Ishibuchi
Hiroshi Morimoto
Atsushi Fukunari
Hiroyoshi Inoue
Yoichi Naka
Original Assignee
Yoshitomi Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yoshitomi Pharmaceutical filed Critical Yoshitomi Pharmaceutical
Publication of ID21775A publication Critical patent/ID21775A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epoxy Compounds (AREA)
IDW990226A 1996-10-25 1996-10-25 Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya ID21775A (id)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP28447996 1996-10-25
JP5578697 1997-03-11
JP26130597 1997-09-26

Publications (1)

Publication Number Publication Date
ID21775A true ID21775A (id) 1999-07-22

Family

ID=27295710

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW990226A ID21775A (id) 1996-10-25 1996-10-25 Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya

Country Status (16)

Country Link
US (1) US6015829A (id)
EP (1) EP0936217B1 (id)
JP (1) JP3220987B2 (id)
KR (1) KR100345942B1 (id)
CN (1) CN1105708C (id)
AT (1) ATE208379T1 (id)
AU (1) AU731055B2 (id)
CA (1) CA2269721C (id)
DE (1) DE69708142T2 (id)
DK (1) DK0936217T3 (id)
ES (1) ES2167720T3 (id)
ID (1) ID21775A (id)
IL (1) IL129409A (id)
PL (1) PL332946A1 (id)
PT (1) PT936217E (id)
WO (1) WO1998018765A1 (id)

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ES2331579T3 (es) 2004-08-27 2010-01-08 Astellas Pharma Inc. Derivado de 2-fenilpiridina.
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WO2007019153A2 (en) * 2005-08-03 2007-02-15 Tap Pharmaceutical Products, Inc. Methods for treating hypertension
US7947707B2 (en) 2005-10-07 2011-05-24 Kissei Pharmaceutical Co., Ltd. Nitrogenated heterocyclic compound and pharmaceutical composition comprising the same
US7816558B2 (en) 2005-10-07 2010-10-19 Astellas Pharma Inc. Triarylcarboxylic acid derivative
ATE555810T1 (de) * 2006-02-24 2012-05-15 Astellas Pharma Inc Mittel zur behandlung oder prävention von verdauungsgeschwüren
WO2008010315A1 (en) 2006-07-19 2008-01-24 Nippon Medical School Foundation Therapeutic agent for amyotrophic lateral sclerosis
BRPI0718611A2 (pt) * 2006-11-13 2014-02-25 Takeda Pharmaceuticals North America Inc Métodos para preservar a função renal utilizando inibidores da xantina oxidoredutase.
US20090124623A1 (en) * 2006-11-13 2009-05-14 Christopher Lademacher Methods for preserving and/or increasing renal function using xanthine oxidoreductase inhibitors
EP2120956A4 (en) * 2007-01-19 2010-01-20 Takeda Pharmaceuticals North A METHODS FOR PREVENTING OR REDUCING THE NUMBER OF DROUGHT ERYTHEMES USING XANTHINE OXYDOREDUCTASE INHIBITORS AND INFLAMMATORY AGENTS
EP2133331A4 (en) * 2007-04-11 2011-06-22 Kissei Pharmaceutical FIVE-GLASS HETEROCYCLIC DERIVATIVE AND ITS USE IN MEDICAL PURPOSES
BRPI0810524B8 (pt) * 2007-04-11 2021-05-25 Kissei Pharmaceutical derivado de (aza)indol, inibidor de xantina oxidase e composição farmacêutica compreendendo o dito derivado
JP5330990B2 (ja) * 2007-04-11 2013-10-30 キッセイ薬品工業株式会社 含窒素複素環化合物およびそれを含有する医薬組成物
CN101386605B (zh) * 2008-10-23 2010-09-08 中国科学院上海药物研究所 非布司他新型晶体及其制备方法
US20100311756A1 (en) * 2009-01-22 2010-12-09 Takeda Pharmaceuticals North America, Inc. Methods for delaying the progression of at least one of cardiac hypertrophy, cardiac remodeling or left ventricular function or the onset of heart failure in subjects in need of treatment thereof
PL2404908T3 (pl) 2009-02-27 2014-12-31 Teijin Ltd Sposób wytwarzania podstawionej fenylem pochodnej heterocyklicznej przez sprzężenie z użyciem katalizatora metalu przejściowego
CN101580495A (zh) * 2009-05-25 2009-11-18 沈阳药科大学 5-取代苯基-3-异噁唑甲酸及其酯类化合物、组合物及其制备方法
TWI423962B (zh) 2009-10-07 2014-01-21 Lg Life Sciences Ltd 有效作為黃嘌呤氧化酶抑制劑之新穎化合物、其製備方法及含該化合物之醫藥組成物
MX339829B (es) * 2010-02-19 2016-06-13 Takeda Pharmaceuticals Usa Inc Metodo para estabilizar daño de articulacion en sujetos utilizando inhibidores de xantina oxidoreductasa.
SG187843A1 (en) 2010-08-27 2013-03-28 Teijin Pharma Ltd Method for producing phenyl-substituted heterocyclic derivative by means of coupling method using a palladium compound
WO2012033941A1 (en) 2010-09-10 2012-03-15 Takeda Pharmaceuticals North America, Inc. Methods for concomitant treatment of theophylline and febuxostat
CN102766099B (zh) * 2012-08-07 2015-09-23 沈阳药科大学 具有黄嘌呤氧化酶抑制活性的化合物及其盐、制备方法和用途
CN103848798B (zh) 2012-11-30 2016-01-06 镇江新元素医药科技有限公司 2-芳基硒唑化合物及其药物组合物
PT2980085T (pt) 2013-03-29 2018-04-09 Teijin Pharma Ltd Compostos farmaceuticamente activos
CN105294584A (zh) * 2015-11-30 2016-02-03 中国医科大学 1-取代苯基-1h-1,2,3-三唑类化合物、制备方法及其用途
CN106279024B (zh) * 2016-07-19 2018-09-14 华南理工大学 一种黄嘌呤氧化还原酶抑制剂及其制备方法与应用
CN106632245B (zh) * 2016-09-30 2019-11-15 华南理工大学 氮取代基苯基吡唑类黄嘌呤氧化还原酶抑制剂及制备与应用
CN108218777A (zh) * 2017-12-13 2018-06-29 华南理工大学 一种硫取代苯基吡唑类xor抑制剂及制备与应用
CN110078668B (zh) * 2019-05-16 2023-03-24 华南理工大学 一种苯基咪唑类xor抑制剂及制备与应用
CN119431324B (zh) * 2024-10-23 2025-10-31 沈阳药科大学 1-(4/5-氰基-6-取代嘧啶-2-基)-1h-吡唑-4-甲酸类化合物及其制备方法与应用

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JP3113110B2 (ja) * 1993-01-19 2000-11-27 帝人株式会社 イソキサゾールおよびイソチアゾール誘導体

Also Published As

Publication number Publication date
CN1105708C (zh) 2003-04-16
CA2269721C (en) 2003-04-29
EP0936217B1 (en) 2001-11-07
US6015829A (en) 2000-01-18
EP0936217A4 (en) 2000-01-05
AU731055B2 (en) 2001-03-22
EP0936217A1 (en) 1999-08-18
KR20000052738A (ko) 2000-08-25
AU4723097A (en) 1998-05-22
HK1021982A1 (en) 2000-07-21
PL332946A1 (en) 1999-10-25
CA2269721A1 (en) 1998-05-07
IL129409A0 (en) 2000-02-17
ES2167720T3 (es) 2002-05-16
DK0936217T3 (da) 2002-03-04
DE69708142D1 (de) 2001-12-13
WO1998018765A1 (fr) 1998-05-07
ATE208379T1 (de) 2001-11-15
JP3220987B2 (ja) 2001-10-22
PT936217E (pt) 2002-05-31
IL129409A (en) 2002-02-10
KR100345942B1 (ko) 2002-07-27
CN1240432A (zh) 2000-01-05
DE69708142T2 (de) 2002-07-11

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