HRP20110750T1 - PIPERIDINSKI AGONISTI GPCR-a - Google Patents

PIPERIDINSKI AGONISTI GPCR-a Download PDF

Info

Publication number
HRP20110750T1
HRP20110750T1 HR20110750T HRP20110750T HRP20110750T1 HR P20110750 T1 HRP20110750 T1 HR P20110750T1 HR 20110750 T HR20110750 T HR 20110750T HR P20110750 T HRP20110750 T HR P20110750T HR P20110750 T1 HRP20110750 T1 HR P20110750T1
Authority
HR
Croatia
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
isopropyl
piperidin
Prior art date
Application number
HR20110750T
Other languages
English (en)
Croatian (hr)
Inventor
Colin Thor Fyfe Matthew
Perpetua Jeevaratnam Revathy
Keily John
Andrew Swain Simon
Sarah Bertram Lisa
Original Assignee
Prosidion Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700125A external-priority patent/GB0700125D0/en
Priority claimed from GB0708746A external-priority patent/GB0708746D0/en
Priority claimed from GB0719763A external-priority patent/GB0719763D0/en
Application filed by Prosidion Limited filed Critical Prosidion Limited
Publication of HRP20110750T1 publication Critical patent/HRP20110750T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
HR20110750T 2007-01-04 2008-01-04 PIPERIDINSKI AGONISTI GPCR-a HRP20110750T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0700125A GB0700125D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708746A GB0708746D0 (en) 2007-05-08 2007-05-08 GPCR agonists
GB0719763A GB0719763D0 (en) 2007-10-10 2007-10-10 GPCR agonists
PCT/GB2008/050013 WO2008081207A1 (en) 2007-01-04 2008-01-04 Piperidine gpcr agonists

Publications (1)

Publication Number Publication Date
HRP20110750T1 true HRP20110750T1 (hr) 2011-11-30

Family

ID=39199058

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110750T HRP20110750T1 (hr) 2007-01-04 2008-01-04 PIPERIDINSKI AGONISTI GPCR-a

Country Status (20)

Country Link
US (1) US20100105732A1 (OSRAM)
EP (2) EP2114935B1 (OSRAM)
JP (1) JP2010514831A (OSRAM)
AR (1) AR064735A1 (OSRAM)
AT (1) ATE517103T1 (OSRAM)
BR (1) BRPI0806500A2 (OSRAM)
CA (1) CA2674455A1 (OSRAM)
CL (1) CL2008000018A1 (OSRAM)
CY (1) CY1112474T1 (OSRAM)
DK (1) DK2114935T3 (OSRAM)
EA (1) EA015130B1 (OSRAM)
HR (1) HRP20110750T1 (OSRAM)
PE (1) PE20081659A1 (OSRAM)
PL (1) PL2114935T3 (OSRAM)
PT (1) PT2114935E (OSRAM)
RS (1) RS51943B (OSRAM)
SA (1) SA08280757B1 (OSRAM)
SI (1) SI2114935T1 (OSRAM)
TW (1) TW200835482A (OSRAM)
WO (1) WO2008081207A1 (OSRAM)

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CL2008000017A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
EP2200609A1 (en) 2007-09-10 2010-06-30 Prosidion Limited Compounds for the treatment of metabolic disorders
JP5095824B2 (ja) 2007-10-10 2012-12-12 ノバルティス アーゲー スピロピロリジン類およびｈｃｖおよびｈｉｖ感染に対するその使用
GB0812649D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
GB0812641D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
GB0812648D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
ES2403120T3 (es) 2008-12-24 2013-05-14 Cadila Healthcare Limited Nuevos derivados de oxima
GB0904284D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
GB0904287D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
GB0904285D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
BR112012000831A2 (pt) 2009-06-24 2019-09-24 Boehringer Ingelheim Int compostos, composições farmacêuticas e métodos relacionados
TW201113269A (en) 2009-06-24 2011-04-16 Boehringer Ingelheim Int New compounds, pharmaceutical composition and methods relating thereto
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
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GB201006166D0 (en) 2010-04-14 2010-05-26 Prosidion Ltd Compounds for the treatment of metabolic disorders
GB201006167D0 (en) 2010-04-14 2010-05-26 Prosidion Ltd Compounds for the treatment of metabolic disorders
TW201209054A (en) 2010-05-28 2012-03-01 Prosidion Ltd Novel compounds
EP2582709B1 (de) 2010-06-18 2018-01-24 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
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AR083904A1 (es) 2010-11-18 2013-04-10 Prosidion Ltd Derivados de 1,4-pirrolidinas disustituidos y 3-il-aminas y sus usos en el tratamiento de desordenes metabolicos
GB201114389D0 (en) 2011-08-22 2011-10-05 Prosidion Ltd Novel compounds
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Also Published As

Publication number Publication date
CA2674455A1 (en) 2008-07-10
EP2114935B1 (en) 2011-07-20
RS51943B (sr) 2012-02-29
ATE517103T1 (de) 2011-08-15
EP2377864A1 (en) 2011-10-19
PT2114935E (pt) 2011-10-17
DK2114935T3 (da) 2011-10-31
PL2114935T3 (pl) 2012-03-30
US20100105732A1 (en) 2010-04-29
BRPI0806500A2 (pt) 2014-04-22
SI2114935T1 (sl) 2011-11-30
AR064735A1 (es) 2009-04-22
PE20081659A1 (es) 2008-10-24
EP2114935A1 (en) 2009-11-11
CL2008000018A1 (es) 2008-08-01
CY1112474T1 (el) 2015-12-09
WO2008081207A1 (en) 2008-07-10
EA015130B1 (ru) 2011-06-30
EA200900880A1 (ru) 2010-02-26
HK1135705A1 (en) 2010-06-11
JP2010514831A (ja) 2010-05-06
TW200835482A (en) 2008-09-01
SA08280757B1 (ar) 2011-01-15

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