PE20081659A1 - Agonistas de gpcr - Google Patents

Agonistas de gpcr

Info

Publication number
PE20081659A1
PE20081659A1 PE2008000084A PE2008000084A PE20081659A1 PE 20081659 A1 PE20081659 A1 PE 20081659A1 PE 2008000084 A PE2008000084 A PE 2008000084A PE 2008000084 A PE2008000084 A PE 2008000084A PE 20081659 A1 PE20081659 A1 PE 20081659A1
Authority
PE
Peru
Prior art keywords
oxadiazol
piperidin
compounds
propoxi
isopropyl
Prior art date
Application number
PE2008000084A
Other languages
English (en)
Spanish (es)
Inventor
Lisa Sarah Bertram
Matthew Colin Thor Fyfe
John Keily
Simon Andrew Swain
Revathy Perpetua Jeevaratnam
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700125A external-priority patent/GB0700125D0/en
Priority claimed from GB0708746A external-priority patent/GB0708746D0/en
Priority claimed from GB0719763A external-priority patent/GB0719763D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Publication of PE20081659A1 publication Critical patent/PE20081659A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
PE2008000084A 2007-01-04 2008-01-03 Agonistas de gpcr PE20081659A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0700125A GB0700125D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708746A GB0708746D0 (en) 2007-05-08 2007-05-08 GPCR agonists
GB0719763A GB0719763D0 (en) 2007-10-10 2007-10-10 GPCR agonists

Publications (1)

Publication Number Publication Date
PE20081659A1 true PE20081659A1 (es) 2008-10-24

Family

ID=39199058

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2008000084A PE20081659A1 (es) 2007-01-04 2008-01-03 Agonistas de gpcr

Country Status (20)

Country Link
US (1) US20100105732A1 (OSRAM)
EP (2) EP2377864A1 (OSRAM)
JP (1) JP2010514831A (OSRAM)
AR (1) AR064735A1 (OSRAM)
AT (1) ATE517103T1 (OSRAM)
BR (1) BRPI0806500A2 (OSRAM)
CA (1) CA2674455A1 (OSRAM)
CL (1) CL2008000018A1 (OSRAM)
CY (1) CY1112474T1 (OSRAM)
DK (1) DK2114935T3 (OSRAM)
EA (1) EA015130B1 (OSRAM)
HR (1) HRP20110750T1 (OSRAM)
PE (1) PE20081659A1 (OSRAM)
PL (1) PL2114935T3 (OSRAM)
PT (1) PT2114935E (OSRAM)
RS (1) RS51943B (OSRAM)
SA (1) SA08280757B1 (OSRAM)
SI (1) SI2114935T1 (OSRAM)
TW (1) TW200835482A (OSRAM)
WO (1) WO2008081207A1 (OSRAM)

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US20100063081A1 (en) * 2005-06-30 2010-03-11 Stuart Edward Bradly CPCR Agonists
CL2008000017A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
US20100286112A1 (en) 2007-09-10 2010-11-11 Oscar Barba Compounds for the treatment of metabolic disorders
CN101868452B (zh) 2007-10-10 2014-08-06 诺华股份有限公司 螺环吡咯烷类与其对抗hcv和hiv感染的应用
GB0812649D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
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GB0812648D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
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GB0904284D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
GB0904285D0 (en) * 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
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TW201113269A (en) 2009-06-24 2011-04-16 Boehringer Ingelheim Int New compounds, pharmaceutical composition and methods relating thereto
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WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
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CN104610393A (zh) * 2015-02-13 2015-05-13 佛山市赛维斯医药科技有限公司 一类含氨基葡萄糖和卤代吡啶结构化合物及其用途
CN104610390A (zh) * 2015-02-13 2015-05-13 佛山市赛维斯医药科技有限公司 一种含氨基葡萄糖和腈基吡啶结构的gpr119激动剂及其用途

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Also Published As

Publication number Publication date
EP2377864A1 (en) 2011-10-19
CA2674455A1 (en) 2008-07-10
SA08280757B1 (ar) 2011-01-15
PL2114935T3 (pl) 2012-03-30
SI2114935T1 (sl) 2011-11-30
HK1135705A1 (en) 2010-06-11
JP2010514831A (ja) 2010-05-06
BRPI0806500A2 (pt) 2014-04-22
ATE517103T1 (de) 2011-08-15
EP2114935A1 (en) 2009-11-11
US20100105732A1 (en) 2010-04-29
TW200835482A (en) 2008-09-01
PT2114935E (pt) 2011-10-17
DK2114935T3 (da) 2011-10-31
AR064735A1 (es) 2009-04-22
CL2008000018A1 (es) 2008-08-01
EP2114935B1 (en) 2011-07-20
CY1112474T1 (el) 2015-12-09
EA015130B1 (ru) 2011-06-30
WO2008081207A1 (en) 2008-07-10
RS51943B (sr) 2012-02-29
EA200900880A1 (ru) 2010-02-26
HRP20110750T1 (hr) 2011-11-30

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