DK2114935T3 - Piperidin-GPCR-agonister - Google Patents

Piperidin-GPCR-agonister

Info

Publication number
DK2114935T3
DK2114935T3 DK08702096.2T DK08702096T DK2114935T3 DK 2114935 T3 DK2114935 T3 DK 2114935T3 DK 08702096 T DK08702096 T DK 08702096T DK 2114935 T3 DK2114935 T3 DK 2114935T3
Authority
DK
Denmark
Prior art keywords
gpcr agonists
piperidine
piperidine gpcr
agonists
gpcr
Prior art date
Application number
DK08702096.2T
Other languages
English (en)
Inventor
John Keily
Lisa Sarah Bertram
Matthew Colin Thor Fyfe
Revathy Perpetua Jeevaratnam
Simon Andrew Swain
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700125A external-priority patent/GB0700125D0/en
Priority claimed from GB0708746A external-priority patent/GB0708746D0/en
Priority claimed from GB0719763A external-priority patent/GB0719763D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Application granted granted Critical
Publication of DK2114935T3 publication Critical patent/DK2114935T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
DK08702096.2T 2007-01-04 2008-01-04 Piperidin-GPCR-agonister DK2114935T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0700125A GB0700125D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708746A GB0708746D0 (en) 2007-05-08 2007-05-08 GPCR agonists
GB0719763A GB0719763D0 (en) 2007-10-10 2007-10-10 GPCR agonists
PCT/GB2008/050013 WO2008081207A1 (en) 2007-01-04 2008-01-04 Piperidine gpcr agonists

Publications (1)

Publication Number Publication Date
DK2114935T3 true DK2114935T3 (da) 2011-10-31

Family

ID=39199058

Family Applications (1)

Application Number Title Priority Date Filing Date
DK08702096.2T DK2114935T3 (da) 2007-01-04 2008-01-04 Piperidin-GPCR-agonister

Country Status (21)

Country Link
US (1) US20100105732A1 (da)
EP (2) EP2114935B1 (da)
JP (1) JP2010514831A (da)
AR (1) AR064735A1 (da)
AT (1) ATE517103T1 (da)
BR (1) BRPI0806500A2 (da)
CA (1) CA2674455A1 (da)
CL (1) CL2008000018A1 (da)
CY (1) CY1112474T1 (da)
DK (1) DK2114935T3 (da)
EA (1) EA015130B1 (da)
HK (1) HK1135705A1 (da)
HR (1) HRP20110750T1 (da)
PE (1) PE20081659A1 (da)
PL (1) PL2114935T3 (da)
PT (1) PT2114935E (da)
RS (1) RS51943B (da)
SA (1) SA08280757B1 (da)
SI (1) SI2114935T1 (da)
TW (1) TW200835482A (da)
WO (1) WO2008081207A1 (da)

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BRPI0516407A (pt) * 2004-12-24 2008-09-02 Prosidion Ltd agonistas de receptor acoplado à proteìna g (gpr116) e uso destes para o tratamento de obesidade e diabetes
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GB0904284D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
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GB0904285D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
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WO2010149685A1 (en) 2009-06-24 2010-12-29 Boehringer Ingelheim International Gmbh New compounds, pharmaceutical composition and methods relating thereto
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GB201006167D0 (en) 2010-04-14 2010-05-26 Prosidion Ltd Compounds for the treatment of metabolic disorders
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JP6463631B2 (ja) 2011-06-09 2019-02-06 ライゼン・ファーマシューティカルズ・エスアー Ｇｐｒ−１１９のモジュレータとしての新規化合物
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CN104610393A (zh) * 2015-02-13 2015-05-13 佛山市赛维斯医药科技有限公司 一类含氨基葡萄糖和卤代吡啶结构化合物及其用途
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Also Published As

Publication number Publication date
CA2674455A1 (en) 2008-07-10
EP2114935B1 (en) 2011-07-20
PL2114935T3 (pl) 2012-03-30
BRPI0806500A2 (pt) 2014-04-22
EP2377864A1 (en) 2011-10-19
PT2114935E (pt) 2011-10-17
PE20081659A1 (es) 2008-10-24
CY1112474T1 (el) 2015-12-09
WO2008081207A1 (en) 2008-07-10
EA015130B1 (ru) 2011-06-30
SI2114935T1 (sl) 2011-11-30
EA200900880A1 (ru) 2010-02-26
HK1135705A1 (en) 2010-06-11
TW200835482A (en) 2008-09-01
EP2114935A1 (en) 2009-11-11
AR064735A1 (es) 2009-04-22
JP2010514831A (ja) 2010-05-06
RS51943B (en) 2012-02-29
ATE517103T1 (de) 2011-08-15
US20100105732A1 (en) 2010-04-29
CL2008000018A1 (es) 2008-08-01
HRP20110750T1 (hr) 2011-11-30
SA08280757B1 (ar) 2011-01-15

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