DK2181990T3 - Piperidinderivat - Google Patents

Piperidinderivat

Info

Publication number
DK2181990T3
DK2181990T3 DK08828181.1T DK08828181T DK2181990T3 DK 2181990 T3 DK2181990 T3 DK 2181990T3 DK 08828181 T DK08828181 T DK 08828181T DK 2181990 T3 DK2181990 T3 DK 2181990T3
Authority
DK
Denmark
Prior art keywords
piperidine
Prior art date
Application number
DK08828181.1T
Other languages
English (en)
Inventor
Akio Kakefuda
Kazushi Watanabe
Akio Kamikawa
Kentaro Enjo
Takashi Furutani
Minoru Yasuda
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Application granted granted Critical
Publication of DK2181990T3 publication Critical patent/DK2181990T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4465Non condensed piperidines, e.g. piperocaine only substituted in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/08Antiseborrheics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
DK08828181.1T 2007-08-31 2008-08-28 Piperidinderivat DK2181990T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007225378 2007-08-31
PCT/JP2008/065429 WO2009028618A1 (ja) 2007-08-31 2008-08-28 ピペリジン誘導体

Publications (1)

Publication Number Publication Date
DK2181990T3 true DK2181990T3 (da) 2012-09-10

Family

ID=40387332

Family Applications (1)

Application Number Title Priority Date Filing Date
DK08828181.1T DK2181990T3 (da) 2007-08-31 2008-08-28 Piperidinderivat

Country Status (20)

Country Link
US (1) US8513422B2 (da)
EP (1) EP2181990B1 (da)
JP (1) JP5327051B2 (da)
KR (1) KR20100050444A (da)
CN (1) CN101821253B (da)
AU (1) AU2008292420A1 (da)
BR (1) BRPI0815787A2 (da)
CA (1) CA2696799A1 (da)
CY (1) CY1113417T1 (da)
DK (1) DK2181990T3 (da)
ES (1) ES2392120T3 (da)
HR (1) HRP20120837T1 (da)
MX (1) MX2010002268A (da)
PL (1) PL2181990T3 (da)
PT (1) PT2181990E (da)
RU (1) RU2470020C2 (da)
SI (1) SI2181990T1 (da)
TW (1) TW200924765A (da)
WO (1) WO2009028618A1 (da)
ZA (1) ZA201000917B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5609150B2 (ja) * 2009-02-27 2014-10-22 アステラス製薬株式会社 ピペリジン誘導体
JP2012102017A (ja) * 2009-03-03 2012-05-31 Astellas Pharma Inc インドール化合物
JP2012102018A (ja) * 2009-03-03 2012-05-31 Astellas Pharma Inc アミド化合物
JP5851998B2 (ja) * 2009-10-27 2016-02-03 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺虫剤および殺ダニ剤としてのハロアルキル置換アミド

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9116732D0 (en) * 1991-08-02 1991-09-18 Fujisawa Pharmaceutical Co Indole derivatives
AU680870B2 (en) * 1993-04-28 1997-08-14 Astellas Pharma Inc. New heterocyclic compounds
WO1998028292A1 (en) 1996-12-23 1998-07-02 Smithkline Beecham Corporation Novel piperidine containing compounds
CN1429104A (zh) 1998-03-11 2003-07-09 内部研究股份有限公司 5型和3型17β-羟基类固醇脱氢酶的抑制剂及其用法
EP1102582A2 (en) * 1998-08-07 2001-05-30 Endorecherche Inc. Inhibitors of type 3 3alpha-hydroxysteroid dehydrogenase
EP1341761A1 (en) * 2000-10-10 2003-09-10 Smithkline Beecham Corporation SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS
WO2002072548A2 (en) 2001-03-09 2002-09-19 Ortho-Mcneil Pharmaceutical, Inc. Heterocyclic compounds and their use as histamine h4 ligands.
US7129225B2 (en) 2001-10-22 2006-10-31 The Research Foundation Of State University Of New York Protection against and treatment of hearing loss
AU2002360561A1 (en) 2001-12-11 2003-06-23 Sepracor, Inc. 4-substituted piperidines, and methods of use thereof
WO2004064736A2 (en) 2003-01-17 2004-08-05 Threshold Pharmaceuticals, Inc. Treatment of benign prostatic hyperplasia using energolytic agents
JP4629657B2 (ja) 2003-04-11 2011-02-09 ハイ・ポイント・ファーマスーティカルズ、エルエルシー 11β−ヒドロキシステロイドデヒドロゲナーゼ1型化活性化合物
AU2004268949A1 (en) 2003-08-21 2005-03-10 Osi Pharmaceuticals, Inc. N-substituted benzimidazolyl C-kit inhibitors
WO2005040112A1 (en) * 2003-10-14 2005-05-06 Oxagen Limited Compounds with pgd2 antagonist activity
JP2005162657A (ja) 2003-12-02 2005-06-23 Takeda Chem Ind Ltd カンナビノイド受容体調節剤
JPWO2005082905A1 (ja) * 2004-02-26 2007-08-02 協和醗酵工業株式会社 二環性複素環化合物
CA2564953A1 (en) * 2004-05-03 2005-11-24 Janssen Pharmaceutica N.V. Novel indole derivatives as selective androgen receptor modulators (sarms)
US7288553B2 (en) * 2004-05-03 2007-10-30 Janssen Pharmaceutica N.V. Indole derivatives as selective androgen receptor modulator (SARMS)
AU2005254658B2 (en) * 2004-06-21 2011-06-16 F. Hoffmann-La Roche Ag Indole derivatives as histamine receptor antagonists
JP2009509932A (ja) 2005-09-07 2009-03-12 プレキシコン,インコーポレーテッド Ppar活性化合物
WO2007056155A1 (en) 2005-11-03 2007-05-18 Chembridge Research Laboratories, Inc. Heterocyclic compounds as tyrosine kinase modulators
WO2007100066A1 (ja) * 2006-03-02 2007-09-07 Astellas Pharma Inc. 17βHSDtype5阻害剤

Also Published As

Publication number Publication date
EP2181990A1 (en) 2010-05-05
EP2181990B1 (en) 2012-08-08
CN101821253A (zh) 2010-09-01
US8513422B2 (en) 2013-08-20
SI2181990T1 (sl) 2012-10-30
RU2470020C2 (ru) 2012-12-20
WO2009028618A1 (ja) 2009-03-05
JPWO2009028618A1 (ja) 2010-12-02
ES2392120T3 (es) 2012-12-04
US20100256189A1 (en) 2010-10-07
TW200924765A (en) 2009-06-16
CA2696799A1 (en) 2009-03-05
PT2181990E (pt) 2012-10-16
CY1113417T1 (el) 2016-06-22
PL2181990T3 (pl) 2013-01-31
RU2010112412A (ru) 2011-10-10
HRP20120837T1 (hr) 2012-11-30
CN101821253B (zh) 2013-07-17
ZA201000917B (en) 2011-04-28
EP2181990A4 (en) 2011-09-07
KR20100050444A (ko) 2010-05-13
JP5327051B2 (ja) 2013-10-30
BRPI0815787A2 (pt) 2015-02-24
MX2010002268A (es) 2010-03-25
AU2008292420A1 (en) 2009-03-05

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