HK1137448A1 - Serine-threonine protein kinase and parp modulators - parp - Google Patents

Serine-threonine protein kinase and parp modulators - parp

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Publication number
HK1137448A1
HK1137448A1 HK10102364.2A HK10102364A HK1137448A1 HK 1137448 A1 HK1137448 A1 HK 1137448A1 HK 10102364 A HK10102364 A HK 10102364A HK 1137448 A1 HK1137448 A1 HK 1137448A1
Authority
HK
Hong Kong
Prior art keywords
parp
serine
protein kinase
modulators
threonine protein
Prior art date
Application number
HK10102364.2A
Other languages
English (en)
Chinese (zh)
Inventor
‧楚埃
‧皮埃爾
‧惠藤
Original Assignee
生華生物科技股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 生華生物科技股份有限公司 filed Critical 生華生物科技股份有限公司
Publication of HK1137448A1 publication Critical patent/HK1137448A1/xx

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    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
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    • C07D221/18—Ring systems of four or more rings
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
HK10102364.2A 2006-09-01 2010-03-05 Serine-threonine protein kinase and parp modulators - parp HK1137448A1 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US84206106P 2006-09-01 2006-09-01
US84454206P 2006-09-13 2006-09-13
US84668306P 2006-09-22 2006-09-22
US87393606P 2006-12-07 2006-12-07
US89571607P 2007-03-19 2007-03-19
PCT/US2007/077464 WO2008028168A2 (en) 2006-09-01 2007-08-31 Serine-threonine protein kinase and parp modulators

Publications (1)

Publication Number Publication Date
HK1137448A1 true HK1137448A1 (en) 2010-07-30

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
HK10102364.2A HK1137448A1 (en) 2006-09-01 2010-03-05 Serine-threonine protein kinase and parp modulators - parp

Country Status (17)

Country Link
US (2) US7956064B2 (ja)
EP (1) EP2061765B1 (ja)
JP (1) JP5399905B2 (ja)
KR (1) KR20090050094A (ja)
AU (1) AU2007289065B2 (ja)
BR (1) BRPI0719123A2 (ja)
CA (2) CA2974246C (ja)
DK (1) DK2061765T3 (ja)
ES (1) ES2528316T3 (ja)
HK (1) HK1137448A1 (ja)
IL (1) IL197088A0 (ja)
MX (1) MX2009002298A (ja)
NO (1) NO20090854L (ja)
PL (1) PL2061765T3 (ja)
PT (1) PT2061765E (ja)
RU (1) RU2681209C2 (ja)
WO (1) WO2008028168A2 (ja)

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EP2004654B1 (en) 2006-04-04 2013-05-22 The Regents of the University of California Pyrazolopyrimidine derivatives for use as kinase antagonists
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