HK1121169A1 - Hcv ns3 protease inhibitors hcv ns3 - Google Patents
Hcv ns3 protease inhibitors hcv ns3Info
- Publication number
- HK1121169A1 HK1121169A1 HK08112711.5A HK08112711A HK1121169A1 HK 1121169 A1 HK1121169 A1 HK 1121169A1 HK 08112711 A HK08112711 A HK 08112711A HK 1121169 A1 HK1121169 A1 HK 1121169A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- hcv
- protease inhibitors
- protease
- inhibitors
- inhibitors hcv
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/18—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US70076405P | 2005-07-20 | 2005-07-20 | |
US72456605P | 2005-10-07 | 2005-10-07 | |
PCT/US2006/027831 WO2007015855A1 (en) | 2005-07-20 | 2006-07-14 | Hcv ns3 protease inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1121169A1 true HK1121169A1 (en) | 2009-04-17 |
Family
ID=37467463
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK08112711.5A HK1121169A1 (en) | 2005-07-20 | 2008-11-20 | Hcv ns3 protease inhibitors hcv ns3 |
Country Status (38)
Country | Link |
---|---|
US (2) | US7470664B2 (de) |
EP (2) | EP1924593B9 (de) |
JP (2) | JP4621282B2 (de) |
KR (1) | KR101296095B1 (de) |
AR (1) | AR057456A1 (de) |
AT (1) | ATE443075T1 (de) |
AU (1) | AU2006276189B9 (de) |
BR (1) | BRPI0613633A2 (de) |
CA (1) | CA2615022C (de) |
CR (1) | CR9621A (de) |
CY (1) | CY1109671T1 (de) |
DE (1) | DE602006009280D1 (de) |
DK (1) | DK1924593T3 (de) |
DO (2) | DOP2006000171A (de) |
EA (1) | EA013331B1 (de) |
EC (1) | ECSP088107A (de) |
ES (2) | ES2332821T3 (de) |
GE (1) | GEP20115248B (de) |
GT (1) | GT200600317A (de) |
HK (1) | HK1121169A1 (de) |
HN (1) | HN2008000087A (de) |
HR (1) | HRP20090627T1 (de) |
IL (1) | IL188618A0 (de) |
JO (1) | JO2593B1 (de) |
MA (1) | MA30198B1 (de) |
MX (1) | MX2008000866A (de) |
MY (1) | MY142240A (de) |
NO (1) | NO20080879L (de) |
NZ (1) | NZ565223A (de) |
PE (1) | PE20070364A1 (de) |
PL (1) | PL1924593T3 (de) |
PT (1) | PT1924593E (de) |
RS (1) | RS51101B (de) |
SG (1) | SG164376A1 (de) |
SI (1) | SI1924593T1 (de) |
TN (1) | TNSN08033A1 (de) |
TW (1) | TWI387603B (de) |
WO (2) | WO2007015787A1 (de) |
Families Citing this family (110)
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EP1905777B2 (de) * | 2005-07-04 | 2018-06-27 | Zannan Scitech Co., Ltd. | Rutheniumkomplexligand, rutheniumkomplex, geträgerter rutheniumkomplexkatalysator und herstellungsverfahren und anwendung davon |
US7470664B2 (en) * | 2005-07-20 | 2008-12-30 | Merck & Co., Inc. | HCV NS3 protease inhibitors |
EP1924594A2 (de) * | 2005-07-25 | 2008-05-28 | Intermune, Inc. | Neue makrocyclische inhibitoren der replikation des hepatitis-c-virus |
JP4705984B2 (ja) * | 2005-08-01 | 2011-06-22 | メルク・シャープ・エンド・ドーム・コーポレイション | Hcvns3プロテアーゼ阻害剤としての大環状ペプチド |
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