HK1058201A1 - Novel indole derivatives and their use as medicaments - Google Patents

Novel indole derivatives and their use as medicaments

Info

Publication number
HK1058201A1
HK1058201A1 HK04100997A HK04100997A HK1058201A1 HK 1058201 A1 HK1058201 A1 HK 1058201A1 HK 04100997 A HK04100997 A HK 04100997A HK 04100997 A HK04100997 A HK 04100997A HK 1058201 A1 HK1058201 A1 HK 1058201A1
Authority
HK
Hong Kong
Prior art keywords
medicaments
indole derivatives
novel indole
novel
derivatives
Prior art date
Application number
HK04100997A
Other languages
English (en)
Inventor
Peter Emig
Gerald Bacher
Dietmar Reichert
Silke Baasner
Beate Aue
Bernd Nickel
Eckhard Gunther
Original Assignee
Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh filed Critical Zentaris Gmbh
Publication of HK1058201A1 publication Critical patent/HK1058201A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK04100997A 2000-07-28 2004-02-13 Novel indole derivatives and their use as medicaments HK1058201A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10037310A DE10037310A1 (de) 2000-07-28 2000-07-28 Neue Indolderivate und deren Verwendung als Arzneimittel
PCT/EP2001/008644 WO2002010152A2 (de) 2000-07-28 2001-07-26 Neue indolderivate und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
HK1058201A1 true HK1058201A1 (en) 2004-05-07

Family

ID=7650860

Family Applications (1)

Application Number Title Priority Date Filing Date
HK04100997A HK1058201A1 (en) 2000-07-28 2004-02-13 Novel indole derivatives and their use as medicaments

Country Status (31)

Country Link
US (3) US7365081B2 (ja)
EP (3) EP2163552A1 (ja)
JP (1) JP5113973B2 (ja)
KR (1) KR100810453B1 (ja)
CN (1) CN1215066C (ja)
AR (1) AR055209A1 (ja)
AT (1) ATE392420T1 (ja)
AU (2) AU8975801A (ja)
BG (1) BG66457B1 (ja)
BR (1) BR0112807A (ja)
CA (3) CA2354210C (ja)
CY (1) CY1108770T1 (ja)
CZ (1) CZ304197B6 (ja)
DE (2) DE10037310A1 (ja)
DK (1) DK1309585T3 (ja)
ES (1) ES2303532T3 (ja)
HK (1) HK1058201A1 (ja)
HU (1) HU229254B1 (ja)
IL (2) IL153930A0 (ja)
MX (1) MXPA03000644A (ja)
NO (1) NO324594B1 (ja)
NZ (1) NZ524404A (ja)
PL (1) PL208673B1 (ja)
PT (1) PT1309585E (ja)
RU (1) RU2270196C9 (ja)
SI (1) SI1309585T1 (ja)
SK (1) SK288085B6 (ja)
TW (1) TWI291955B (ja)
UA (1) UA80670C2 (ja)
WO (1) WO2002010152A2 (ja)
ZA (1) ZA200300584B (ja)

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EP1484329A1 (de) * 2003-06-06 2004-12-08 Zentaris GmbH Indolderivate mit Apoptose induzierender Wirkung
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US7211588B2 (en) * 2003-07-25 2007-05-01 Zentaris Gmbh N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation
US20050124623A1 (en) 2003-11-26 2005-06-09 Bender John A. Diazaindole-dicarbonyl-piperazinyl antiviral agents
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US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
GB2431927B (en) 2005-11-04 2010-03-17 Amira Pharmaceuticals Inc 5-Lipoxygenase-activating protein (FLAP) inhibitors
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
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US7807671B2 (en) 2006-04-25 2010-10-05 Bristol-Myers Squibb Company Diketo-piperazine and piperidine derivatives as antiviral agents
EP2610244A1 (en) 2006-08-07 2013-07-03 Ironwood Pharmaceuticals, Inc. Indole compounds
AU2009325091A1 (en) 2008-05-23 2010-06-17 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein inhibitor
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen

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EA003876B1 (ru) 1998-02-25 2003-10-30 Дженетикс Инститьют, Ллс Ингибиторы фосфолипазных ферментов
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Also Published As

Publication number Publication date
NO324594B1 (no) 2007-11-26
AU2001289758B2 (en) 2006-07-06
US7989453B2 (en) 2011-08-02
KR20030017658A (ko) 2003-03-03
DE50113867D1 (de) 2008-05-29
MXPA03000644A (es) 2003-06-06
EP2163552A1 (de) 2010-03-17
SK2222003A3 (en) 2004-04-06
HUP0300677A2 (hu) 2003-11-28
EP1939195A1 (de) 2008-07-02
CA2354210C (en) 2010-09-14
NO20030382L (no) 2003-02-20
SK288085B6 (sk) 2013-06-03
IL153930A (en) 2008-11-03
DE10037310A1 (de) 2002-02-07
NO20030382D0 (no) 2003-01-24
CY1108770T1 (el) 2014-04-09
AU8975801A (en) 2002-02-13
ES2303532T3 (es) 2008-08-16
CN1447805A (zh) 2003-10-08
US20030100597A1 (en) 2003-05-29
US20080108819A1 (en) 2008-05-08
WO2002010152A2 (de) 2002-02-07
IL153930A0 (en) 2003-07-31
RU2270196C2 (ru) 2006-02-20
CA2354210A1 (en) 2002-01-28
KR100810453B1 (ko) 2008-03-07
CA2704691A1 (en) 2002-01-28
PT1309585E (pt) 2008-06-09
CZ304197B6 (cs) 2013-12-27
RU2270196C9 (ru) 2007-11-27
CN1215066C (zh) 2005-08-17
HU229254B1 (en) 2013-10-28
PL361356A1 (en) 2004-10-04
BG107560A (bg) 2003-10-31
ZA200300584B (en) 2003-07-18
BR0112807A (pt) 2003-07-01
US7365081B2 (en) 2008-04-29
ATE392420T1 (de) 2008-05-15
JP5113973B2 (ja) 2013-01-09
TWI291955B (en) 2008-01-01
PL208673B1 (pl) 2011-05-31
US8008324B2 (en) 2011-08-30
UA80670C2 (en) 2007-10-25
EP1309585B1 (de) 2008-04-16
CZ2003500A3 (cs) 2004-03-17
JP2004505075A (ja) 2004-02-19
DK1309585T3 (da) 2008-06-23
CA2704693A1 (en) 2002-01-28
US20080153875A1 (en) 2008-06-26
BG66457B1 (bg) 2014-10-31
EP1309585A2 (de) 2003-05-14
WO2002010152A3 (de) 2002-08-01
SI1309585T1 (sl) 2008-08-31
NZ524404A (en) 2004-08-27
AR055209A1 (es) 2007-08-15

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20150726