PT1309585E - Novos derivados de indole e sua utilização como medicamentos - Google Patents

Novos derivados de indole e sua utilização como medicamentos Download PDF

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Publication number
PT1309585E
PT1309585E PT01969522T PT01969522T PT1309585E PT 1309585 E PT1309585 E PT 1309585E PT 01969522 T PT01969522 T PT 01969522T PT 01969522 T PT01969522 T PT 01969522T PT 1309585 E PT1309585 E PT 1309585E
Authority
PT
Portugal
Prior art keywords
medicaments
indole derivatives
novel indole
novel
derivatives
Prior art date
Application number
PT01969522T
Other languages
English (en)
Portuguese (pt)
Inventor
Peter Emig
Dietmar Reichert
Bernd Nickel
Gerald Bacher
Eckhard Guenther
Silke Baasner
Beate Aue
Original Assignee
Aeterna Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aeterna Zentaris Gmbh filed Critical Aeterna Zentaris Gmbh
Publication of PT1309585E publication Critical patent/PT1309585E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
PT01969522T 2000-07-28 2001-07-26 Novos derivados de indole e sua utilização como medicamentos PT1309585E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10037310A DE10037310A1 (de) 2000-07-28 2000-07-28 Neue Indolderivate und deren Verwendung als Arzneimittel

Publications (1)

Publication Number Publication Date
PT1309585E true PT1309585E (pt) 2008-06-09

Family

ID=7650860

Family Applications (1)

Application Number Title Priority Date Filing Date
PT01969522T PT1309585E (pt) 2000-07-28 2001-07-26 Novos derivados de indole e sua utilização como medicamentos

Country Status (31)

Country Link
US (3) US7365081B2 (ja)
EP (3) EP1309585B1 (ja)
JP (1) JP5113973B2 (ja)
KR (1) KR100810453B1 (ja)
CN (1) CN1215066C (ja)
AR (1) AR055209A1 (ja)
AT (1) ATE392420T1 (ja)
AU (2) AU8975801A (ja)
BG (1) BG66457B1 (ja)
BR (1) BR0112807A (ja)
CA (3) CA2704693A1 (ja)
CY (1) CY1108770T1 (ja)
CZ (1) CZ304197B6 (ja)
DE (2) DE10037310A1 (ja)
DK (1) DK1309585T3 (ja)
ES (1) ES2303532T3 (ja)
HK (1) HK1058201A1 (ja)
HU (1) HU229254B1 (ja)
IL (2) IL153930A0 (ja)
MX (1) MXPA03000644A (ja)
NO (1) NO324594B1 (ja)
NZ (1) NZ524404A (ja)
PL (1) PL208673B1 (ja)
PT (1) PT1309585E (ja)
RU (1) RU2270196C9 (ja)
SI (1) SI1309585T1 (ja)
SK (1) SK288085B6 (ja)
TW (1) TWI291955B (ja)
UA (1) UA80670C2 (ja)
WO (1) WO2002010152A2 (ja)
ZA (1) ZA200300584B (ja)

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EP1641777A1 (de) * 2003-06-05 2006-04-05 Zentaris GmbH Indolderivate mit apoptose induzierender wirkung
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US7211588B2 (en) * 2003-07-25 2007-05-01 Zentaris Gmbh N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation
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US7807671B2 (en) 2006-04-25 2010-10-05 Bristol-Myers Squibb Company Diketo-piperazine and piperidine derivatives as antiviral agents
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MX2010012814A (es) 2008-05-23 2010-12-20 Amira Pharmaceuticals Inc Inhibidor de proteina activadora de 5-lipoxigenasa.
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen

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US5480883A (en) * 1991-05-10 1996-01-02 Rhone-Poulenc Rorer Pharmaceuticals Inc. Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase
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Also Published As

Publication number Publication date
NZ524404A (en) 2004-08-27
US7365081B2 (en) 2008-04-29
RU2270196C9 (ru) 2007-11-27
CA2354210C (en) 2010-09-14
ATE392420T1 (de) 2008-05-15
KR100810453B1 (ko) 2008-03-07
EP1939195A1 (de) 2008-07-02
JP5113973B2 (ja) 2013-01-09
CN1447805A (zh) 2003-10-08
EP1309585A2 (de) 2003-05-14
JP2004505075A (ja) 2004-02-19
HUP0300677A2 (hu) 2003-11-28
US20080153875A1 (en) 2008-06-26
MXPA03000644A (es) 2003-06-06
UA80670C2 (en) 2007-10-25
CA2704693A1 (en) 2002-01-28
RU2270196C2 (ru) 2006-02-20
AU2001289758B2 (en) 2006-07-06
SK288085B6 (sk) 2013-06-03
BG66457B1 (bg) 2014-10-31
CA2354210A1 (en) 2002-01-28
SK2222003A3 (en) 2004-04-06
CZ304197B6 (cs) 2013-12-27
BR0112807A (pt) 2003-07-01
IL153930A (en) 2008-11-03
SI1309585T1 (sl) 2008-08-31
HK1058201A1 (en) 2004-05-07
NO20030382D0 (no) 2003-01-24
IL153930A0 (en) 2003-07-31
CN1215066C (zh) 2005-08-17
CY1108770T1 (el) 2014-04-09
KR20030017658A (ko) 2003-03-03
HU229254B1 (en) 2013-10-28
BG107560A (bg) 2003-10-31
NO324594B1 (no) 2007-11-26
ES2303532T3 (es) 2008-08-16
WO2002010152A3 (de) 2002-08-01
PL208673B1 (pl) 2011-05-31
TWI291955B (en) 2008-01-01
EP1309585B1 (de) 2008-04-16
DE10037310A1 (de) 2002-02-07
ZA200300584B (en) 2003-07-18
US7989453B2 (en) 2011-08-02
WO2002010152A2 (de) 2002-02-07
US8008324B2 (en) 2011-08-30
AU8975801A (en) 2002-02-13
PL361356A1 (en) 2004-10-04
CZ2003500A3 (cs) 2004-03-17
US20080108819A1 (en) 2008-05-08
AR055209A1 (es) 2007-08-15
NO20030382L (no) 2003-02-20
EP2163552A1 (de) 2010-03-17
DE50113867D1 (de) 2008-05-29
DK1309585T3 (da) 2008-06-23
CA2704691A1 (en) 2002-01-28
US20030100597A1 (en) 2003-05-29

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