HK1030883A1 - Preventives/remedies for glaucoma - Google Patents

Preventives/remedies for glaucoma

Info

Publication number
HK1030883A1
HK1030883A1 HK01101779A HK01101779A HK1030883A1 HK 1030883 A1 HK1030883 A1 HK 1030883A1 HK 01101779 A HK01101779 A HK 01101779A HK 01101779 A HK01101779 A HK 01101779A HK 1030883 A1 HK1030883 A1 HK 1030883A1
Authority
HK
Hong Kong
Prior art keywords
glaucoma
prophylaxis
treatment
agent
compound
Prior art date
Application number
HK01101779A
Other languages
English (en)
Inventor
Mitsuyoshi Azuma
Yukuo Yoshida
Mitsunori Waki
Masayoshi Uehata
Original Assignee
Senju Pharma Co
Mitsubishi Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senju Pharma Co, Mitsubishi Pharma Corp filed Critical Senju Pharma Co
Priority to HK05102430.9A priority Critical patent/HK1069120A1/xx
Priority to HK05102431.8A priority patent/HK1069121A1/xx
Publication of HK1030883A1 publication Critical patent/HK1030883A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4409Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 4, e.g. isoniazid, iproniazid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicinal Preparation (AREA)
  • Pyrane Compounds (AREA)
HK01101779A 1998-08-17 2001-03-12 Preventives/remedies for glaucoma HK1030883A1 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
HK05102430.9A HK1069120A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of glaucoma
HK05102431.8A HK1069121A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of asthenopia and pseudomyopia

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP24776298 1998-08-17
JP12296099 1999-04-28
PCT/JP1999/004403 WO2000009162A1 (fr) 1998-08-17 1999-08-13 Medicaments preventifs/curatifs pour le glaucome

Publications (1)

Publication Number Publication Date
HK1030883A1 true HK1030883A1 (en) 2001-05-25

Family

ID=26459997

Family Applications (3)

Application Number Title Priority Date Filing Date
HK01101779A HK1030883A1 (en) 1998-08-17 2001-03-12 Preventives/remedies for glaucoma
HK05102430.9A HK1069120A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of glaucoma
HK05102431.8A HK1069121A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of asthenopia and pseudomyopia

Family Applications After (2)

Application Number Title Priority Date Filing Date
HK05102430.9A HK1069120A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of glaucoma
HK05102431.8A HK1069121A1 (en) 1998-08-17 2001-03-12 Agent for prophylaxis and treatment of asthenopia and pseudomyopia

Country Status (12)

Country Link
US (2) US6673812B1 (ja)
EP (3) EP1459743B9 (ja)
JP (2) JP3720264B2 (ja)
KR (1) KR100616466B1 (ja)
CN (2) CN1293878C (ja)
AT (3) ATE527993T1 (ja)
AU (1) AU5198199A (ja)
CA (2) CA2307285C (ja)
DE (1) DE69927936T2 (ja)
ES (3) ES2247822T3 (ja)
HK (3) HK1030883A1 (ja)
WO (1) WO2000009162A1 (ja)

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Also Published As

Publication number Publication date
DE69927936T2 (de) 2006-06-29
ES2372572T3 (es) 2012-01-23
EP1034793A1 (en) 2000-09-13
CN1494903A (zh) 2004-05-12
WO2000009162A1 (fr) 2000-02-24
EP1459743B1 (en) 2011-10-19
EP1459743A2 (en) 2004-09-22
EP1459742B1 (en) 2011-10-12
AU5198199A (en) 2000-03-06
EP1459742A3 (en) 2007-12-26
US20030125351A1 (en) 2003-07-03
JP3720264B2 (ja) 2005-11-24
KR20010015761A (ko) 2001-02-26
CN1195547C (zh) 2005-04-06
JP4490748B2 (ja) 2010-06-30
US6649625B2 (en) 2003-11-18
EP1034793B1 (en) 2005-10-26
ES2374518T3 (es) 2012-02-17
EP1459742B9 (en) 2012-05-02
EP1459743A8 (en) 2005-02-02
US6673812B1 (en) 2004-01-06
EP1459743B9 (en) 2012-08-01
CN1287494A (zh) 2001-03-14
ATE529102T1 (de) 2011-11-15
CA2307285A1 (en) 2000-02-24
KR100616466B1 (ko) 2006-08-29
HK1069121A1 (en) 2005-05-13
HK1069120A1 (en) 2005-05-13
ATE307609T1 (de) 2005-11-15
JP2004277432A (ja) 2004-10-07
CN1293878C (zh) 2007-01-10
EP1459742A2 (en) 2004-09-22
EP1459743A3 (en) 2007-12-26
CA2635412C (en) 2011-06-21
EP1034793A4 (en) 2003-07-09
DE69927936D1 (de) 2005-12-01
CA2307285C (en) 2009-03-31
ES2247822T3 (es) 2006-03-01
CA2635412A1 (en) 2000-02-24
ATE527993T1 (de) 2011-10-15

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