GEP20043385B - Pyrimidine Carboxamides Useful as Inhibitors of PDE4 Isozymes, Pharmaceutical Compositions Containing the Same - Google Patents

Pyrimidine Carboxamides Useful as Inhibitors of PDE4 Isozymes, Pharmaceutical Compositions Containing the Same

Info

Publication number
GEP20043385B
GEP20043385B GE4896A GEAP2001004896A GEP20043385B GE P20043385 B GEP20043385 B GE P20043385B GE 4896 A GE4896 A GE 4896A GE AP2001004896 A GEAP2001004896 A GE AP2001004896A GE P20043385 B GEP20043385 B GE P20043385B
Authority
GE
Georgia
Prior art keywords
inhibitors
pharmaceutical compositions
same
compositions containing
chronic
Prior art date
Application number
GE4896A
Other languages
English (en)
Inventor
Robert James Chambers
Thomas Victor Magee
Anthony Marfat
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of GEP20043385B publication Critical patent/GEP20043385B/en

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Diabetes (AREA)
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  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
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  • Neurology (AREA)
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  • Urology & Nephrology (AREA)
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  • Ophthalmology & Optometry (AREA)
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GE4896A 2000-01-31 2001-01-30 Pyrimidine Carboxamides Useful as Inhibitors of PDE4 Isozymes, Pharmaceutical Compositions Containing the Same GEP20043385B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31

Publications (1)

Publication Number Publication Date
GEP20043385B true GEP20043385B (en) 2004-04-13

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GE4896A GEP20043385B (en) 2000-01-31 2001-01-30 Pyrimidine Carboxamides Useful as Inhibitors of PDE4 Isozymes, Pharmaceutical Compositions Containing the Same

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US (1) US6740655B2 (Direct)
EP (1) EP1252157B1 (Direct)
JP (1) JP2003522165A (Direct)
KR (1) KR20020071029A (Direct)
CN (1) CN1404480A (Direct)
AP (1) AP2002002590A0 (Direct)
AR (1) AR027336A1 (Direct)
AT (1) ATE269860T1 (Direct)
AU (1) AU2700301A (Direct)
BG (1) BG106868A (Direct)
BR (1) BR0107934A (Direct)
CA (1) CA2396458C (Direct)
CO (1) CO5271669A1 (Direct)
CR (1) CR6714A (Direct)
CZ (1) CZ20022413A3 (Direct)
DE (1) DE60103976T2 (Direct)
DK (1) DK1252157T3 (Direct)
DZ (1) DZ3406A1 (Direct)
EA (1) EA005028B1 (Direct)
EE (1) EE200200426A (Direct)
ES (1) ES2223772T3 (Direct)
GE (1) GEP20043385B (Direct)
GT (1) GT200100023A (Direct)
HK (1) HK1054232A1 (Direct)
HN (1) HN2001000018A (Direct)
HU (1) HUP0204271A3 (Direct)
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PE (1) PE20011059A1 (Direct)
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SV (1) SV2001000298A (Direct)
TN (1) TNSN01019A1 (Direct)
TR (1) TR200402292T4 (Direct)
UY (1) UY26570A1 (Direct)
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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
WO2001047493A1 (en) * 1999-12-24 2001-07-05 Glaxo Group Limited Pharmaceutical aerosol formulation of salmeterol and fluticasone propionate
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
YU39503A (sh) * 2000-11-22 2006-05-25 F. Hoffmann-La Roche Ag. Derivati pirimidina
CA2436551A1 (en) 2001-01-31 2002-08-08 Pfizer Products Inc. Thiazolyl-, oxazolyl-, pyrrolyl-, and imidazolyl-acid amide derivatives useful as inhibitors of pde4 isozymes
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