FI962464A0 - Kristallina N-acetylneuraminsyraderivat och förfarande för framställning av dem - Google Patents

Kristallina N-acetylneuraminsyraderivat och förfarande för framställning av dem

Info

Publication number
FI962464A0
FI962464A0 FI962464A FI962464A FI962464A0 FI 962464 A0 FI962464 A0 FI 962464A0 FI 962464 A FI962464 A FI 962464A FI 962464 A FI962464 A FI 962464A FI 962464 A0 FI962464 A0 FI 962464A0
Authority
FI
Finland
Prior art keywords
crystalline
preparation
methods
acid derivatives
acetylamino acid
Prior art date
Application number
FI962464A
Other languages
English (en)
Finnish (fi)
Other versions
FI962464A (sv
FI120453B (sv
Inventor
Christopher Williamson
William James White
Vipulkumar Pater
Original Assignee
Biota Scient Management
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Management filed Critical Biota Scient Management
Publication of FI962464A publication Critical patent/FI962464A/sv
Publication of FI962464A0 publication Critical patent/FI962464A0/sv
Application granted granted Critical
Publication of FI120453B publication Critical patent/FI120453B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI962464A 1993-12-17 1996-06-13 Förfarande för framställning av kristallina N-acetylneuraminsyraderivat FI120453B (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB939325841A GB9325841D0 (en) 1993-12-17 1993-12-17 Chemical compounds
GB9325841 1993-12-17
PCT/EP1994/004154 WO1995016680A1 (en) 1993-12-17 1994-12-15 Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation
EP9404154 1994-12-15

Publications (3)

Publication Number Publication Date
FI962464A FI962464A (sv) 1996-06-13
FI962464A0 true FI962464A0 (sv) 1996-06-13
FI120453B FI120453B (sv) 2009-10-30

Family

ID=10746778

Family Applications (1)

Application Number Title Priority Date Filing Date
FI962464A FI120453B (sv) 1993-12-17 1996-06-13 Förfarande för framställning av kristallina N-acetylneuraminsyraderivat

Country Status (44)

Country Link
US (2) US6294572B1 (sv)
EP (1) EP0734382B1 (sv)
JP (1) JP3317972B2 (sv)
KR (1) KR100403256B1 (sv)
CN (2) CN1502621A (sv)
AP (2) AP9600810A0 (sv)
AT (1) ATE199255T1 (sv)
BG (1) BG63338B1 (sv)
BR (2) BR9408340A (sv)
CA (1) CA2177990C (sv)
CO (1) CO4340619A1 (sv)
CZ (1) CZ289234B6 (sv)
DE (1) DE69426726T2 (sv)
DK (1) DK0734382T3 (sv)
EE (1) EE03353B1 (sv)
EG (1) EG20597A (sv)
ES (1) ES2155517T3 (sv)
FI (1) FI120453B (sv)
GB (1) GB9325841D0 (sv)
GR (1) GR3035681T3 (sv)
HK (1) HK1014187A1 (sv)
HR (1) HRP941001B1 (sv)
HU (1) HU221971B1 (sv)
IL (1) IL112011A (sv)
IS (1) IS4240A (sv)
MA (1) MA23396A1 (sv)
MY (1) MY116221A (sv)
NO (1) NO314759B1 (sv)
NZ (1) NZ277789A (sv)
OA (2) OA10325A (sv)
PE (1) PE31095A1 (sv)
PL (1) PL186384B1 (sv)
PT (1) PT734382E (sv)
RO (1) RO114792B1 (sv)
RU (1) RU2134690C1 (sv)
SA (1) SA94150417B1 (sv)
SG (1) SG46669A1 (sv)
SI (1) SI0734382T1 (sv)
SK (1) SK282972B6 (sv)
SV (1) SV1994000076A (sv)
TW (1) TW452577B (sv)
UA (1) UA46723C2 (sv)
WO (1) WO1995016680A1 (sv)
ZA (1) ZA9410003B (sv)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9325841D0 (en) * 1993-12-17 1994-02-23 Glaxo Group Ltd Chemical compounds
BR9607098A (pt) 1995-02-27 1997-11-04 Gilead Sciences Inc Novos inibidores seletivos de neuraminidas virais ou bacterianas
US5866601A (en) * 1995-02-27 1999-02-02 Gilead Sciences, Inc. Carbocyclic compounds
US5763483A (en) * 1995-12-29 1998-06-09 Gilead Sciences, Inc. Carbocyclic compounds
US6340702B1 (en) 1996-07-22 2002-01-22 Sankyo Company, Limited Neuraminic acid derivatives, their preparation and their medical use
US6451766B1 (en) 1996-07-22 2002-09-17 Sankyo Company, Limited Neuraminic acid derivatives, their preparation and their medical use
PT823428E (pt) * 1996-07-22 2002-04-29 Sankyo Co Derivados do acido neuraminico sua preparacao e sua utilizacao em medicina
US5859284A (en) * 1996-08-23 1999-01-12 Gilead Sciences, Inc. Preparation of carbocyclic compounds
US6518438B2 (en) 1996-08-23 2003-02-11 Gilead Sciences, Inc. Preparation of cyclohexene carboxylate derivatives
US5994377A (en) * 1996-10-21 1999-11-30 Gilead Sciences, Inc. Piperidine compounds
US5886213A (en) * 1997-08-22 1999-03-23 Gilead Sciences, Inc. Preparation of carbocyclic compounds
TW480247B (en) * 1997-12-12 2002-03-21 Gilead Sciences Inc Novel compounds useful as neuraminidase inhibitors and pharmaceutical compositions containing same
TWI291462B (en) * 2000-04-25 2007-12-21 Daiichi Sankyo Co Ltd Hydrate crystal of neuraminic acid compound
US20080063722A1 (en) * 2006-09-08 2008-03-13 Advanced Inhalation Research, Inc. Composition of a Spray-Dried Powder for Pulmonary Delivery of a Long Acting Neuraminidase Inhibitor (LANI)
BR112014014635A2 (pt) * 2011-12-16 2017-06-13 Daiichi Sankyo Co Ltd método para fabricar um composto, e, composto
CN109232677B (zh) * 2018-10-18 2021-12-28 中国科学院合肥物质科学研究院 一种使n-乙酰神经氨酸水合物转化为n-乙酰神经氨酸的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK282950B6 (sk) * 1990-04-24 2003-01-09 Biota Scientific Management Pty Ltd Deriváty alfa-D-neuramínovej kyseliny, spôsob ich prípravy, ich použitie a farmaceutické prípravky na ich báze
CA2081068C (en) * 1991-10-23 2005-11-29 Laurence Mark Von Itzstein Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of .alpha.-d-neuraminic acid
US5639786A (en) 1992-12-04 1997-06-17 Biota Scientific Management, Pty., Ltd. Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of α-D-neuraninic acid
GB9325841D0 (en) * 1993-12-17 1994-02-23 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
GB9325841D0 (en) 1994-02-23
IL112011A (en) 1998-08-16
NZ277789A (en) 1999-04-29
ZA9410003B (en) 1995-07-25
AU689185B2 (en) 1998-03-26
MY116221A (en) 2003-12-31
HU221971B1 (hu) 2003-03-28
NO962545L (no) 1996-06-14
RO114792B1 (ro) 1999-07-30
AP9400705A0 (en) 1995-01-31
HU9601642D0 (en) 1996-08-28
JPH09506601A (ja) 1997-06-30
KR100403256B1 (ko) 2004-04-30
SA94150417B1 (ar) 2005-12-18
HRP941001B1 (en) 2001-06-30
CA2177990A1 (en) 1995-06-22
WO1995016680A1 (en) 1995-06-22
CN1132829C (zh) 2003-12-31
AU1314495A (en) 1995-07-03
US6294572B1 (en) 2001-09-25
PT734382E (pt) 2001-06-29
SV1994000076A (es) 1995-10-26
ES2155517T3 (es) 2001-05-16
EP0734382B1 (en) 2001-02-21
BR9408340A (pt) 1997-08-19
MA23396A1 (fr) 1995-07-01
FI962464A (sv) 1996-06-13
SG46669A1 (en) 1998-02-20
CZ289234B6 (cs) 2001-12-12
PE31095A1 (es) 1995-10-18
CO4340619A1 (es) 1996-07-30
IS4240A (is) 1995-06-18
OA11275A (en) 2002-11-20
EP0734382A1 (en) 1996-10-02
CN1142820A (zh) 1997-02-12
BR1100548KB1 (pt) 2011-11-01
ATE199255T1 (de) 2001-03-15
PL186384B1 (pl) 2004-01-30
JP3317972B2 (ja) 2002-08-26
US20020037865A1 (en) 2002-03-28
CZ169396A3 (en) 1996-11-13
HK1014187A1 (en) 1999-09-24
NO314759B1 (no) 2003-05-19
HRP941001A2 (en) 1997-06-30
DE69426726D1 (de) 2001-03-29
BG100709A (bg) 1997-01-31
GR3035681T3 (en) 2001-06-29
DE69426726T2 (de) 2001-06-21
NO962545D0 (no) 1996-06-14
SK78596A3 (en) 1997-03-05
SK282972B6 (sk) 2003-01-09
UA46723C2 (uk) 2002-06-17
BG63338B1 (bg) 2001-10-31
DK0734382T3 (da) 2001-03-19
AP9600810A0 (en) 1996-07-31
TW452577B (en) 2001-09-01
CN1502621A (zh) 2004-06-09
SI0734382T1 (en) 2001-08-31
OA10325A (en) 1997-10-07
AP541A (en) 1996-10-01
FI120453B (sv) 2009-10-30
PL315055A1 (en) 1996-09-30
EG20597A (en) 1999-09-30
HUT74938A (en) 1997-03-28
CA2177990C (en) 2000-04-25
IL112011A0 (en) 1995-03-15
RU2134690C1 (ru) 1999-08-20
EE03353B1 (et) 2001-02-15

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