FI69461C - Analogifoerfarande foer framstaellning av nya saosom laekemedelsaktivaemnen anvaendbara bensotiofen-2-on-3-karboxamider - Google Patents

Analogifoerfarande foer framstaellning av nya saosom laekemedelsaktivaemnen anvaendbara bensotiofen-2-on-3-karboxamider Download PDF

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Publication number
FI69461C
FI69461C FI771044A FI771044A FI69461C FI 69461 C FI69461 C FI 69461C FI 771044 A FI771044 A FI 771044A FI 771044 A FI771044 A FI 771044A FI 69461 C FI69461 C FI 69461C
Authority
FI
Finland
Prior art keywords
benzo
oxo
formula
dihydro
compound
Prior art date
Application number
FI771044A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI771044A (da
FI69461B (fi
Inventor
Raymond Bernasconi
Pier Giorgio Ferrini
Richard Goeschke
Jacques Gosteli
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH453876A external-priority patent/CH630082A5/de
Priority claimed from CH1599476A external-priority patent/CH629797A5/de
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of FI771044A publication Critical patent/FI771044A/fi
Publication of FI69461B publication Critical patent/FI69461B/fi
Application granted granted Critical
Publication of FI69461C publication Critical patent/FI69461C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/64—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D333/70—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI771044A 1976-04-09 1977-04-04 Analogifoerfarande foer framstaellning av nya saosom laekemedelsaktivaemnen anvaendbara bensotiofen-2-on-3-karboxamider FI69461C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH453876 1976-04-09
CH453876A CH630082A5 (de) 1976-04-09 1976-04-09 Verfahren zur herstellung von oxothiaverbindungen.
CH1599476A CH629797A5 (en) 1976-12-20 1976-12-20 Process for the preparation of salts of oxothia compounds
CH1599476 1976-12-20

Publications (3)

Publication Number Publication Date
FI771044A FI771044A (da) 1977-10-10
FI69461B FI69461B (fi) 1985-10-31
FI69461C true FI69461C (fi) 1986-02-10

Family

ID=25695718

Family Applications (1)

Application Number Title Priority Date Filing Date
FI771044A FI69461C (fi) 1976-04-09 1977-04-04 Analogifoerfarande foer framstaellning av nya saosom laekemedelsaktivaemnen anvaendbara bensotiofen-2-on-3-karboxamider

Country Status (27)

Country Link
US (1) US4320138A (da)
JP (1) JPS52125158A (da)
AR (3) AR218869A1 (da)
AT (1) AT357148B (da)
CA (1) CA1112248A (da)
CS (4) CS207394B2 (da)
CY (1) CY1138A (da)
DD (1) DD130659A5 (da)
DE (1) DE2713584C2 (da)
DK (1) DK152046C (da)
ES (1) ES457528A1 (da)
FI (1) FI69461C (da)
FR (1) FR2347363A1 (da)
GB (1) GB1544339A (da)
GR (1) GR70652B (da)
HK (1) HK6182A (da)
HU (1) HU180438B (da)
IE (1) IE44987B1 (da)
IL (1) IL51847A (da)
KE (1) KE3185A (da)
MY (1) MY8200244A (da)
NL (1) NL7703802A (da)
NO (1) NO146810C (da)
NZ (1) NZ183747A (da)
PL (3) PL110653B1 (da)
SE (1) SE432930B (da)
SU (4) SU795475A3 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH634840A5 (de) * 1978-06-29 1983-02-28 Ciba Geigy Ag 2-oxo-2,3-dihydro-benzo(b)thiophen-verbindung und daraus hergestellte pharmazeutische praeparate.
AT392787B (de) * 1978-06-29 1991-06-10 Ciba Geigy Ag Verfahren zur herstellung des neuen n-(2-thienyl)-2-oxo-2,3-dihydro-benzo(b)thiophen-3-carboxamids

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3413308A (en) * 1966-09-02 1968-11-26 Dow Chemical Co Substituted benzo(b)thiophene-2-carboxanilides
US3655693A (en) * 1969-06-25 1972-04-11 Merck & Co Inc Anti-inflammatory salicyclic acid derivatives
US3676463A (en) * 1970-10-15 1972-07-11 Pfizer Oxobenzofuran carboxamides
US3971814A (en) * 1972-11-27 1976-07-27 Warner-Lambert Company Benzo(b)thiophene derivatives
GB1571847A (en) * 1974-01-02 1980-07-23 Systems Eng & Mfg Waste water treatment

Also Published As

Publication number Publication date
CS207395B2 (en) 1981-07-31
HU180438B (en) 1983-03-28
AT357148B (de) 1980-06-25
PL197311A1 (pl) 1978-01-16
CS207393B2 (en) 1981-07-31
MY8200244A (en) 1982-12-31
DD130659A5 (de) 1978-04-19
NZ183747A (en) 1979-01-11
FR2347363A1 (fr) 1977-11-04
NO771231L (no) 1977-10-11
NO146810B (no) 1982-09-06
SE7704033L (sv) 1977-10-10
DK152046C (da) 1988-07-18
JPS52125158A (en) 1977-10-20
FI771044A (da) 1977-10-10
CS207394B2 (en) 1981-07-31
HK6182A (en) 1982-02-19
JPS6218556B2 (da) 1987-04-23
ATA248577A (de) 1979-11-15
FI69461B (fi) 1985-10-31
SE432930B (sv) 1984-04-30
IL51847A0 (en) 1977-06-30
IL51847A (en) 1981-09-13
DE2713584A1 (de) 1977-10-20
SU791239A3 (ru) 1980-12-23
CS207392B2 (en) 1981-07-31
FR2347363B1 (da) 1979-03-09
KE3185A (en) 1982-04-02
SU898956A3 (ru) 1982-01-15
DK152046B (da) 1988-01-25
CY1138A (en) 1982-05-07
NO146810C (no) 1982-12-15
GB1544339A (en) 1979-04-19
NL7703802A (nl) 1977-10-11
AR224614A1 (es) 1981-12-30
ES457528A1 (es) 1978-08-16
IE44987L (en) 1977-10-09
PL110653B1 (en) 1980-07-31
PL111456B1 (en) 1980-08-30
SU795475A3 (ru) 1981-01-07
US4320138A (en) 1982-03-16
DK158777A (da) 1977-10-10
PL111459B1 (en) 1980-08-30
DE2713584C2 (de) 1986-09-04
GR70652B (da) 1982-12-03
IE44987B1 (en) 1982-06-02
SU738510A3 (ru) 1980-05-30
CA1112248A (en) 1981-11-10
AR225401A1 (es) 1982-03-31
AR218869A1 (es) 1980-07-15

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MM Patent lapsed

Owner name: CIBA-GEIGY AG